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PKA/cAMP inhibitor/activator kit

Catalog No. CL0143

PKA/cAMP inhibitor/activator kit 包含 PKA/cAMP 抑制剂/激活剂,G 蛋白偶联受体首先将信号传至腺苷酸环化酶,调节 cAMP 的含量,cAMP 决定PKA 的活性,PKA 负责很多蛋白的磷酸化,比如受体、离子通道、转录因子等,这是细胞快速应答胞外信号的过程。还有一类细胞缓慢应答胞外信号的过程,是cAMP 信号通路对细胞基因表达的影响。TargetMol 为您提供34种精选PKA/cAMP 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

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PKA/cAMP inhibitor/activator kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,500 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
T0465Ellagic acid476-66-4302.1910mMCarbonic Anhydrase; Casein Kinase; Endogenous Metabolite; Hedgehog/Smoothened; PKA; PKC; Reactive Oxygen Species; Syk; Topoisomerase
T0610Piceatannol10083-24-6244.2410mMApoptosis; Autophagy; PKA; PKC; Serine/threonin kinase; Syk
T0830Bithionol97-18-7356.0410mMcAMP; Parasite
T1418Bucladesine sodium16980-89-5491.3710mMPDE; PKA
T1920Capivasertib1143532-39-1428.9210mMAkt; Autophagy; mTOR; PKA
T2205Acefylline652-37-9238.210mMAdenosine Receptor; HDAC; PAD; PDE; PKA; TNF
T2244ESI-09263707-16-0330.7710mMcAMP; Virus Protease
T2356Ro-3306872573-93-8351.4510mMApoptosis; CDK; ERK; PKA; PKC; SGK
T2482AT131481056901-62-2313.7810mMAkt; PKA; ROCK; S6 Kinase; SGK
T2851Daphnetin486-35-1178.1410mMAutophagy; EGFR; Parasite; PKA; PKC
T3050ML-7 hydrochloride110448-33-4452.7410mMMyosin; PKA; PKC; Serine/threonin kinase; YAP
T3060Fasudil hydrochloride105628-07-7327.8310mMAutophagy; Calcium Channel; HIV Protease; PKA; PKC; ROCK; Serine/threonin kinase
T3269Metadoxine74536-44-0298.2910mM5-HT Receptor; PKA
T4444A-674563 HCl (552325-73-2(free base))T4444394.910mMAkt; CDK; ERK; PKA; PKC
T6250H-89 dihydrochloride130964-39-5519.2810mMAutophagy; PKA; S6 Kinase
T6304AT7867857531-00-1337.8510mMAkt; PKA; S6 Kinase
T6536HJC0350885434-70-8277.3810mMcAMP
T6680Staurosporine62996-74-1466.5310mMAntibacterial; Antibiotic; Antifungal; Apoptosis; PKA; PKC; Src
T67478-Bromo-cAMP sodium salt76939-46-3430.0810mMPKA
T4S2128Bilobetin521-32-4552.4910mMPKA; PPAR
T7648HA-10084468-24-6277.3410mMMyosin; PKA; PKC
T15485HJC01971383539-73-8339.4510mMcAMP; Ras
T14069A-3 hydrochloride78957-85-4321.2210mMCaMK; Casein Kinase; PKA; PKC
TN13347-Methoxyrosmanol113085-62-4360.4510mMcAMP
T6139LA-674563 2HCl(552325-73-2(fb-2hcl))T6139L431.3610mMAkt; CDK; ERK; PKA; PKC
T15247ESI-055184-64-5274.3810mMcAMP
TP1789LMalantide acetate(86555-35-3 free base)TP1789L1693.9710mMPKA; PKC
T12616LCE3F4143703-25-7351.0110mMcAMP
T15658KH7330676-02-3419.310mMAChR; cAMP
T21983LPKI 14-22 amide, myristoylated AcetateT21983L1269.5410mMPKA
T21674LPKA inhibitor fragment (6-22) amide AcetateT21674L1928.1110mMPKA
T9613TDI-10229T9613313.7910mMcAMP
T27525HA-100491742-10-8293.3510mMPKA;PKC;Serine/threonin kinase
T11212EPAC 5376753302826-61-5367.2110mMcAMP

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产品应用

  • 信号通路研究
  • 预实验探索

包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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