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human_metabolite_library
/library/human_metabolite_library
人代谢物化合物库
Human Metabolite Library
产品编号: L2570

人代谢物包括内源性代谢物和外源性代谢物;内源性代谢物,顾名思义,就是人体内产生和发现的一些代谢产物,如柠檬酸循环的任何中间代谢物,这些代谢物参与机体重要的生理过程,可作为潜在的药物先导物。外源性代谢物不在机体内产生与发现,来源于外界,包括药物、毒素和食品添加剂等,研究外源性代谢物在人体内如何发生代谢,有助于加快药物发现和毒理学的研究。在药物发现中,了解药物的代谢物有助于对药物作用机理的研究。

TargetMol 人代谢物化合物库收集了4532 种内源性和外源性代谢物,包括羧酸、氨基酸、生物胺、核苷酸、维生素、单糖、双糖、脂类、碳水化合物等不同种类代谢物。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
产品规格
  • 4532种人代谢物的独特集合,用于高通量、高内涵筛选;
  • 研究人体代谢疾病、探索癌症发病机制和寻找新药的有效工具;
  • 部分化合物已上市或进入临床,具有生物安全保障和良好的生物活性;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
化合物库定制
我们的化合物库可以灵活定制!了解更多
化合物库咨询
化合物库组成
Endogenous Metabolite (1006)
Apoptosis (455)
Antibacterial (403)
Autophagy (385)
Antibiotic (267)
COX (162)
Antifungal (134)
NF-κB (127)
Parasite (118)
5-HT Receptor (102)
Reactive Oxygen Species (99)
DNA/RNA Synthesis (99)
HIV Protease (96)
P450 (84)
AChR (77)
Influenza Virus (72)
Antioxidant (70)
Calcium Channel (69)
Dopamine Receptor (68)
Adrenergic Receptor (68)
Histamine Receptor (64)
PPAR (62)
Potassium Channel (57)
GABA Receptor (54)
Estrogen/progestogen Receptor (53)
PDE (51)
TNF (51)
Ferroptosis (49)
Sodium Channel (47)
PI3K (41)
Topoisomerase (40)
Estrogen Receptor/ERR (38)
Virus Protease (37)
ERK (37)
HSV (37)
EGFR (37)
Prostaglandin Receptor (37)
Microtubule Associated (37)
VEGFR (36)
p38 MAPK (35)
Mitophagy (35)
Nucleoside Antimetabolite/Analog (35)
Caspase (35)
Glucocorticoid Receptor (35)
NO Synthase (35)
Dehydrogenase (34)
MMP (34)
AChE (34)
Akt (33)
SARS-CoV (33)
HCV Protease (31)
Reverse Transcriptase (31)
RAAS (29)
AMPK (29)
PDGFR (28)
IL Receptor (28)
STAT (28)
Adenosine Receptor (27)
HDAC (27)
PKC (26)
TRP/TRPV Channel (26)
Drug Metabolite (26)
ROS (26)
c-Kit (26)
ATPase (25)
Lipoxygenase (25)
Nrf2 (24)
Anti-infection (24)
Tyrosinase (24)
PARP (22)
Androgen Receptor (22)
FLT (22)
Proteasome (21)
DNA Alkylator/Crosslinker (21)
JNK (21)
Progesterone Receptor (21)
iGluR (21)
BCL (21)
Antifection (20)
JAK (20)
P-gp (20)
Beta Amyloid (20)
Carbonic Anhydrase (19)
Antiviral (19)
FGFR (19)
HBV (18)
MAO (18)
CDK (18)
NMDAR (18)
Mitochondrial Metabolism (18)
mTOR (18)
ribosome (18)
Phospholipase (18)
Amino Acids and Derivatives (17)
Opioid Receptor (17)
GluR (16)
TLR (15)
GPR (15)
HIF/HIF Prolyl-Hydroxylase (15)
NOS (14)
Transferase (14)
Src (14)
Phosphatase (14)
MRP (14)
Tyrosine Kinases (14)
Interleukin (14)
Chloride channel (13)
Reductase (13)
Wnt/beta-catenin (13)
Serotonin Transporter (13)
DNA Alkylation (13)
TGF-beta/Smad (13)
Monoamine Oxidase (13)
Bcr-Abl (12)
Glucosidase (12)
Retinoid Receptor (12)
Proton pump (11)
Raf (11)
DPP-4 (11)
CaMK (11)
MEK (11)
HMG-CoA Reductase (11)
DHFR (10)
PKA (10)
Antifolate (10)
Gamma-secretase (10)
Fatty Acid Synthase (10)
Epigenetic Reader Domain (10)
Norepinephrine (10)
HSP (10)
Sirtuin (10)
HIF (10)
Thrombin (10)
Thyroid hormone receptor(THR) (9)
c-Met/HGFR (9)
Aryl Hydrocarbon Receptor (9)
Immunology/Inflammation related (9)
E1/E2/E3 Enzyme (9)
Hedgehog/Smoothened (9)
Xanthine Oxidase (9)
IGF-1R (9)
Trk receptor (9)
IκB/IKK (9)
