药物代谢杂质库 | 陶术生物

药物代谢杂质库现货

Drug Metabolite/Impurity Library

产品编号： L5800

随着科研深入，科学家们发现已经上市的药物异构体/代谢产物中很多都是有明确的生物活性的。比如：左丙氧芬(levopropoxyphene)曾是 FDA 批准的镇咳药，而它的旋光异构体右丙氧芬(Dextropropoxyphene)是则有镇痛效果。再比如右旋索它洛尔属于 III 类抗心律失常药，而左旋体则为β-受体阻滞剂。这些化合物在科研上已有的药理评价数据较为丰富，作为老药新用的切入点较为理想。

TargetMol 作为全球知名的化合物库供应商，积极关注科研动态，药物代谢杂质库共有200 种产品，多样性好，重复供应能力强，为您提供药物筛选的一站式服务。

陶术生物的所有产品和服务仅用于科学研究，我们不为任何个人用途提供产品和服务。

产品规格

技术资料

陶术生物化合物库目录(28.1MB)

库化合物信息

Excel

SDF

产品描述

200 种药物异构体/代谢产物的特有集合，可用于高通量、高内涵筛选；
可提供基于筛选片段的衍生物以及定制合成服务，降低您的合成成本，缩短研发时间；
结构多样，药效显著，可渗透细胞；
详细的说明书，化合物结构、靶点信息、IC50值、活性描述等；
NMR、HPLC/LCMS等多种检测技术保证产品结构正确，纯度高，减少假阳性。

化合物库定制

我们的化合物库可以灵活定制！了解更多

化合物库咨询

化合物库组成

Endogenous Metabolite (35)

Apoptosis (9)

Autophagy (8)

Antibiotic (6)

DNA/RNA Synthesis (6)

Amino Acids and Derivatives (5)

Drug Metabolite (5)

5-HT Receptor (4)

Antibacterial (4)

Antioxidant (4)

COX (4)

Nucleoside Antimetabolite/Analog (4)

AChR (3)

Estrogen/progestogen Receptor (3)

Adenosine Receptor (2)

Adrenergic Receptor (2)

Aromatase (2)

c-Kit (2)

Dopamine Receptor (2)

Estrogen Receptor/ERR (2)

Factor Xa (2)

HIV Protease (2)

Microtubule Associated (2)

Mitophagy (2)

NF-κB (2)

P450 (2)

PDGFR (2)

ROS (2)

VEGFR (2)

Androgen Receptor (1)

Antifungal (1)

Aryl Hydrocarbon Receptor (1)

ATPase (1)

Calcium Channel (1)

CAT (1)

c-Myc (1)

c-RET (1)

CXCR (1)

Dehydrogenase (1)

DNA Alkylator/Crosslinker (1)

DPP-4 (1)

GABA Receptor (1)

Glucokinase (1)

Glutathione Peroxidase (1)

Histamine Receptor (1)

IGF-1R (1)

iGluR (1)

IL Receptor (1)

Lipoxygenase (1)

Neurokinin receptor (1)

NMDAR (1)

Norepinephrine (1)

P2 Receptor (1)

P2X Receptor (1)

p38 MAPK (1)

PAK (1)

Parasite (1)

PDE (1)

P-gp (1)

PI3K (1)

PPAR (1)

Proton pump (1)

Raf (1)

S6 Kinase (1)

Sodium Channel (1)

Thyroid hormone receptor(THR) (1)

Topoisomerase (1)

Trk receptor (1)

Tyrosinase (1)

Xanthine Oxidase (1)

化合物库信息示例

Empty	1000025-07-9	1000413-72-8	229005-80-5	1000787-75-6	946387-07-1	1000998-59-3	1175526-27-8	1001288-58-9	1001350-96-4	1001404-83-6	Empty
Empty	Vadadustat	TAK875	TAK-779	Tegobuvir	RN-1734	BMS-687453	AM211	FT011	BMS754807	AAI101	Empty
Empty	1001625-82-6	1001645-58-4	1001753-24-7	1001908-89-9	1002304-34-8	1002-84-2	100291-86-9	100299-08-9	10030-52-1	10040-45-6	Empty
Empty	RPW-24	SRT1720 hydrochloride	INH6	SRT 2183	AMG208	Pentadecanoic acid	Apiopaeonoside	Pemirolast potassium	L-Anserine nitrate salt	Sodium Picosulfate	Empty
Empty	100427-26-7	1004316-88-4	10045-45-1	100462-37-1	1004990-28-6	100-51-6	1005-24-9	1005264-47-0	1005334-57-5	1005342-46-0	Empty
Empty	Lercanidipine	Cobicistat	1-Ethyl-2-benzimidazolinone	ROSIRIDIN	PF-AKT400	Benzyl alcohol	1-Methylnicotinamide chloride	MX69	CVT-10216	LCL161	Empty
Empty	1005491-05-3	100-55-0	1005504-62-0	1005883-72-6	100643-71-8	1007207-67-1	10075-50-0	1007647-73-5	100784-20-1	10083-24-6	Empty
Empty	Tirasemtiv	Roniacol	Rg3039	Z433927330	Desloratadine	CH5132799	5-Bromoindole	Smurf1-IN-A01	Halosulfuron-methyl	Piceatannol	Empty
Empty	100872-83-1	100874-08-6	1009119-64-5	1009119-65-6	100929-71-3	1009298-09-2	1009298-59-2	100929-99-5	1009734-33-1	10097-84-4	Empty
Empty	ML346	SB 4	Daclatasvir	Daclatasvir dihydrochloride	NADPH (tetracyclohexanamine)	AZD8055	Vistusertib	PAβN dihydrochloride	HZ1157	Rotundine	Empty
Empty	1009816-48-1	1009817-63-3	1009820-21-6	100986-85-4	101001-34-7	1010411-21-8	1010-60-2	1011244-68-0	1011301-27-1	1011529-10-4	Empty
Empty	Thiamet G	B-AP15	Silmitasertib	Levofloxacin	Pamicogrel	GSK369796 Dihydrochloride	2-Chloronaphthoquinone	TFAP	Tenovin3	Azvudine	Empty
Empty	101152-94-7	101155-02-6	1011557-82-6	1011-74-1	101-20-2	1012054-59-9	101-21-3	101-26-8	101303-98-4	1013101-36-4	Empty
Empty	Milnacipran hydrochloride	BW-A78U	Tenovin-6	DL-Normetanephrine hydrochloride	Triclocarban	CUDC101	Chlorpropham	Mestinon	Zacopride hydrochloride	PF04691502	Empty
Empty	101-31-5	1013-69-0	1013750-77-0	1013753-99-5	10138-52-0	1013920-15-4	1013937-63-7	1014691-61-2	101477-54-7	101494-95-5	Empty
Empty	L-Hyoscyamine	Noreugenin	ML-030	BC-1382	Gadolinium chloride	Vorolanib	VTP-27999 TFA	GSK0660	Lomerizine hydrochloride	8-CHLOROQUINAZOLIN-4(1H)-ONE	Empty

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