首页化合物库经典已知活性库
经典已知活性库
BIOACTIVE COMPOUND LIBRARY

Catalog No.L4000

经典已知活性库是7739个具有生物活性,能引起细胞、组织甚至个体生物学反应的化合物的集合。包括了正在进行临床前研究的药物分子,临床期的药物分子和已经上市的药物。靶点明确,信息全面,非常适合完成药物功能重定位、小分子诱导细胞分化以及机制研究中蛋白靶点确认等科研工作。

由于活性明确,靶点已知,很多科学家会从已知活性库中选择可以用于细胞诱导分化的小分子,通过单一或几个小分子的联合作用,选择出将各种体细胞诱导成为诱导多能干细胞,神经前体细胞,心肌细胞等,甚至还有使用小分子组合在体内完成诱导分化的成功尝试。

为了保证客户的最佳使用效果,我们把已知活性库中需要现配现用的多肽以及其他药物分子以干粉形式提供(设置为PartB),尽可能增加新的药物筛选机会,增加成功筛选到目标分子的几率。

包含L4000已知活性库在内,陶素生化可以提供多达4万种生物活性已知的小分子化合物,可以满足您在各个阶段的科研工作需要,欢迎随时和我们联系。

Pack Size Price
100 μL * 10 mM (in DMSO) RMB 528967.00
250 μL * 10 mM (in DMSO) RMB 799522.00
1 mg RMB 799522.00
产品特性
  • 7739个已知活性化合物的集合,可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认;
  • 所有化合物都有相应的靶点信息的描述,靶点信息已知;
  • 是老药新用、细胞诱导靶点筛选的有效工具;
  • 涵盖多个疾病研究领域,如癌症、代谢、免疫和心血管系统等;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • 结构多样,药效显著,可渗透细胞;
  • NMR、HPLC/ LCMS多重检测,保证产品结构准确,纯度高,保障实验顺利进行。
包装与存储
  • 形式:可提供1 mg、5 mg的干粉以及DMSO 10 mM浓度的各种规格溶液;
  • 包装:化合物溶液置于带旋盖和二维码的储存管中,后排列于96孔板;
  • 保存:干粉可保存两年;溶于DMSO,-20 °C可保存一年,-80 °C 可保存两年,避免反复冻融;
  • 运输:蓝冰运输。
化合物库组成成分
AChR (179)
5-HT Receptor (158)
COX (133)
Adrenergic Receptor (132)
Antibiotic (119)
Antibacterial (115)
Endogenous Metabolite (100)
DNA/RNA Synthesis (99)
Dopamine Receptor (95)
PI3K (89)
EGFR (88)
VEGFR (86)
Histamine Receptor (81)
Estrogen/progestogen Receptor (75)
CDK (68)
Sodium Channel (67)
Potassium Channel (66)
Autophagy (64)
NF-κB (59)
P450 (57)
Calcium Channel (55)
HDAC (54)
Bcr-Abl (53)
GABA Receptor (52)
JAK (52)
PDGFR (51)
Dehydrogenase (51)
Src (51)
PPAR (50)
Glucocorticoid Receptor (49)
Antioxidant (49)
Topoisomerase (49)
mTOR (48)
PDE (46)
FLT (46)
FGFR (45)
Microtubule Associated (45)
TNF (45)
Epigenetic Reader Domain (43)
c-Kit (43)
Histone Methyltransferase (40)
HIV Protease (40)
GluR (39)
GR (39)
Vitamin (38)
p38 MAPK (37)
Raf (37)
ERK (36)
Akt (35)
RAAS (35)
ALK (33)
STAT (33)
Wnt/beta-catenin (32)
ATPase (32)
c-Met/HGFR (32)
ribosome (32)
PKC (31)
MAO (30)
Antifungal (30)
GSK-3 (30)
TRP/TRPV Channel (30)
Tyrosine Kinases (29)
Androgen Receptor (29)
MMP (28)
NMDAR (28)
Norepinephrine (26)
IL Receptor (26)
Opioid Receptor (25)
Aurora Kinase (25)
BCL (25)
Carbonic Anhydrase (25)
DNA-PK (25)
GPR (24)
Antifection (24)
HSP (24)
MEK (24)
ROS (23)
IκB/IKK (22)
HCV Protease (21)
HER (21)
Amino Acids and Derivatives (21)
AMPK (21)
DNA Alkylation (21)
Sirtuin (21)
TGF-beta/Smad (20)
Antiviral (20)
Prostaglandin Receptor (20)
PKA (19)
Phospholipase (19)
PARP (19)
JNK (19)
TAM Receptor (19)
Tyrosinase (19)
S6 Kinase (19)
HIF (18)
p53 (18)
ATM/ATR (18)
Caspase (18)
Glucokinase (18)
P2 Receptor (17)
ROCK (17)
Hedgehog/Smoothened (17)
IGF-1R (16)
MRP (16)
Reverse Transcriptase (16)
Gamma-secretase (16)
CaMK (16)
Apoptosis (16)
Serine Protease (16)
Trk receptor (16)
Transferase (15)
Syk (15)
BTK (15)
Cannabinoid Receptor (15)
Casein Kinase (15)
Cysteine Protease (15)
DUB (15)
Proteasome (15)
Mdm2 (15)
Histone Demethylase (15)
Lipoxygenase (14)
NOS (14)
c-RET (14)
CXCR (14)
Thrombin (14)
Retinoid Receptor (14)
Beta Amyloid (13)
Adenosine Receptor (13)
NADPH (13)
Phosphatase (13)
Reductase (12)
Parasite (12)
AhR (12)
Chk (12)
CCR (12)
DHFR (12)
FAK (12)
TLR (12)
Serine/threonin kinase (11)
S1P Receptor (11)
DPP-4 (11)
CFTR (11)
