首页AutophagyProtease-activated Receptor
Protease-activated Receptor
T1893 ML 161 ML 161 is the inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC50: 0.26 μM for the inhibition of platelet P-selectin expression on human platelets
T1986L Atopaxar Hydrobromide Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute
T3098 Vorapaxar sulfate Vorapaxar sulfate is a potent and orally active thrombin receptor (PAR-1) antagonist.
T4186 AC264613 AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 production by lipopoly
T7013 Vorapaxar Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).
T7137 I-191 I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
T7380 Protease-Activated Receptor-4 Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4)  agonist, with Antiplatelet Therapy
T7496 Thrombin Receptor Activator for Peptide Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of coronary heart disease
T7513 Protease-Activated Receptor-2, amide Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M)
T7573 TFLLR-NH2(2TFA) TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T7573L TFLLR-NH2 2TFA(197794-83-5(free base)) TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T7623 PAR-4 Agonist Peptide, amide PAR-4 Agonist Peptide, amide is an agonist of proteinase-activated receptor-4 (PAR-4).
T7625 TRAP-6(2TFA) TRAP-6(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
T7674 Thrombin Receptor Activator for Peptide Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of coronary heart disease
T7740 Protease-Activated Receptor-4 diTFA(245443-52-1(free base)) Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
T8917 IUN76750 IUN76750 is a PAR-​2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
T8917 IUN76750 IUN76750 is a PAR-​2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
TP1046L PAR-2 Activating Peptide acetate(171436-38-7 free base) PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2).
TP1046L PAR-2 Activating Peptide acetate(171436-38-7 free base) PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2).
TP1065 PAR-4 Agonist Peptide, amide TFA PAR-4 Agonist Peptide, amide TFA is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked by a PAR-4 antagon
TP1378 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) 2-Furoyl-LIGRLO-amide is a potent and selective protease-activated receptor 2 (PAR2) agonist.
TP1904L FSLLRY-NH2 TFA(245329-02-6 free base) FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK
TP1925L tcY-NH2 TFA(327177-34-4 free base) tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
TQ0012 AZ3451 AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
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