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Prostaglandin Receptor

Prostaglandin Receptor

Prostaglandin receptors or prostanoid receptors represent a sub-class of cell surface membrane receptors that are regarded as the primary receptors for one or more of the classical, naturally occurring prostanoids viz., prostaglandin D2, , PGE2, PGF2alpha, prostacyclin (PGI2), thromboxane A2 (TXA2), and PGH2.[1] They are named based on the prostanoid to which they preferentially bind and respond, e.g. the receptor responsive to PGI2 at lower concentrations than any other prostanoid is named the Prostacyclin receptor (IP). One exception to this rule is the receptor for thromboxane A2 (TP) which binds and responds to PGH2 and TXA2 equally well.
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Cat. No. Product Name CAS No. Purity Chemical Structure
T3P2855 Chamigrenal
恰米醛
19912-84-6
β-Chamigrenal has anti-inflammatory activity, it has inhibitory effects on lipopolysaccharide-induced nitric oxide and prostaglandin E2 production in RAW 264.7 m...
TN1109 3-O-Acetyl-16α-hydroxydehydrotrametenolic acid
3-O-乙酰基-16Α-羟基松苓新酸
168293-14-9
3-O-Acetyl-16α-hydroxydehydrotrametenolic acid (3-O-Acetyl-16 alpha-hydroxydehydrotrametenolic acid) 是三萜类化合物。它能够作用于 LPS 刺激的 Raw264.7 细胞,减少NO 产生和 iNOS 表达,具有消炎作用。
TN4592 Murrangatin
化合物 TN4592
37126-91-3 98%
Murrangatin may be a valuable anti-tumor-promoting agent, it can significantly inhibit Epstein-Barr virus early antigen (EBV-EA) activation, and preserve the hig...
TN5248 Voleneol
化合物 TN5248
70389-88-7 98%
1β,6α-Dihydroxyeudesm-4(15)-ene (Voleneol,DE) can attenuate the lipopolysaccharide (LPS)-induced inflammation in BV2 microglial cells, it also can dose-dependent...
TN3366 Ailanthoidol
化合物 TN3366
156398-61-7 98%
Ailanthoidol has anti-inflammatory activity, it inhibits inflammatory reactions by macrophages and protects mice from endotoxin shock. It also possesses potentia...
T13488 2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
化合物 T13488
137089-36-2 98%
2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide is a compound that inhibits stress-induced ulcer. It can maintain the content of phospholipase A2 and pros...
T4484 1,7-Dihydroxy-2,3-methylenedioxyxanthone
1,7-二羟基-2,3-亚甲二氧基呫吨酮
183210-63-1 98%
1,7-Dihydroxy-2,3-methylenedioxyxanthone has antiulcerogenic, anti-oxidation, and antihyperalgesic activities, it can inhibit the carrageenan-induced hyperalgesi...
T14500 BAY-1316957
化合物 T14500
1613264-40-6 98%
BAY-1316957 is a highly potent and selective EP4 receptor antagonist. With an IC50 of 15.3 nM. Good oral bioavailability[1].
T78582 15-keto-Prostaglandin E2
化合物 15-keto-Prostaglandin E2
26441-05-4 98%
15-keto-Prostaglandin E2为内源性代谢产物,通过与STAT3Cys259残基结合,抑制STAT3激活作用。该化合物能够结合并稳定EP2与EP4受体,进而抑制乳腺癌细胞生长与进展,并通过激活PPAR-γ促进真菌生长。
T78584 Prostaglandin D3
化合物 Prostaglandin D3
71902-47-1 98%
Prostaglandin D3 (PGD3) 是具有抑制人类血小板聚集和调节自主神经传递功能的前列腺素类化合物。
T78710 AMX12006
化合物 AMX12006
2639775-01-0 98%
AMX12006为一种口服活性EP4拮抗剂,显示出高度的选择性与有效性,IC50为4.3 nM,并具备细胞毒性和抗肿瘤活性。
T79432 NXT-10796
化合物 NXT-10796
98%
NXT-10796为具口服活性且肠道限制性EP4受体激动剂。
TN4465 Luvangetin
化合物 TN4465
483-92-1 98%
Luvangetin may have anti-inflammatory activity, it can inhibit NO and PGE2 production in LPS-stimulated BV2 cells. Luvangetin shows significant protection agains...
TN4038 Eupatolide
泽兰内酯
6750-25-0 98%
Eupatolide 是从 Inula japonica 的花中分离出来的,具有抗炎活性。 Eupatolide 可用于研究乳腺癌细胞对 TRAIL 的耐药性。
TN3587 Capillarisin
化合物 TN3587
56365-38-9 98%
Capillarisin is a novel blocker of STAT3 activation and thus may have a potential in negative regulation of growth, metastasis, and chemoresistance of tumor cell...
T16388 Omidenepag isopropyl
化合物 T16388
1187451-19-9 98%
Omidenepag isopropyl is converted to the active product Omidenepag during corneal penetration. Omidenepag isopropyl is a selective EP2 receptor agonist. Omidenep...
