T39472
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NVP-CGM097 (stereoisomer) is a non-bioactive stereoisomer of NVP-CGM097, which is a potent and selective inhibitor of MDM2. |
T4171
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NMDAR
iGluR
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PEAQX (NVP-AAM077) 是 NR2A 高效选择性 NMDA 受体拮抗剂,IC50值为270nM。 |
T39858
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NVP-BSK805 trihydrochloride is a potent ATP-competitive inhibitor of JAK2, exhibiting IC50 values of 0.48 nM, 31.63 nM, 18.68 nM, and 10.76 nM against JAK2 JH1, JAK1 JH1, JAK3 JH1, and TYK2 JH1, respectively. |
T7418
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c-RET
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BBT594 (NVP-BBT594) 是受体酪氨酸激酶 RET 抑制剂,常用于研究癌症。 |
TQ0313
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PI3K
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NVP-BAG956 is an ATP-competitive PI3K inhibitor (IC50s: 34/56/112/444 nM for PI3Kδ/PI3Kα/PI3Kγ/PI3Kβ). |
T40292
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Ras
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Opnurasib (JDQ-443) 是一种可口服且具有选择性和有效性的共价 KRAS G12C 抑制剂,具有抗肿瘤活性,可用于研究晚期非小细胞肺癌。 |
T68740
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NVP-TAC544 is a novel focal adhesion kinase (FAK) inhibitor, potently blocking kinase activity of FAK along with Aurora A, activated Cdc42-associated kinase 1 (ACK1), Met, insulin receptor (IR), TrkA, and IGF-1R. |
T39481
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NVP-DPP728 dihydrochloride is a highly potent, selective, and orally active inhibitor of dipeptidyl peptidase IV (DPP-IV), with a binding affinity (K i ) of 11 nM. This compound proves useful for investigating diabetes mellitus in research studies. |
T11838
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Smo
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LEQ506 是一种 Smo 抑制剂,对 hSmo 和 mSmo 的 IC50 分别为 2 nM 和 4 nM。 |
T15727
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Smo
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Sonidegib diphosphate (LDE225 diphosphate) 是 Smo 的选择性拮抗剂,能够抑制鼠 Smo (IC50:1.3 nM)和人 Smo (IC50:2.5 nM)。 |