T69788
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Daledalin is an antidepressant which was synthesized and trialed for depression in the early 1970s, but was never marketed. It is a selective norepinephrine reuptake inhibitor, with no significant effects on the reuptake of serotonin and dopamine, and no antihistamine or anticholinergic properties. |
T71773
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Levomepromazine Maleate is a Tricyclic antidepressant (TCA), acting as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also having other activities including antihistamine, antiadrenergic, antiserotonergic, anticholinergic, and sodium channel-blocking effects. |
T71631
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Eucatropine,作为一种有效的毒蕈碱型乙酰胆碱受体(mAChR)抑制剂,具有0.583 μM的IC50值,归类为抗胆碱能剂。 |
T61309
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(R)-Oxybutynin (Aroxybutynin) is an orally active muscarinic receptor antagonist, which exhibits antimuscarinic, antispasmodic, and anticholinergic activity. This compound, being the (R)-isomer of Oxybutynin, competitively antagonizes Carbachol-induced contractions. It is particularly useful in researching neurogenic bladder dysfunction-related incontinence [1] [2] [3]. |
T31396
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Dexbrompheniramine is an antihistamine with anticholinergic properties. It is used to treat allergic diseases such as hay fever or urticaria. It can compete with histamine for H1 receptor sites on effector cells of the gastrointestinal tract, blood vessel |
T69516
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Thenalidine is an antihistamine with anticholinergic properties used as an antipruritic drug. It was withdrawn from the US, Canadian, and UK markets due to a risk of neutropenia. Thenalidine is an antagonist of the H1-receptor. |
T62218
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Parapenzolate bromide 是一种口服具有活力的 mAChR 拮抗剂。Parapenzolate bromide 是一种抗胆碱能剂,也是一种解痉挛剂。 |
T38952
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Triperiden is a chemical compound that serves as an inhibitor of influenza virus multiplication. Specifically, it exerts its antiviral activity by targeting the haemagglutinin of fowl plague virus (FPV) and inhibiting the conformational change in the haemagglutinin at acid pH. Additionally, Triperiden is classified as an anticholinergic anti-parkinsonism drug. |
T70473
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Parapenzolate Free Base is a safe and effective anticholinergic drug possessing antisecretory and antimotility properties and prolonged duration of action. Clinical investigation has shown that after an oral dose of the drug there was inhibition of both basal and histamine-stimulated acid outputs. |
T68735
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Ciclotropium (free base) is quaternary ammonium compound with anticholinergic and parasympatholytic activity. Oral Cyclotropium bromide inhibited fasting and meal-stimulated colonic motility significantly without causing adverse side effects. After cyclotropium bromide, there was a significant correlation between antral contraction amplitude and gastric emptying. |