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preclinical_compound_library
/library/preclinical_compound_library
临床前化合物库
Preclinical Compound Library
产品编号: L3410

701 个临床前小分子化合物的独特集合,靶点明确,有详细的临床分期和适应症信息,可用于高通量、高内涵筛选。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
产品规格
  • 701种临床前小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 拥有明确的靶点信息;有详细的临床分期和适应症信息;
  • 是新药研发过程中的热门先导化合物;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。
化合物库定制
我们的化合物库可以灵活定制!了解更多
化合物库咨询
化合物库组成
Apoptosis (128)
Autophagy (110)
Endogenous Metabolite (36)
Antibacterial (35)
Antibiotic (33)
VEGFR (25)
CDK (24)
HIV Protease (20)
PI3K (19)
PDGFR (19)
FGFR (19)
EGFR (18)
DNA/RNA Synthesis (18)
Influenza Virus (17)
NF-κB (17)
JAK (16)
Adrenergic Receptor (13)
Dopamine Receptor (12)
Histamine Receptor (12)
Epigenetic Reader Domain (12)
mTOR (12)
5-HT Receptor (12)
FLT (12)
c-Kit (12)
Src (11)
Parasite (11)
Calcium Channel (11)
HDAC (11)
Sodium Channel (11)
Microtubule Associated (11)
Ferroptosis (10)
c-Met/HGFR (10)
PDE (10)
c-RET (10)
AChR (10)
Adenosine Receptor (9)
Phosphatase (9)
Mitophagy (9)
PPAR (9)
E1/E2/E3 Enzyme (9)
Raf (9)
Reactive Oxygen Species (9)
Aurora Kinase (9)
HSP (9)
ATM/ATR (9)
Potassium Channel (9)
DNA-PK (8)
PKC (8)
iGluR (8)
Bcr-Abl (8)
BCL (8)
GluR (8)
COX (8)
SARS-CoV (8)
ALK (8)
MEK (8)
p53 (8)
p38 MAPK (7)
Dehydrogenase (7)
Antifungal (7)
GSK-3 (7)
NMDAR (7)
ROS (7)
IGF-1R (7)
Trk receptor (7)
STAT (7)
PLK (7)
Mdm2 (6)
Histone Methyltransferase (6)
DNA Alkylator/Crosslinker (6)
Tyrosine Kinases (6)
Topoisomerase (6)
Akt (6)
Casein Kinase (6)
Beta Amyloid (6)
P450 (6)
Proteasome (5)
HBV (5)
FXR (5)
Opioid Receptor (5)
Chk (5)
Lipoxygenase (5)
TGF-beta/Smad (5)
Reverse Transcriptase (5)
PDK (5)
AMPK (5)
GABA Receptor (5)
Ras (5)
TAM Receptor (5)
Estrogen/progestogen Receptor (4)
LPL Receptor (4)
RAAS (4)
Wnt/beta-catenin (4)
PARP (4)
Pim (4)
Serine Protease (4)
TRP/TRPV Channel (4)
ERK (4)
Gamma-secretase (4)
BTK (4)
IL Receptor (4)
Endothelin Receptor (4)
Sirtuin (4)
Hydroxylase (4)
TNF (4)
Cannabinoid Receptor (4)
Syk (4)
S6 Kinase (4)
Sigma receptor (4)
HIF/HIF Prolyl-Hydroxylase (4)
FAK (4)
HER (4)
HCV Protease (3)
Integrin (3)
CRM1 (3)
NADPH (3)
JNK (3)
Virus Protease (3)
PKA (3)
Estrogen Receptor/ERR (3)
Serine/threonin kinase (3)
Cysteine Protease (3)
Nucleoside Antimetabolite/Analog (3)
Glucokinase (3)
ROCK (3)
Glucocorticoid Receptor (3)
Mitochondrial Metabolism (3)
Guanylate cyclase (3)
Smo (3)
Hedgehog/Smoothened (3)
MMP (3)
Norepinephrine (3)
DUB (3)
Interleukin (3)
MAPK (3)
Prostaglandin Receptor (3)
TLR (3)
Aminopeptidase (3)
Nrf2 (3)
MELK (3)
Retinoid Receptor (3)
c-Fms (3)
LPA Receptor (3)
Phospholipase (3)
HIF (3)
Complement System (3)
ROS Kinase (3)
ATPase (2)
Proton pump (2)
PROTACs (2)
NOS (2)
Transferase (2)
ROR (2)
Ligands for Target Protein for PROTAC (2)
Reductase (2)
IFNAR (2)
Histone Demethylase (2)
TOPK (2)
Progesterone Receptor (2)
MRP (2)
Liver X Receptor (2)
Leukotriene Receptor (2)
Caspase (2)
IRE1 (2)
FAAH (2)
HSV (2)
Vasopressin Receptor (2)
Xanthine Oxidase (2)
Androgen Receptor (2)
STING (2)
Histone Acetyltransferase (2)
transporter (2)
PAI-1 (2)
IκB/IKK (2)
Acetyl-CoA Carboxylase (2)
Ligand for E3 Ligase (2)
ribosome (2)
CRISPR/Cas9 (2)
GPR (2)
Oxytocin Receptor (2)
NADPH-oxidase (2)
HMG-CoA Reductase (2)
Kinesin (2)
S1P Receptor (2)
advanced glycation end products (1)
Chloride channel (1)
Taste receptor (1)
Adenylyl cyclase (1)
Carbonic Anhydrase (1)
Monocarboxylate transporter (1)
NPC1L1 (1)
MALT (1)
NEDD8 (1)
DprE1 (1)
Amino Acids and Derivatives (1)
Antioxidant (1)
P2Y Receptor (1)
LTR (1)
Na+/Ca2+ Exchanger (1)
PERK (1)
Tie-2 (1)
Glutathione Peroxidase (1)
gp120/CD4 (1)
Factor Xa (1)
CaSR (1)
GNRH Receptor (1)
Rho (1)
Antifolate (1)
cell cycle arrest (1)
PYK2 (1)
NAMPT (1)
Aryl Hydrocarbon Receptor (1)
CSF-1R (1)
IAP (1)
SIK (1)
FLAP (1)
RIP kinase (1)
UGT (1)
PAFR (1)
P2X Receptor (1)
GlyT (1)
Monoamine Transporter (1)
Molecular Glues (1)
Isocitrate Dehydrogenase (IDH) (1)
DPP-4 (1)
DNA Alkylation (1)
PAK (1)
CCR (1)
Bradykinin Receptor (1)
CXCR (1)
OX Receptor (1)
Somatostatin (1)
Epoxide Hydrolase (1)
Telomerase (1)
Lipid (1)
Wee1 (1)
BCRP (1)
OXPHOS (1)
AChE (1)
P-gp (1)
MNK (1)
GPCR19 (1)
Ephrin Receptor (1)
ASK (1)
Hippo pathway (1)
Carboxypeptidase (1)
Melanocortin Receptor (1)
Adenosine deaminase (1)
Gap Junction Protein (1)
Discoidin Domain Receptor (DDR) (1)
Neurokinin receptor (1)
Platelet aggregation (1)
NOD (1)
DNA Methyltransferase (1)
BMI-1 (1)
Thrombin (1)
lysosomal autophagy (1)
NOD-like Receptor (NLR) (1)
MLK (1)
PKM (1)
NO Synthase (1)
化合物库信息示例
Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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