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NMDAR
T0051 Urethane Urethane was an antineoplastic agent .Now is used for other medicinal purposes.
T0349 Riluzole Riluzole is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMYOTROPHIC LATERAL SCLEROSIS.
T0802 Procaine hydrochloride Procaine Hydrochloride is the hydrochloride salt form of procaine, a benzoic acid derivative with local anesthetic and antiarrhythmic properties. Procaine binds to and inhibi
T0954 Anestan Halothane is a nonflammable, halogenated, hydrocarbon anesthetic that provides relatively rapid induction with little or no excitement. Analgesia may not be adequate. NITROUS OXIDE
T1186 Ifenprodil Tartrate Ifenprodil is a selective NMDA receptor (glutamate) antagonist.
T1308 Orphenadrine hydrochloride Orphenadrine hydrochloride is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
T1324 Phosphoserine Phosphoserine is the phosphoric acid ester of serine.
T1443 Memantine hydrochloride Memantine hydrochloride is an AMANTADINE derivative that has some dopaminergic effects. Memantine hydrochloride has been proposed as an antiparkinson agent.
T1751 Eliprodil Eliprodil(SL-820715), a non-competitive NR2B-NMDA receptor antagonist(IC50: 1 uM), less effective for NR2A- and NR2C-containing receptors(IC50> 100 uM). It has been used in trials
T1897 MDL 29951 MDL-29951 is a novel glycine antagonist of NMDA receptor activation.
T1909 L701324 L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.
T1946 Felbamate Felbamate is an Anti-epileptic Agent. The physiologic effect of felbamate is by means of Decreased Central Nervous System Disorganized Electrical Activity.
T2362 QNZ46 QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.
T3320 Dizocilpine Maleate (+)-MK-801 is a potent noncompetitive antagonist of the NMDA receptor (RECEPTORS, N-METHYL-D-ASPARTATE) with Kd of 37.2 nM in rat brain membranes. The drug has been considered fo
T4171 PEAQX PEAQX(NVP-AAM 077) is an effective and orally available NMDA antagonist. It can inhibit human NMDA receptors for 1A/2A(IC50: 270 nM), rather than 1A/2B(29, 600 nM).
T4225 Dextrorphan tartrate Dextrorphan D-tartrate is a noncompetitive NMDA glutamate receptor antagonist.
T6259 Dizocilpine MK-801 (Dizocilpine) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.
T6504 Flupirtine maleate Flupirtine maleate, a centrally acting non-opioid analgesia, is the salt form of Flupirtine. It is an NMDA receptor antagonist , and also a specific neuronal potassium channel open
T6608 NMDA N-Methyl-D-aspartic acid is an amino acid that, as the D-isomer, is the defining agonist for the NMDA receptor subtype of glutamate receptors.
T6975 Sarcosine Sarcosine is a competitive inhibitor of the type I glycine transporter (GlyT1) and an N-methyl-D-aspartate receptor (NMDAR) co-agonist.
T4096 Quinolinic acid Quinolinic acid is an endogenous N-methyl-D-aspartate (NMDA) receptor agonist synthesized from L-tryptophan via the kynurenine pathway.
T4979 Procyclidine hydrochloride Procyclidine is a potent anticholinergic agent and also have NMDA antagonist properties.
T5385 Radiprodil Radiprodil (RGH-896) is an orally active and selective NMDA NR2B receptors antagonist. It was a potential treatment of neuropathic pain associated with diabetic peripheral neuropat
T4885 D-Aspartic acid D-Aspartic acid (D-Asp) is an endogenous amino acid existing in invertebrates and vertebrates. It can regulate testosterone synthesis and is an agonist of NMDA receptor.
T4752 1-Aminocyclopropanecarboxylic acid 1-Aminocyclopropanecarboxylic acid (ACPC) is an intermediate in the synthesis of ethylene, the plant hormone responsible for biological processes ranging from seed germination to o
T5080 Spermidine hydrochloride Spermidine, a natural polyamine, is a novel autophagy inducer and negatively modulates N-methyl-d-aspartate (NMDA).
T5819 Rapastinel Trifluoroacetate Rapastinel Trifluoroacetate is an NMDA receptor modulator with glycine-site partial agonist properties.
TQ0027 Transcrocetinate disodium Transcrocetinate disodium, extracted from saffron (Crocus sativus L.), is a high-affinity antagonist of NMDA receptor.
TQ0233 Traxoprodil Traxoprodil (CP101,606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).
TQ0279 Ibotenic acid Ibotenic acid has agonist activity at both the NMDA and trans-ACPD or metabotropic quisqualate receptors.
T7778 Glypromate Glypromate is a neuroprotective agent, is a weak NMDA receptor agonist
T3486 3-MATIDA
T7867 Flutriafol Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist
T7870 TCN-201 TCN-201 is a selective antagonist of NMDA receptors containing the NR2A subunit.
T8394 (R)-Serine (R)-Serine is an endogenous amino acid,is a potent co-agonist at the NMDA glutamate receptor.
TN1420 Bacopaside I Bacopaside I is a modulator of Aquaporin-1 channel, has neuroprotective functions, it has anti-Alzheimer's disease, it ameliorates cognitive impairment in APP/PS1 mice via immune-m
TN1432 Bacopasaponin C Bacopasaponin C may have antioxidant activity, it also shows anti-leishmanial property.
T8351 UBP551 UBP551 is a potent and selective NMDA receptors modulator.
T16332 NKH477 NKH477 is a novel water-soluble forskolin derivative that improves cardiac failure mainly through its beneficial effects on diastolic cardiac function. NKH477 shows an antiprolifer
T16473 Perzinfotel Perzinfotel displays high affinity (IC50=30 nM) for the glutamate site. Perzinfotel is an effective, selective, and competitive NMDA receptor antagonist with neuroprotective effect
T8626 4-oxo-1,4-dihydroquinoline-2-carboxylic acid 4-oxo-1,4-dihydroquinoline-2-carboxylic acid is a GluR and NMDA inhibitor.
TN2641 15-Methoxypinusolidic acid 15-Methoxypinusolidic acid has anti-inflammatory effects, it inhibits LPS-induced iNOS expression and NO production, independent on MAPK and NF-kappaB. 15-Methoxypinusolidic acid s
TN5263 1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one Xanthohumol has anti-hepatitis C virus, anti-carcinogenic, free radical-scavenging, and anti-inflammatory activities, it can inhibit HIV-1 induced cytopathic effects, the productio
T0556 6-Methoxy-2-naphthoic acid 6-Methoxy-2-naphthoic acid is an modulator of NMDAR.
T8450 TCN213 TCN213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over NR1/NR2B
T6352 (-)-MK 801 Maleate MK-801 is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.
T22733 DL-AP5 NMDA antagonist
T0015 Mephenesin Mephenesin is a centrally acting muscle relaxant with a short duration of action.
T0015 Mephenesin Mephenesin is a centrally acting muscle relaxant with a short duration of action.
T17293 ZL006 ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.
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