TN5033 Skullcapflavone I
化合物 TN5033
41060-16-6 98%
Skullcapflavone I has anti-inflammatory and anti-allergic potential, it can significantly inhibit LPS stimulated NO and PGE(2) release in J774A.1 macrophages and...
TN1485 Chicanine
襄五脂素
78919-28-5 98%
Chicanine has anti-inflammatory activity in macrophages by down-regulating LPS-induced inflammatory cytokines in IκBα±/MAPK/ERK signaling pathways.
T16011 Manumycin A
手霉素A
52665-74-4 98%
Manumycin A is an antibiotic. Manumycin A induces apoptosis and exerts antitumor activity. Manumycin A inhibits exosome biogenesis and secretion via targeted inh...
T14842 BW 245C
化合物 BW 245C
72814-32-5 98%
BW 245C 是一种选择性的前列腺素类DP受体(DP1)激动剂,是一种前列腺素类似物,对胶原蛋白的聚集反应有抑制作用,可用于研究中风等疾病。
Chamigrenal
T3P2855
β-Chamigrenal has anti-inflammatory activity, it has inhibitory effects on lipopolysaccharide-induced nitric oxide and prostaglandin E2 production in RAW 264.7 m...
3-O-Acetyl-16α-hydroxydehydrotrametenolic acid
TN1109
3-O-Acetyl-16α-hydroxydehydrotrametenolic acid (3-O-Acetyl-16 alpha-hydroxydehydrotrametenolic acid) 是三萜类化合物。它能够作用于 LPS 刺激的 Raw264.7 细胞,减少NO 产生和 iNOS 表达,具有消炎作用。
Murrangatin
TN4592
Murrangatin may be a valuable anti-tumor-promoting agent, it can significantly inhibit Epstein-Barr virus early antigen (EBV-EA) activation, and preserve the hig...
Voleneol
TN5248
1β,6α-Dihydroxyeudesm-4(15)-ene (Voleneol,DE) can attenuate the lipopolysaccharide (LPS)-induced inflammation in BV2 microglial cells, it also can dose-dependent...
Ailanthoidol
TN3366
Ailanthoidol has anti-inflammatory activity, it inhibits inflammatory reactions by macrophages and protects mice from endotoxin shock. It also possesses potentia...
2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
T13488
2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide is a compound that inhibits stress-induced ulcer. It can maintain the content of phospholipase A2 and pros...
1,7-Dihydroxy-2,3-methylenedioxyxanthone
T4484
1,7-Dihydroxy-2,3-methylenedioxyxanthone has antiulcerogenic, anti-oxidation, and antihyperalgesic activities, it can inhibit the carrageenan-induced hyperalgesi...
BAY-1316957
T14500
BAY-1316957 is a highly potent and selective EP4 receptor antagonist. With an IC50 of 15.3 nM. Good oral bioavailability[1].
15-keto-Prostaglandin E2
T78582
15-keto-Prostaglandin E2为内源性代谢产物,通过与STAT3Cys259残基结合,抑制STAT3激活作用。该化合物能够结合并稳定EP2与EP4受体,进而抑制乳腺癌细胞生长与进展,并通过激活PPAR-γ促进真菌生长。
Prostaglandin D3
T78584
Prostaglandin D3 (PGD3) 是具有抑制人类血小板聚集和调节自主神经传递功能的前列腺素类化合物。
AMX12006
T78710
AMX12006为一种口服活性EP4拮抗剂,显示出高度的选择性与有效性,IC50为4.3 nM,并具备细胞毒性和抗肿瘤活性。
NXT-10796
T79432
NXT-10796为具口服活性且肠道限制性EP4受体激动剂。
Luvangetin
TN4465
Luvangetin may have anti-inflammatory activity, it can inhibit NO and PGE2 production in LPS-stimulated BV2 cells. Luvangetin shows significant protection agains...
Eupatolide
TN4038
Eupatolide 是从 Inula japonica 的花中分离出来的,具有抗炎活性。 Eupatolide 可用于研究乳腺癌细胞对 TRAIL 的耐药性。
Capillarisin
TN3587
Capillarisin is a novel blocker of STAT3 activation and thus may have a potential in negative regulation of growth, metastasis, and chemoresistance of tumor cell...
Omidenepag isopropyl
T16388
Omidenepag isopropyl is converted to the active product Omidenepag during corneal penetration. Omidenepag isopropyl is a selective EP2 receptor agonist. Omidenep...
Skullcapflavone I
TN5033
Skullcapflavone I has anti-inflammatory and anti-allergic potential, it can significantly inhibit LPS stimulated NO and PGE(2) release in J774A.1 macrophages and...
Chicanine
TN1485
Chicanine has anti-inflammatory activity in macrophages by down-regulating LPS-induced inflammatory cytokines in IκBα±/MAPK/ERK signaling pathways.
Manumycin A
T16011
Manumycin A is an antibiotic. Manumycin A induces apoptosis and exerts antitumor activity. Manumycin A inhibits exosome biogenesis and secretion via targeted inh...
BW 245C
T14842
BW 245C 是一种选择性的前列腺素类DP受体(DP1)激动剂,是一种前列腺素类似物,对胶原蛋白的聚集反应有抑制作用,可用于研究中风等疾病。
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