目录号 | 产品详情 | 靶点 | |
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T23682 | |||
AHR-16303B oxalate is a novel antagonist of 5-HT2 receptors. | |||
T10271 | Others | ||
AHR antagonist 4 is a potent aryl hydrocarbon receptor (AHR) antagonist(example 293; IC50: 82.2 nM).It has anti-cancer effects. | |||
T1409 | Sodium Channel Carbonic Anhydrase | ||
Methocarbamol (AHR 85) 是口服有效的中枢肌肉松弛剂,可阻断肌肉Nav1.4通道,阻断作用具有可逆性。Methocarbamol 具有用于肌肉痉挛和疼痛综合症研究的潜力。 | |||
T20986 | |||
AHR agonist 3 is an agent with therapeutic activity. | |||
T29750L | |||
AHR-1900 free base is a butyrophenone derivative which may be used in the treatment of schizophrenia. | |||
T1610 | Others | ||
Metaxalone (Methaxalonum) 具有肌肉松弛作用。 | |||
T10272 | Others | ||
AHR antagonist 5 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist(example 39; IC50 < 0.5 μΜ). It significantly inhibits tumor growth combined with checkpoint inhibitor anti-PD-1. | |||
T71590 | |||
AHR-5645B fumarate is a substituted benzamide that has been shown to inhibit 3H-spiperone binding to bovine anterior pituitary membranes. | |||
T7202 | AhR Aryl Hydrocarbon Receptor | ||
ITE 是一种有效的芳烃受体 (AhR) 内源性激动剂,Ki 值为 3 nM。它具有免疫抑制作用。 | |||
T21966 | GSK-3 Aryl Hydrocarbon Receptor CDK | ||
MeBIO 是一种芳烃受体激动剂,对 GSK-3 和 CDK1/CyclinB 的 IC50 分别为 44 和 55 μM。 MeBIO 不影响 GSK-3β。 |
目录号 | 产品名/同用名 | 种属 | 表达系统 | ||
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TMPH-00958 | AHR Protein, Human, Recombinant (His) | Human | E. coli | ||
AHR Protein, Human, Recombinant (His) is expressed in E. coli.
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TMPJ-00423 | TIM-1/KIM-1/HAVCR1 Protein, Mouse, Recombinant (His) | Mouse | Human Cells | ||
TIM-1/KIM-1/HAVCR belongs to the immunoglobulin superfamily that cosisits 305 amino acid (aa). It is expressed by stimulated T-cells. TIM-1/KIM-1/HAVCR may play a role in T-helper cell development and the regulation of asthma and allergic diseases. Receptor for TIMD4. And may have a role in kidney injury and repair. Belongs to the T-cell and airway phenotype regulator (Tapr) locus, a single chromosomal region that confers reduced T-helper type 2 responsiveness and protects against airway hyperactivity (AHR), the hallmark of human asthma.
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