Apoptosis inducer (11)
LRRK2 (11)
MAPK (11)
Integrin (11)
HMG-CoA Reductase (10)
Proton pump (10)
PLK (10)
DNA gyrase (10)
Sigma receptor (10)
Thyroid hormone receptor(THR) (10)
SGLT (9)
DNA Methyltransferase (9)
Aromatase (9)
CAT (9)
Chloride channel (9)
P-gp (9)
OX Receptor (9)
NOD (9)
IDO (9)
HSV (8)
HIF/HIF Prolyl-Hydroxylase (8)
HBV (8)
LTR (8)
Lipase (8)
Kinesin (8)
PDK (8)
Pim (8)
Rho (8)
ABC (8)
FAAH (8)
Factor Xa (8)
FXR (7)
c-Fms (7)
CSF-1R (7)
BACE (7)
PERK (7)
Lipid (7)
UGT (7)
Vasopressin Receptor (6)
transporter (6)
Liver X Receptor (6)
GPCR19 (6)
Hydroxylase (6)
Influenza Virus (6)
Platelet aggregation (6)
p97 (6)
PAI-1 (6)
c-Myc (6)
Annexin A (6)
Endothelin Receptor (6)
Fatty Acid Synthase (6)
Ferroptosis (6)
Free radical scavengers (5)
GNRH Receptor (5)
Ephrin Receptor (5)
CRM1 (5)
Nrf2 (5)
NAMPT (5)
PKM (5)
ROR (5)
IAP (5)
MPO (5)
Tie-2 (5)
Telomerase (5)
SGK (4)
Monocarboxylate transporter (4)
MLK (4)
LPA Receptor (4)
LDL (4)
PYK2 (4)
Protease-activated Receptor (4)
Porcupine (4)
Neurokinin receptor (4)
OCT (4)
PAK (4)
DprE1 (4)
DYRK (4)
E1/E2/E3 Enzyme (4)
cholecystokinin (4)
cell cycle arrest (4)
Cell wall (4)
CETP (4)
BMI-1 (3)
cAMP (3)
Carboxypeptidase(CPG2) (3)
Arginase (3)
ACAT (3)
Acetyl-CoA Carboxylase (3)
ACK (3)
advanced glycation end products (3)
Aminopeptidase (3)
Dynamin (3)
Decarboxylase (3)
DNA (3)
GRK (3)
GST (3)
Glucagon Receptor (3)
GluCls (3)
PD-1/PD-L1 (3)
PAFR (3)
Na-K-Cl cotransporter (3)
Nucleoside Antimetabolite/Analog (3)
NPC1L1 (3)
PGE Synthase (3)
Phosphorylase (3)
Ras (3)
LIM Kinase (3)
Monoamine Transporter (3)
MNK (3)
MT Receptor (3)
MTH1 (3)
Mitophagy (3)
Hck (3)
Histone Acetyltransferase (2)
Immunology & Inflammation related (2)
Mitochondrial Metabolism (2)
Melatonin Receptor (2)
KSP (2)
lysosomal autophagy (2)
PED (2)
OAT (2)
NADPH-oxidase (2)
Gap Junction Protein (2)
GTPase (2)
Glutathione reductase (2)
GlyT (2)
Discoidin Domain Receptor (DDR) (2)
Acyltransferase (2)
ASK (2)
ATP Citrate Lyase (2)
Bombesin Receptor (2)
BCRP (2)
CaSR (2)
Survivin (2)
Transaminase (2)
VDA (2)
Wee1 (2)
Wnk (2)
Xanthine Oxidase (1)
TOPK (1)
Thioredoxin (1)
Stemness kinase (1)
Somatostatin (1)
Serotonin Transporter (1)
Salt-Inducible Kinase (1)
CGRP Receptor (1)
Beta-Secretase (1)
BVDV (1)
Anion Exchanger (1)
Apelin receptor (1)
Adiponectin receptor (1)
AChE (1)
DNA Alkylator/Crosslinker (1)
CPT (1)
Electron transport (1)
FABP (1)
gp120/CD4 (1)
Glutaminase (1)
GSNOR (1)
GPX (1)
GHSR (1)
Fas/FasL (1)
FOXO1 (1)
N-Acetylglucosaminyltransferase (1)
NKCC (1)
NOD-like Receptor (NLR) (1)
P2X Receptor (1)
RAR/RXR (1)
PTEN (1)
MALT (1)
Keap1-Nrf (1)
LHRH (1)
MELK (1)
Monoamine Oxidase (1)
Integrase (1)
Interleukin Related (1)
IP3 Receptor  (1)
IRAK (1)
Hydrogenase (1)
iGluR (1)
Histone Acetylation (1)
hCE (1)
Hippo pathway (1)
陶素化合物库特点:
  • 详细的化学结构
  • 二维码储存管
  • 蓝冰干冰运输
  • NMR和HPLC保证产品纯度

默认产品规格为:
  • 1mg/well (powder)
  • 100μL/well (10mM solution)
  • 250μL/well (10mM solution)

* 产品高度可定制化,用户可以选择自己的化合物组库。
技术支持
在订购、运输、储存和使用我们的产品的任何阶段,您遇到的任何问题,均可以通过拨打我们的热线电话400-998-7375,或者邮箱 info@tsbiochem.com,直接联系到我们。我们会在24小时内尽快联系您。
订购方式
联系陶素
电话:400-821-2233
传真:021-34692979
邮箱:info@tsbiochem.com


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