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selected_plant_sourced_compound_library
/library/selected_plant_sourced_compound_library
植物来源化合物库
Selected Plant-Sourced Compound Library
产品编号: L4600

自然界创造了几乎无穷无尽的分子实体,为药物研发特别是新型药效团的发现创造了无限资源。在全球范围内,天然产物自古以来一直都是传统治疗的支柱。植物作为药物治疗疾病具有悠久的历史,植物来源的化合物具有更好的耐受性和可接受性。迄今为止,已对35,000-70,000种植物进行了药用筛选。半合成纯药物阿司匹林,是基于从白柳中分离出的天然产品水杨苷,由拜耳于1899年推出。此后陆续分离出了多种早期药物,如洋地黄毒苷、奎宁和毛果芸香碱等,其中一些仍在使用中,以及其他一些近期出现的植物衍生化合物,这些化合物经过开发并已作为药物销售,其中包括:来自短叶红豆杉的紫杉醇,用于肺部、卵巢癌和乳腺癌;青蒿素来自中国传统植物青蒿,用于对抗多药耐药性疟疾;水飞蓟素从水飞蓟种子中提取,用于治疗肝脏疾病。 TargetMol 植物来源化合物库精选3076 个植物来源天然产物的独特集合,具有良好的成药潜力,可用于天然产物来源的化合物筛选和新药研发。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
产品规格
  • 3076个植物来源天然产物的独特集合;
  • 可用于高通量筛选和高内涵筛选;
  • 处于临床前研究或临床期实验阶段,是颇具研究潜力的天然产物集合;
  • 包含青蒿素,人参皂苷等热门的天然产物;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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化合物库组成
Endogenous Metabolite (441)
Apoptosis (346)
Antibacterial (228)
Autophagy (207)
NF-κB (180)
Antifungal (109)
Antioxidant (106)
COX (89)
Reactive Oxygen Species (88)
Parasite (74)
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TNF (58)
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Antibiotic (48)
HIV Protease (46)
NO Synthase (46)
p38 MAPK (45)
ERK (45)
IL Receptor (45)
Anti-infection (45)
Akt (42)
Caspase (39)
STAT (39)
PPAR (38)
Calcium Channel (38)
GABA Receptor (37)
Tyrosinase (37)
DNA/RNA Synthesis (36)
AMPK (33)
BCL (31)
Nrf2 (31)
Virus Protease (29)
MMP (29)
PI3K (27)
JNK (27)
Topoisomerase (26)
Lipoxygenase (26)
ROS (25)
5-HT Receptor (25)
Microtubule Associated (25)
Ferroptosis (24)
PKC (24)
NOS (23)
Estrogen Receptor/ERR (23)
TRP/TRPV Channel (23)
Dehydrogenase (22)
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Estrogen/progestogen Receptor (21)
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化合物库信息示例
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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