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ubiquitination_compound_library
/library/ubiquitination_compound_library
泛素化化合物库
Ubiquitination Compound Library
产品编号: L8600

泛素化是泛素在一系列特殊的酶催化下对靶蛋白进行特异性修饰的过程,这些特殊的酶包括泛素激活酶、结合酶、连结酶和降解酶等。泛素化被认为是蛋白质翻译后修饰的一个重要途径,在细胞凋亡、细胞周期调控、DNA 损伤修复及膜转运等细胞过程中起重要作用,与肿瘤、心血管等疾病的发病密切相关。作为近年来生物化学研究的一个重大成果,泛素化已然成为研究、开发新药物的新靶点。

TargetMol 泛素化化合物库收集了214 种泛素化相关的小分子,作用靶点包括proteasome, E1/E2/E3 Enzyme, DUB, p97等,满足泛素化相关研究的客户需求。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
产品规格
  • 214种泛素化相关的小分子,用于高通量和高内涵筛选;
  • 作用靶点包括proteasome, E1/E2/E3 Enzyme, DUB, p97等;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
化合物库定制
我们的化合物库可以灵活定制!了解更多
化合物库咨询
化合物库组成
Proteasome (62)
E1/E2/E3 Enzyme (49)
Apoptosis (44)
DUB (41)
p53 (30)
Autophagy (29)
DPP-4 (20)
Mdm2 (18)
NF-κB (13)
Ferroptosis (8)
p97 (7)
Cysteine Protease (5)
Antibacterial (5)
Sirtuin (5)
HIV Protease (4)
Dehydrogenase (4)
NEDD8 (3)
Mitophagy (3)
PARP (3)
Caspase (3)
IAP (3)
BCL (3)
Epigenetic Reader Domain (3)
IκB/IKK (3)
PROTACs (2)
Antifungal (2)
DNA Alkylator/Crosslinker (2)
PPAR (2)
Aryl Hydrocarbon Receptor (2)
Bcr-Abl (2)
MMP (2)
COX (2)
SARS-CoV (2)
Endogenous Metabolite (2)
Ligand for E3 Ligase (2)
HDAC (2)
Antibiotic (2)
HCV Protease (1)
Src (1)
Amino Acids and Derivatives (1)
p38 MAPK (1)
Factor Xa (1)
Serine Protease (1)
PKC (1)
ERK (1)
RIP kinase (1)
PDE (1)
CDK (1)
NMDAR (1)
Mitochondrial Metabolism (1)
Molecular Glues (1)
Reactive Oxygen Species (1)
JAK (1)
HSV (1)
IGF-1R (1)
HSP (1)
TLR (1)
Aminopeptidase (1)
Neprilysin (1)
Retinoid Receptor (1)
AMPK (1)
TNF (1)
Potassium Channel (1)
Syk (1)
DNA Methyltransferase (1)
BMI-1 (1)
TAM Receptor (1)
Protease-activated Receptor (1)
HIF/HIF Prolyl-Hydroxylase (1)
化合物库信息示例
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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