目录号 | 产品详情 | 靶点 | |
---|---|---|---|
T3455 | Discoidin Domain Receptor (DDR) FLT ROS ROS Kinase c-Met/HGFR | ||
Merestinib 是一种有效的口服生物可利用的具有抗肿瘤活性的c-Met 抑制剂。 | |||
T15808 | ROCK | ||
Merestinib dihydrochloride is an effective and orally bioavailable c-Met inhibitor (Ki=2 nM). It has anti-tumor activities and also has potent activity against MST1R (IC50=11 nM), FLT3 (IC50=7 nM), AXL (IC50=2 nM), MERTK (IC50=10 nM), TEK (IC50=63 nM), RO |