Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
TN5192 | Tuberosin
化合物 TN5192
|
41347-45-9 | 98% |
|
Tuberosin shows anti-inflammatory and antioxidant activities.It demonstrated a significantly potent inhibition on yeast α-glucosidase in a dose dependent manner.... | ||||
TN5090 | Tachioside
化合物 TN5090
|
109194-60-7 | 98% |
|
Tachioside has antiobesity, antioxidant and α-glucosidase inhibitory activities, it decreases lipid content in 3T3-L1 adipocytes by inhibiting lipogenesis, shows... | ||||
TN4793 | Pinoresinol diacetate
化合物 TN4793
|
32971-25-8 | 98% |
|
Pinoresinol diacetate inhibits the enzyme α-glucosidase in vitro and may therefore act as a hypoglycemic agent. | ||||
T10751 | Cefetrizole
头孢三唑
|
65307-12-2 | 98% |
|
Ceftezole is an α-Glucosidase inhibitor (IC50: 2.1 μM; Ki: 0.578 μM). | ||||
TN5094 | Tangshenoside I
党参苷 I
|
117278-74-7 | 98% |
|
Tangshenoside I might be a potential bioactive marker related to the hematopoietic and immunologic functions of Codonopsis Radix, which could be recommended as t... | ||||
TN3745 | Cyclomusalenone
化合物 TN3745
|
30452-60-9 | 98% |
|
Cyclomusalenone is a potent α-glucosidase inhibitor. | ||||
T11749 | KDM4-IN-2
化合物 T11749
|
2369607-62-3 | 98% |
|
KDM4-IN-2 is a potent and selective KDM4/KDM5 dual inhibitor with Kis of 4 and 7 nM for KDM4A and KDM5B, respectively. | ||||
TN4174 | Guajadial
化合物 TN4174
|
959860-49-2 | 98% |
|
Guajadial shows α-glucosidase inhibitory activities significantly and its activity was better than that of Acarbose.Guajadial may act as Selective Estrogen Recep... | ||||
T16480 | PF-04991532
化合物 T16480
|
1215197-37-7 | 98% |
|
PF-04991532 is an effective, hepatoselective glucokinase activator. It has EC50s of 80 and 100 nM in human and rat, respectively. | ||||
T6759 | AP-III-a4
化合物AP-III-a4
|
1177827-73-4 | 99.90% |
|
AP-III-a4 (ENOblock) 是第一个非底物类似物,可直接与烯醇酶结合,IC50=0.576 uM,可阻碍体内癌细胞转移。 | ||||
T36491 | POMHEX
化合物POMHEX
|
2004714-34-3 | 99.88% |
|
Pomhex 是一种具有抗癌活性的细胞渗透性强效烯醇化酶抑制剂,可用于癌症致死率的研究。Pomhex是一种外消旋混合物,是一种强效且具有选择性的ENO2抑制剂。 | ||||
T11741 | KAN0438757
化合物KAN0438757
|
1451255-59-6 | 99.8% |
|
KAN0438757 是一种选择性强效的代谢激酶 PFKFB3 抑制剂,IC50值为 0.19 μM。 | ||||
T64320 | ML251
化合物ML251
|
1486482-16-9 | 99.79% |
|
ML251 是一种有效的新型纳摩尔 T. brucei 和 T. cruzi 磷酸果糖激酶抑制剂,对 T. brucei PFK 和 T. cruzi PFK 的 IC50值为 0.37和 0.13 μM,可研究寄生虫。 | ||||
T15159 | Dorzagliatin
化合物Dorzagliatin
|
1191995-00-2 | 99.74% |
|
Dorzagliatin (HMS5552) 是双重作用的葡萄糖激酶 (glucokinase;GK) 激活剂,可改善 2 型糖尿病的血糖控制,提高胰腺 β 细胞功能。 | ||||
T22223 | 3PO
化合物3PO
|
18550-98-6 | 99.67% |
|
3PO 是一种 PFKFB3 的小分子抑制剂,IC50值为22.9 μM。它抑制几种人类恶性造血和腺癌细胞系的增殖,IC50在1.4到24 μM 之间。它抑制葡萄糖摄取,并降低 Fru-2,6-BP、乳酸、ATP、NAD+ 和 NADH 的细胞内浓度。 | ||||
T3312 | AM-2394
化合物AM2394
|
1442684-77-6 | 99.58% |
|
AM-2394 是新型的 glucokinase 激活剂 (GKA)。它能够激活葡萄糖激酶 (GK),EC50=60 nM。 | ||||
T3386 | Kaempferitrin
山奈苷
|
482-38-2 | 99.51% |
|
Kaempferitrin (Lespenephryl) 是天然黄酮苷类化合物,具有缓解疼痛、抗糖尿病、消炎、抗肿瘤和化疗作用,可激活胰岛素信号传导。 | ||||
T3104 | Globalagliatin
化合物LY2608204
|
1234703-40-2 | 99.41% |
|
Globalagliatin (LY2608204) 是一种葡萄糖激酶 (GK) 活化剂,EC50=42 nM。 | ||||
T26712 | AZD-1656
化合物AZD-1656
|
919783-22-5 | 99.37% |
|
AZD-1656 是口服有效的葡萄糖激酶选择性激活剂,EC50为 60 nM。AZD1656在2 型糖尿病中有研究的价值。 | ||||
T19500 | Palmitelaidic Acid
软脂酸
|
10030-73-6 | 99.36% |
|
trans-Palmitelaidic Acid (trans-Palmitoleic acid) 是palmitoleic acid 的反式异构体。Palmitoleic acid 是血清和组织中最丰富的脂肪酸之一。 |