Topoisomerase inhibitor kit 包含拓扑异构酶抑制剂,拓扑异构酶抑制剂能与相应异构酶易解离复合物结合,形成稳定复合物,阻止复制叉顺利通过,使DNA 链断裂,干扰DNA 的复制和转录。TargetMol 为您提供50种精选拓扑异构酶抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0125 | Epirubicin hydrochloride | 56390-09-1 | 579.98 | 10mM | Apoptosis; DNA/RNA Synthesis; Topoisomerase |
T0250 | Ciprofloxacin monohydrochloride | 93107-08-5 | 367.8 | 10mM | Antibacterial; Antibiotic; DNA gyrase; Topoisomerase |
T0274 | Cinoxacin | 28657-80-9 | 262.22 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T0331 | Moxifloxacin hydrochloride | 186826-86-8 | 437.89 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T0425 | Pefloxacin Mesylate | 70458-95-6 | 429.46 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T0486 | Irinotecan hydrochloride trihydrate | 136572-09-3 | 677.18 | 10mM | Autophagy; Topoisomerase |
T0902 | Ofloxacin | 82419-36-1 | 361.37 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T1020 | Doxorubicin hydrochloride | 25316-40-9 | 579.99 | 10mM | ADC Cytotoxin; AMPK; Antibacterial; Antibiotic; Apoptosis; Autophagy; HBV; HIV Protease; Mitophagy; Topoisomerase |
T1095 | Sparfloxacin | 110871-86-8 | 392.4 | 10mM | Antibacterial; Antibiotic; DNA gyrase; Topoisomerase |
T1121 | Podofilox | 518-28-5 | 414.41 | 10mM | Microtubule Associated; Topoisomerase |
T1123 | Camptothecin | 7689-03-4 | 348.36 | 10mM | ADC Cytotoxin; Antibiotic; Antifungal; Apoptosis; Influenza Virus; MicroRNA; Topoisomerase |
T1174 | Topotecan hydrochloride | 119413-54-6 | 457.92 | 10mM | Apoptosis; Autophagy; Topoisomerase |
T1294 | Fleroxacin | 79660-72-3 | 369.34 | 10mM | Antibacterial; Antibiotic; DNA gyrase; Topoisomerase |
T1306 | Norfloxacin | 70458-96-7 | 319.34 | 10mM | Antibacterial; Antibiotic; DNA gyrase; Endogenous Metabolite; Topoisomerase |
T1492 | Gemifloxacin mesylate | 210353-53-0 | 485.49 | 10mM | Antibacterial; DNA gyrase; Topoisomerase |
T1521 | (±)-10-Hydroxycamptothecin | 64439-81-2 | 364.35 | 10mM | Topoisomerase |
T1523 | Teniposide | 29767-20-2 | 656.66 | 10mM | Topoisomerase |
T1620 | Pazufloxacin Mesylate | 163680-77-1 | 414.4 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T1625 | Lomefloxacin hydrochloride | 98079-52-8 | 387.81 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T1703 | SN-38 | 86639-52-3 | 392.4 | 10mM | ADC Cytotoxin; Autophagy; DNA/RNA Synthesis; Topoisomerase |
T2394 | Pixantrone dimaleate | 144675-97-8 | 557.21 | 10mM | Topoisomerase |
T2764 | (S)-10-Hydroxycamptothecin | 19685-09-7 | 364.36 | 10mM | Apoptosis; Topoisomerase |
T2830 | Betulinic acid | 472-15-1 | 456.71 | 10mM | Aminopeptidase; Apoptosis; Autophagy; Endogenous Metabolite; HIV Protease; Mitophagy; NF-κB; topoisomerase |
T3117 | Marbofloxacin | 115550-35-1 | 362.36 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T3181 | SW044248 | 522650-83-5 | 421.52 | 10mM | Topoisomerase |
T6010 | Idarubicin hydrochloride | 57852-57-0 | 533.95 | 10mM | Antibacterial; Antifungal; Autophagy; Topoisomerase |
T6336 | Amonafide | 69408-81-7 | 283.33 | 10mM | Topoisomerase |
T6407 | β-Lapachone | 4707-32-8 | 242.27 | 10mM | Apoptosis; Autophagy; IDO; Topoisomerase |
T6567 | Levofloxacin | 100986-85-4 | 361.37 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T6588 | Mitoxantrone | 65271-80-9 | 444.48 | 10mM | PKC; Topoisomerase |
T6628 | Pirarubicin | 72496-41-4 | 627.64 | 10mM | Antibacterial; Antibiotic; Autophagy; Topoisomerase |
T4614 | Ellipticine hydrochloride | 5081-48-1 | 282.76 | 10mM | Topoisomerase |
T4952 | 9-Hydroxycamptothecin | 67656-30-8 | 364.35 | 10mM | Topoisomerase |
T5394 | Prulifloxacin | 123447-62-1 | 461.46 | 10mM | Antibacterial; Antibiotic; Topoisomerase |
T5S1952 | 9-Methoxycamptothecin | 39026-92-1 | 378.38 | 10mM | Apoptosis; Topoisomerase |
T5820 | Amsacrine hydrochloride | 54301-15-4 | 429.92 | 10mM | Autophagy; Topoisomerase |
T5853 | Rubitecan | 91421-42-0 | 393.35 | 10mM | Topoisomerase |
T7309 | TAS-103 dihydrochloride | 174634-09-4 | 406.31 | 10mM | Topoisomerase |
T7551 | Belotecan hydrochloride | 213819-48-8 | 469.96 | 10mM | Topoisomerase |
T3S1957 | 9-amino-CPT | 91421-43-1 | 363.4 | 10mM | Topoisomerase |
TQ0063 | Zoliflodacin | 1620458-09-4 | 487.44 | 10mM | Antibacterial; DNA gyrase; DNA/RNA Synthesis; Topoisomerase |
TQ0088 | Exatecan Mesylate | 169869-90-3 | 531.55 | 10mM | Topoisomerase |
T22456 | Voreloxin hydrochloride | 175519-16-1 | 437.9 | 10mM | Apoptosis; Topoisomerase |
T8333 | Aurintricarboxylic acid | 4431-00-9 | 422.35 | 10mM | Apoptosis; Influenza Virus; MicroRNA; P2X Receptor; Topoisomerase |
T15507 | Hycanthone | 3105-97-3 | 356.48 | 10mM | DNA/RNA Synthesis; Parasite; Topoisomerase |
T26046 | Razoxane | 21416-67-1 | 268.27 | 10mM | Topoisomerase |
T36968 | ARN-21934 | 2230854-93-8 | 360.46 | 10mM | Topoisomerase |
T11872L | LMP744 hydrochloride | 308246-57-3 | 488.92 | 10mM | Topoisomerase |
T28475 | Pyrazoloacridine | 99009-20-8 | 367.4 | 10mM | Topoisomerase;Apoptosis |
T60123 | Chimmitecan | 185425-25-6 | 404.42 | 10mM | Topoisomerase |