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PKC inhibitor kit

Catalog No. CL0112

PKC inhibitor kit 包含蛋白激酶C PKC 抑制剂,在第二信使存在时,PKC 成为膜结合的酶,作用于细胞质中的酶和细胞核中的转录因子, 参与糖代谢、细胞分化、基因表达的调控与长时程抑制,如受体脱敏、调节膜结构、调节转录、介导免疫应答、调节细胞生长以及学习和记忆等。TargetMol 为您提供40种精选PKC 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

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PKC inhibitor kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,500 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
TN1299Desmethylglycitein17817-31-1270.210mMCDK; PI3K; PKC
T14072A-443654552325-16-3397.4710mMAkt; Casein Kinase; CDK; Chk; ERK; FLT; GSK-3; MAPK; PKA; PKC; S6 Kinase; Src; VEGFR
T4444A-674563 HCl (552325-73-2(free base))T4444394.910mMAkt; CDK; ERK; PKA; PKC
T7659Bisindolylmaleimide IV119139-23-0327.3410mMPKC
T10549Bisindolylmaleimide VIII acetate138516-31-1458.5110mMApoptosis; PKC
T6S0052Chelerythrine34316-15-9348.3710mMApoptosis; Autophagy; Bcl; PKC
T3684CP21R7125314-13-8317.310mMGSK-3; PKC
T0979Dequalinium chloride522-51-0527.5910mMPKC; Potassium Channel
T6280Enzastaurin170364-57-5515.6110mMApoptosis; Autophagy; PKC
T3060Fasudil hydrochloride105628-07-7327.8310mMAutophagy; Calcium Channel; HIV Protease; PKA; PKC; ROCK; Serine/threonin kinase
T6513Bisindolylmaleimide I133052-90-1412.4810mMPDGFR; PKC
T6313Go 6983133053-19-7442.5110mMPKC
T6285GSK-690693937174-76-0425.4810mMAkt; AMPK; Autophagy; PKC; Serine Protease
T27525HA-100491742-10-8293.3510mMPKA;PKC;Serine/threonin kinase
T5771Hypocrellin A77029-83-5546.5210mMAntibacterial; Parasite; PKC
T5600Darovasertib1874276-76-2472.4710mMPKC
T0033Miltefosine58066-85-6407.5810mMAkt; HIV Protease; PKC
T0158Mitoxantrone dihydrochloride70476-82-3517.410mMPKC; Topoisomerase
T9256N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine1071135-06-2388.5110mMPKC; Serine/threonin kinase
T0610Piceatannol10083-24-6244.2410mMApoptosis; Autophagy; PKA; PKC; Serine/threonin kinase; Syk
T3211Midostaurin120685-11-2570.6410mMPKC
T8764PKC-iota inhibitor 12328094-11-5374.410mMPKC
T9863PKCiota-IN-2 2230055-52-2395.4610mMPKC
T5817PKC-theta inhibitor2253640-49-0454.410mMPKC
T8376PKCβ inhibitor 1257879-35-9411.510mMApoptosis; PKC
T35827LPKCε Inhibitor Peptide acetateT35827L904.0210mMPKC
T5796Plantainoside D147331-98-4640.610mMPKC; RAAS
T60109Protein kinase inhibitor H-784477-87-2291.3710mMPKC
T6643Ro 31-8220 Mesylate138489-18-6553.6510mMPKC
T2356Ro-3306872573-93-8351.4510mMApoptosis; CDK; ERK; PKA; PKC; SGK
T16791Rottlerin82-08-6516.5410mMApoptosis; Autophagy; CaMK; HIV Protease; PKA; PKC
T9605Sangivamycin18417-89-5309.2810mMPKC;Nucleoside Antimetabolite/Analog
T6278Sotrastaurin425637-18-9438.4810mMPKC
T6680Staurosporine62996-74-1466.5310mMAntibacterial; Antibiotic; Antifungal; Apoptosis; PKA; PKC; Src
T4391Syk Inhibitor II (hydrochloride)227449-73-2413.2210mMBTK; PKC; Syk; Tyrosine Kinases
T2441TAS-301193620-69-8357.410mMPKC
T17148TPPB497259-23-1501.5410mMPKC
T7604Valrubicin56124-62-0723.6410mMAntibiotic; PKC
T13384LY-33075 dihydrochloride173897-44-4353.2510mMCaMK; PKC; ROCK
T35407Ζ-Stat3316-02-7384.3610mMPKC

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包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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