目录号 | 产品详情 | 靶点 | |
---|---|---|---|
TMA0003 | cAMP Tyrosinase | ||
Trans-caffeic acid stearyl ester is posited to inhibit melanogenesis signaling while suppressing cAMP levels and, subsequently, MC1R, MITF, tyrosinase, TRP-2 and TRP-1 down-regulation, resulting in the suppression of tyrosinase activity, DOPA oxidase activity and melanin synthesis. | |||
T28035 | Others | ||
MHY908, a novel inhibitor of melanogenesis, potently inhibits mushroom tyrosinase activity in a dose-dependent manner. | |||
T71873 | Others | ||
Temechine hydrobromide is used for the identification of new diterpenoidal alkaloid leads as tyrosinase inhibitors. | |||
TN6605 | |||
4-Nitrocinnamic acid is a photosensitive compound. 4-Nitrocinnamic acid has inhibitory effects on tyrosinase. | |||
T70783 | Others | ||
Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor. | |||
T75613 | Others | ||
7-Methoxy obtusifolin (Compound 4) 是一种竞争性tyrosinase 抑制剂,IC50为 7.0 μM。 | |||
TN3372 | Others | ||
Alboctalol inhibits mushroom tyrosinase activity. | |||
T29898 | Others | ||
alpha-Methylcinnamaldehyde 是 Cinnamaldehyde 的α-取代衍生物,可被用作蘑菇酪氨酸酶的抑制剂。 | |||
TN2223 | IL Receptor NOS COX | ||
Soyacerebroside I demonstrates a potent tyrosinase inhibitory activity. | |||
TN6555 | |||
Safflospermidine A is a potential natural tyrosinase inhibitor,it shows high antityrosinase activity (IC50 of 13.8 μM). |
目录号 | 产品名/同用名 | 种属 | 表达系统 | ||
---|---|---|---|---|---|
TMPH-02270 | Tyrosinase/TYR Protein, Human, Recombinant (His & SUMO) | Human | E. coli | ||
This is a copper-containing oxidase that functions in the formation of pigments such as melanins and other polyphenolic compounds. Catalyzes the initial and rate limiting step in the cascade of reactions leading to melanin production from tyrosine. In addition to hydroxylating tyrosine to DOPA (3,4-dihydroxyphenylalanine), also catalyzes the oxidation of DOPA to DOPA-quinone, and possibly the oxidation of DHI (5,6-dihydroxyindole) to indole-5,6 quinone.
|
|||||
TMPH-02269 | Tyrosinase/TYR Protein, Human, Recombinant (His) | Human | P. pastoris (Yeast) | ||
This is a copper-containing oxidase that functions in the formation of pigments such as melanins and other polyphenolic compounds. Catalyzes the initial and rate limiting step in the cascade of reactions leading to melanin production from tyrosine. In addition to hydroxylating tyrosine to DOPA (3,4-dihydroxyphenylalanine), also catalyzes the oxidation of DOPA to DOPA-quinone, and possibly the oxidation of DHI (5,6-dihydroxyindole) to indole-5,6 quinone.
|
|||||
TMPH-00036 | Polyphenol oxidase 2 Protein, Agaricus bisporus, Recombinant (His & Myc) | Agaricus bisporus | E. coli | ||
Polyphenol oxidase 2 Protein, Agaricus bisporus, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 51.0 kDa and the accession number is O42713.
|
|||||
TMPH-00035 | Polyphenol oxidase 2 Protein, Agaricus bisporus, Recombinant (His) | Agaricus bisporus | Baculovirus Insect Cells | ||
Copper-containing oxidase that catalyzes both the o-hydroxylation of monophenols and the subsequent oxidation of the resulting o-diphenols into reactive o-quinones, which evolve spontaneously to produce intermediates, which associate in dark brown pigments. Involved in the initial step of melanin synthesis. Melanins constitute a mechanism of defense and resistance to stress such as UV radiations, free radicals, gamma rays, dehydratation and extreme temperatures, and contribute to the fungal cell-wall resistance against hydrolytic enzymes in avoiding cellular lysis. Fungal pigments are also involved in the formation and stability of spores.
|
|||||
TMPH-02751 | DCT Protein, Mouse, Recombinant (His & SUMO) | Mouse | E. coli | ||
Catalyzes the conversion of L-dopachrome into 5,6-dihydroxyindole-2-carboxylic acid (DHICA). DCT Protein, Mouse, Recombinant (His & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO tag. The predicted molecular weight is 69.7 kDa and the accession number is P29812.
|
|||||
TMPH-01608 | DCT Protein, Human, Recombinant (His & Myc & SUMO) | Human | E. coli | ||
Catalyzes the conversion of L-dopachrome into 5,6-dihydroxyindole-2-carboxylic acid (DHICA).
|