目录号 | 产品详情 | 靶点 | |
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T17364 | Others | ||
AhR Ligand-Linker Conjugates 1, also known as E3 Ligase Ligand-Linker Conjugates 57, is a chemical compound that combines an IAP ligand for the E3 ubiquitin ligase with a SNIPER linker. It is specifically designed to be used in the development of SNIPER[1]. | |||
T1960 | AhR Aryl Hydrocarbon Receptor | ||
YL-109是一种抗肿瘤剂,可以通过芳烃受体 AhR 信号传导诱导 Hsp70 相互作用蛋白 (CHIP) 表达,具有抑制乳腺癌细胞生长和侵袭性的能力。 | |||
TN1451 | AhR Aryl Hydrocarbon Receptor Glucosidase | ||
Brevifolincarboxylic acid 是从头状蓼中分离得到的一种天然产物,抑制芳烃受体(AhR)。它是一种 α-葡萄糖苷酶抑制剂,IC50 为 323.46 μM。 | |||
T23686 | |||
AHR-activator-1023 is the aryl hydrocarbon receptor activator. It is also a specific FGF2-induced branching morphogenesis modulator. | |||
T15410 | Aryl Hydrocarbon Receptor | ||
GNF351 是芳烃受体 (AhR) 的完全拮抗剂,具有抑制 DRE 依赖性和非依赖性活性的能力。它与结合到 AhR 的光亲和性 AhR 配体竞争,IC50为 62 nM。它在小鼠或人角质形成细胞中的毒性极小。 | |||
T4608 | AhR Aryl Hydrocarbon Receptor | ||
PDM2 是一种有效的选择性芳烃受体 (AhR) 拮抗剂,Ki 为 1.2±0.4 nM。 | |||
T10007 | AhR | ||
1,4-Chrysenequinone (Chrysene-1,4-dione) 是多环芳香烃类,是芳烃受体 (AhR) 的激活剂 | |||
T10270 | Aryl Hydrocarbon Receptor | ||
BAY 2416964 是一种可口服的芳基烃受体拮抗剂,IC50为 341 nM,可用于研究实体瘤。 | |||
T2448 | AhR Aryl Hydrocarbon Receptor | ||
CH-223191 是一种特异性有效的芳烃受体 (AhR) 拮抗剂,可抑制 TCDD 介导的核转位和 AhR 的 DNA 结合,抑制 TCDD 诱导的荧光素酶活性的 IC50值为 0.03 μM。 | |||
T6795 | Decarboxylase Aryl Hydrocarbon Receptor | ||
Carbidopa (Lodosyn) 是一种选择性芳香烃受体(AhR)调节剂,是外周型脱羧酶抑制剂,抑制胰腺癌细胞和肿瘤生长,可用于帕金森病的研究。 |
目录号 | 产品名/同用名 | 种属 | 表达系统 | ||
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TMPH-00958 | AHR Protein, Human, Recombinant (His) | Human | E. coli | ||
AHR Protein, Human, Recombinant (His) is expressed in E. coli.
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TMPJ-00423 | TIM-1/KIM-1/HAVCR1 Protein, Mouse, Recombinant (His) | Mouse | Human Cells | ||
TIM-1/KIM-1/HAVCR belongs to the immunoglobulin superfamily that cosisits 305 amino acid (aa). It is expressed by stimulated T-cells. TIM-1/KIM-1/HAVCR may play a role in T-helper cell development and the regulation of asthma and allergic diseases. Receptor for TIMD4. And may have a role in kidney injury and repair. Belongs to the T-cell and airway phenotype regulator (Tapr) locus, a single chromosomal region that confers reduced T-helper type 2 responsiveness and protects against airway hyperactivity (AHR), the hallmark of human asthma.
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