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Histamine Receptor

Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
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Cat. No. Product Name CAS No. Purity Chemical Structure
T16476 PF-03654746
化合物PF-03654746
935840-31-6 99.1%
PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。
TN3699 Corchoionoside C
化合物 TN3699
185414-25-9 98%
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
T10770 Cetirizine D8
化合物 T10770
774596-22-4 98%
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T77715 H4R antagonist 3
H4R拮抗剂3
1003091-20-0 98%
H4R antagonist 3 是一种新型组胺-4受体 (H4R)拮抗剂,EC50 <10 mM。H4R antagonist 3 具有潜在的炎性活性,可用于研究自身免疫性、过敏性和眼部疾病。
T78126 Dothiepin
度硫平
113-53-1 98%
Dothiepin(Dosulepin; Dothep)是一种具备镇静/抗焦虑作用的抗抑郁药物。该化合物主要通过抑制去甲肾上腺素的再摄取,而非血清素,以增强去肾上腺素能神经传递。同时,Dothiepin作为组胺H1受体的拮抗剂,具备显著的镇痛活性,适用于治疗心因性面部疼痛、特发性纤维肌痛综合征或类风湿关节炎,并且不具有心...
T79786 H4R antagonist 2
化合物 H4R antagonist 2
1148115-99-4 98%
H4R antagonist 2 是Furo[3,2-d]嘧啶衍生的有效H4R拮抗剂,主要用于类风湿性关节炎的研究。
T80645 4-Methylhistamine
化合物 4-Methylhistamine
36507-31-0 98%
4-Methylhistamine 作为一种有效的组胺 4 受体 (H4R) 激动剂,显示出在研究免疫相关疾病,如癌症和自身免疫性疾病方面的应用潜力。
T11729 JTE-952
化合物 T11729
1255303-54-8 98%
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
T15590 Iodophenpropit dihydrobromide
化合物 T15590
145196-87-8 98%
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
TN3483 Bakkenolide D
化合物 TN3483
18456-03-6 98%
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
T12630 (R)-(-)-α-Methylhistamine dihydrobromide
(R)(−)-α-甲基组胺 二盐酸盐
868698-49-1 98%
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
TN2155 Rhodiocyanoside A
化合物Rhodiocyanoside A
168433-86-1 98%
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
T11088 Doxepin D3 Hydrochloride
化合物 T11088
347840-07-7 98%
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
T15722 Lavoltidine
化合物 T15722
76956-02-0 98%
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
T17118 Toreforant
化合物 T17118
952494-46-1 98%
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
T12416 PF-03654746 Tosylate
化合物 T12416
1039399-17-1 98%
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
T12703 ReN-1869 hydrochloride
化合物 T12703
170149-76-5 98%
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
T19443L N-Acetylhistamine acetate
化合物N-Acetylhistamine acetate
98%
N-Acetylhistamine acetate 是一种组胺代谢物。 它可用作过敏反应的组氨酸代谢的潜在生物标志物。
T2S0118 Daurinoline
蝙蝠葛诺林碱
2831-75-6 98%
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
T12228 Niperotidine
尼培替丁
84845-75-0 98%
Niperotidine is an antagonist of histamine H2-receptor.
PF-03654746
T16476
PF-03654746 是组胺 H3 受体的选择性拮抗剂。 PF-03654746 提高了阿尔茨海默病的认知功效和疾病改善作用。 PF-03654746 可用于治疗过敏性鼻炎的研究。
Corchoionoside C
TN3699
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ...
Cetirizine D8
T10770
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
H4R antagonist 3
T77715
H4R antagonist 3 是一种新型组胺-4受体 (H4R)拮抗剂,EC50 <10 mM。H4R antagonist 3 具有潜在的炎性活性,可用于研究自身免疫性、过敏性和眼部疾病。
Dothiepin
T78126
Dothiepin(Dosulepin; Dothep)是一种具备镇静/抗焦虑作用的抗抑郁药物。该化合物主要通过抑制去甲肾上腺素的再摄取,而非血清素,以增强去肾上腺素能神经传递。同时,Dothiepin作为组胺H1受体的拮抗剂,具备显著的镇痛活性,适用于治疗心因性面部疼痛、特发性纤维肌痛综合征或类风湿关节炎,并且不具有心...
H4R antagonist 2
T79786
H4R antagonist 2 是Furo[3,2-d]嘧啶衍生的有效H4R拮抗剂,主要用于类风湿性关节炎的研究。
4-Methylhistamine
T80645
4-Methylhistamine 作为一种有效的组胺 4 受体 (H4R) 激动剂,显示出在研究免疫相关疾病,如癌症和自身免疫性疾病方面的应用潜力。
JTE-952
T11729
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit...
Iodophenpropit dihydrobromide
T15590
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s...
Bakkenolide D
TN3483
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o...
(R)-(-)-α-Methylhistamine dihydrobromide
T12630
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
Rhodiocyanoside A
TN2155
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ...
Doxepin D3 Hydrochloride
T11088
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin...
Lavoltidine
T15722
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg...
Toreforant
T17118
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
PF-03654746 Tosylate
T12416
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
ReN-1869 hydrochloride
T12703
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
N-Acetylhistamine acetate
T19443L
N-Acetylhistamine acetate 是一种组胺代谢物。 它可用作过敏反应的组氨酸代谢的潜在生物标志物。
Daurinoline
T2S0118
Daurinoline is a non-competitive antagonist, it exerts marked relaxation effect on basilar artery of rabbits through non-competitive antagonism, it would have a ...
Niperotidine
T12228
Niperotidine is an antagonist of histamine H2-receptor.
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