Cannabinoid Receptor (9)
Neurokinin receptor (9)
AhR (9)
p53 (9)
HER (9)
FXR (8)
CCR (8)
CXCR (8)
c-RET (8)
Integrin (7)
NADPH (7)
Melatonin Receptor (7)
ABC (7)
Cysteine Protease (7)
Leukotriene Receptor (7)
Monoamine Transporter (7)
SGLT (7)
PGE Synthase (7)
transporter (7)
ALK (7)
NOD (7)
DNA Methyltransferase (7)
Histone Methyltransferase (6)
P2Y Receptor (6)
Glutathione Peroxidase (6)
Factor Xa (6)
GSK-3 (6)
UGT (6)
Endothelin Receptor (6)
Lipid (6)
Aromatase (6)
Platelet aggregation (6)
TAM Receptor (6)
CFTR (6)
CAT (5)
LTR (5)
GNRH Receptor (5)
Serine Protease (5)
MT Receptor (5)
Guanylate cyclase (5)
Epoxide Hydrolase (5)
DNA (5)
MAPK (5)
Acyltransferase (5)
Free radical scavengers (5)
Ligand for E3 Ligase (5)
PLK (5)
NOD-like Receptor (NLR) (5)
S1P Receptor (5)
Arginase (4)
LPL Receptor (4)
BACE (4)
CETP (4)
PERK (4)
CaSR (4)
cell cycle arrest (4)
Glucokinase (4)
IAP (4)
Annexin A (4)
Adiponectin receptor (4)
DNA gyrase (4)
BTK (4)
Smo (4)
FAAH (4)
PTEN (4)
Aurora Kinase (4)
Telomerase (4)
ATP Citrate Lyase (4)
OAT (4)
Aminopeptidase (4)
Histone Acetyltransferase (4)
RSV (4)
GST (4)
Hydroxylase (4)
Adenosine deaminase (4)
Syk (4)
cholecystokinin (4)
FAK (4)
ROS Kinase (4)
Imidazoline Receptor (4)
DNA-PK (3)
IFNAR (3)
Histone Demethylase (3)
Lipase (3)
Serine/threonin kinase (3)
ROCK (3)
CSF-1R (3)
PAFR (3)
LDL (3)
Phosphorylase (3)
GlyT (3)
Molecular Glues (3)
Isocitrate Dehydrogenase (IDH) (3)
PROTAC Linker (3)
cAMP (3)
Indoleamine 2,3-Dioxygenase (IDO) (3)
Glutathione reductase (3)
GPCR19 (3)
Casein Kinase (3)
Neprilysin (3)
c-Fms (3)
S6 Kinase (3)
Ras (3)
Sigma receptor (3)
advanced glycation end products (2)
Mdm2 (2)
Adenylyl cyclase (2)
NPC1L1 (2)
Monocarboxylate transporter (2)
ROR (2)
CRM1 (2)
Ligands for Target Protein for PROTAC (2)
YAP (2)
Na+/Ca2+ Exchanger (2)
Tie-2 (2)
VDA (2)
Rho (2)
Liver X Receptor (2)
Amylase (2)
IRE1 (2)
P2X Receptor (2)
Na-K-Cl cotransporter (2)
Hexokinase (2)
Bombesin Receptor (2)
PAK (2)
Vasopressin Receptor (2)
Bradykinin Receptor (2)
Angiotensin-converting Enzyme (ACE) (2)
OX Receptor (2)
Thrombopoietin Receptor (2)
DUB (2)
BCRP (2)
Beta-Secretase (2)
STING (2)
Ephrin Receptor (2)
Decarboxylase (2)
GluCls (2)
Pyroptosis (2)
ATM/ATR (2)
Carboxypeptidase (2)
CRISPR/Cas9 (2)
CGRP Receptor (2)
Complement System (2)
NADPH-oxidase (2)
Protease-activated Receptor (2)
Apelin receptor (1)
Taste receptor (1)
Transaminase (1)
Hydrogenase (1)
stilbene oxidase (1)
CD38 (1)
CYP19A1 (1)
Dynamin (1)
NEDD8 (1)
aconitase (1)
RAR/RXR  (1)
DYRK (1)
Cell wall (1)
gp120/CD4 (1)
LHRH (1)
TOPK (1)
c-Myc (1)
N-Acetylglucosaminyltransferase (1)
Hck (1)
NAMPT (1)
Glutaminase (1)
RANKL/RANK (1)
IDO (1)
Myosin (1)
FLAP (1)
RIP kinase (1)
MTH1 (1)
Fas/FasL (1)
Glucagon Receptor (1)
Anion Exchanger (1)
Stearoyl-CoA Desaturase (SCD) (1)
Chk (1)
Somatostatin (1)
PAD (1)
ACK (1)
KSP (1)
Wee1 (1)
Survivin (1)
LRRK2 (1)
hCE (1)
PAI-1 (1)
Acetyl-CoA Carboxylase (1)
GPX (1)
PDK (1)
Oxytocin Receptor (1)
IRAK (1)
p97 (1)
PD-1/PD-L1 (1)
Kinesin (1)
化合物库信息示例
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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