×
{{login.error}}
{{login.verifyresult}}
×
6~16个字符、区分大小写、必须包含字母和数字
6~16个字符、区分大小写、必须包含字母和数字
密码已经重置成功,快去使用新密码吧!
登录账号
密码已经重置成功,快去使用新密码吧! 登录账号
×

注册成功

确认
natural_compound_covalent_library
/library/natural_compound_covalent_library
天然产物共价化合物库
Covalent Natural Product Library
产品编号: L6150

天然产物已被证明可以成功的调控某些孤立的但又很重要的靶点,如一系列抗菌靶点,特别是蛋白质与蛋白质相互作用。因此,许多研究人员认为天然产物及其衍生物是研究和操纵蛋白质功能的独特工具。

共价化合物,是一类有机小分子,能与特定的靶蛋白相互作用并形成共价键,导致蛋白质构象的改变,从而抑制蛋白质的活性。除了部分例外,通过共价作用进行的蛋白质修饰通常是不可逆的。

TargetMol 天然产物共价库精心筛选 596 种天然产物共价化合物,不仅具有天然产物的特点,还具有共价化合物的作用机制,性价比高,是药物开发、药理研究、干细胞分化、指纹图谱研究、质量研究等领域的有力工具。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
产品规格
  • 提供产品的生物学信息和药物学信息,为筛选提供理论方向和研究基础;
  • 来源清晰:精选来自动物、植物、微生物的已知活性天然产物;更具体到植物种属,并标注准确英文名与拉丁名,方便您的后期研究确证。
  • 信息全面:从化合物结构到溶解度,从信号通路、作用靶点到生物活性信息均有详细描述。
  • 性价比高:剔除了价格昂贵但成药性差的天然产物,让您用更少的成本得到更多高品质的天然产物。
  • 可根据天然产物来源、天然产物类别、研究领域、药物市场状态等方面自由组合,高度定制。
化合物库定制
我们的化合物库可以灵活定制!了解更多
化合物库咨询
化合物库组成
Endogenous Metabolite (111)
Apoptosis (91)
Antibacterial (69)
Autophagy (48)
Antibiotic (43)
NF-κB (43)
Reactive Oxygen Species (30)
Antifungal (24)
Antioxidant (19)
Influenza Virus (18)
COX (15)
HIV Protease (11)
Parasite (11)
Calcium Channel (10)
Dehydrogenase (10)
ERK (9)
Estrogen/progestogen Receptor (9)
Ferroptosis (9)
GABA Receptor (9)
p38 MAPK (9)
P450 (9)
ribosome (9)
STAT (9)
AChE (8)
Akt (8)
Anti-infection (8)
ATPase (8)
BCL (8)
MMP (8)
TNF (8)
AMPK (7)
Androgen Receptor (7)
Antiviral (7)
HSV (7)
NO Synthase (7)
ROS (7)
Caspase (6)
Glucocorticoid Receptor (6)
Microtubule Associated (6)
NOS (6)
PKC (6)
Progesterone Receptor (6)
AChR (5)
HIF/HIF Prolyl-Hydroxylase (5)
IL Receptor (5)
Immunology/Inflammation related (5)
Mitophagy (5)
Nrf2 (5)
P-gp (5)
SARS-CoV (5)
Tyrosinase (5)
Wnt/beta-catenin (5)
DNA/RNA Synthesis (4)
Drug Metabolite (4)
HBV (4)
HSP (4)
Lipoxygenase (4)
Prostaglandin Receptor (4)
Reductase (4)
TRP/TRPV Channel (4)
VEGFR (4)
Virus Protease (4)
Aromatase (3)
Beta Amyloid (3)
CaMK (3)
EGFR (3)
Epigenetic Reader Domain (3)
Estrogen Receptor/ERR (3)
HDAC (3)
IκB/IKK (3)
JAK (3)
JNK (3)
Mitochondrial Metabolism (3)
Opioid Receptor (3)
PI3K (3)
PPAR (3)
Proteasome (3)
Retinoid Receptor (3)
Sodium Channel (3)
5-HT Receptor (2)
Adrenergic Receptor (2)
Antifolate (2)
BACE (2)
Chloride channel (2)
DNA Methyltransferase (2)
FGFR (2)
HIF (2)
iGluR (2)
Interleukin (2)
MAO (2)
MAPK (2)
NMDAR (2)
Nucleoside Antimetabolite/Analog (2)
p53 (2)
PDE (2)
RAAS (2)
TGF-beta/Smad (2)
Thrombin (2)
TLR (2)
UGT (2)
ABC (1)
Acyltransferase (1)
Antifection (1)
Aurora Kinase (1)
Beta-Secretase (1)
CAT (1)
CDK (1)
c-Met/HGFR (1)
CRISPR/Cas9 (1)
DNA gyrase (1)
Dopamine Receptor (1)
FAK (1)
Free radical scavengers (1)
FXR (1)
Gamma-secretase (1)
Glucagon Receptor (1)
Glucosidase (1)
GluR (1)
Glutathione reductase (1)
GSK-3 (1)
HCV Protease (1)
Hedgehog/Smoothened (1)
HER (1)
Histamine Receptor (1)
Histone Acetyltransferase (1)
Histone Methyltransferase (1)
IAP (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Integrin (1)
Lipid (1)
Mdm2 (1)
Monoamine Oxidase (1)
Monoamine Transporter (1)
mTOR (1)
Oxytocin Receptor (1)
PARP (1)
PD-1/PD-L1 (1)
PDGFR (1)
PGE Synthase (1)
Phosphatase (1)
Phospholipase (1)
PKA (1)
PKM (1)
Potassium Channel (1)
Proton pump (1)
PTEN (1)
Pyroptosis (1)
Raf (1)
RANKL/RANK (1)
RAR/RXR  (1)
Ras (1)
Serine Protease (1)
Sirtuin (1)
Smo (1)
Src (1)
Telomerase (1)
Topoisomerase (1)
Transaminase (1)
Transferase (1)
Tyrosine Kinases (1)
化合物库信息示例
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
联系我们
400-820-0310
service@tsbiochem.com

上海市静安区江场三路238号8楼