目录号 | 产品详情 | 靶点 | |
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T31398 | |||
Dexibuprofen (S-ibuprofen) is a non-steroidal anti-inflammatory drug. Most ibuprofen preparations contain a racemic mixture of two isomers. Dexibuprofen as a cyclooxygenase inhibitor. | |||
T41091 | |||
JTS-653 is a potent and selective in vitro and in vivo antagonist of transient receptor potential vanilloid 1 (TRPV1). It effectively attenuates chronic pain resistant to non-steroidal anti-inflammatory drugs. | |||
T12336 | Others | ||
Oxaprozin D4 is the deuterium labeled Oxaprozin, is a non-steroidal anti-inflammatory drug (NSAID). | |||
T27042 | |||
Clobenoside is a non-steroidal anti-inflammatory agent. Clobenoside also has an edema-protective effect while not influencing blood pressure nor heart rat and not producing any direct vasoactive effects. | |||
T61261 | |||
Isofezolac (LM 22070) is a non-steroidal anti-inflammatory drug (NSAID) known for its potent inhibition of prostaglandin-synthetase. This compound exhibits notable anti-inflammatory and antipyretic properties [1] [2]. | |||
T12047 | Others | ||
Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers. | |||
T11998 | Others | ||
Meloxicam D4 is deuterium labeled Meloxicam. Meloxicam is a non-steroidal antiinflammatory agent, inhibits COX activity,(Target:COX-1; IC50: 36.6 μM ;(Target:COX-2; IC50: 0.49 μM). | |||
T79864 | NOD-like Receptor (NLR) | ||
Usnoflast,作为一种NLRP3调节剂,同时也属于非甾体抗炎药(NSAD)类。 | |||
T67202 | |||
Benvitimod is a non-steroidal anti-inflammatory drug (NSAID) potentially for the treatment of atopic dermatitis. | |||
T11754 | PPAR | ||
Ketorolac D5, a deuterium-labeled version of Ketorolac, is a non-steroidal anti-inflammatory agent that functions as a nonselective COX inhibitor. It exhibits IC50 values of 20 nM for COX-1 and 120 nM for COX-2. |
目录号 | 产品名/同用名 | 种属 | 表达系统 | ||
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TMPH-01640 | MRGPRX2 Protein, Human, Recombinant (His) | Human | E. coli | ||
Mast cell-specific receptor for basic secretagogues, i.e. cationic amphiphilic drugs, as well as endo- or exogenous peptides, consisting of a basic head group and a hydrophobic core. Recognizes and binds small molecules containing a cyclized tetrahydroisoquinoline (THIQ), such as non-steroidal neuromuscular blocking drugs (NMBDs), including tubocurarine and atracurium. In response to these compounds, mediates pseudo-allergic reactions characterized by histamine release, inflammation and airway contraction. Acts as a receptor for a number of other ligands, including peptides and alkaloids, such as cortistatin-14, proadrenomedullin N-terminal peptides PAMP-12 and, at lower extent, PAMP-20, antibacterial protein LL-37, PMX-53 peptide, beta-defensins, and complanadine A.
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