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MAO
T0084 Moclobemide Moclobemide is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties.
T0235 Modaline sulfate Modaline was a 2-methyl-3-piperidinopyrazine derivative found to inhibit monoamine oxidase (MAO) and showed a curative effect for the anti-depressant. Similar to other MAO inhibito
T0300 Pargyline Pargyline is a monoamine oxidase inhibitor with antihypertensive properties.
T0338 Minaprine Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
T0369 Ethaverine hydrochloride Ethaverine hydrochloride is a homologue of papaverine.
T0391 Linezolid Linezolid, the first of the oxazolidinone class, is a synthetic antibiotic used for the therapy of infections resulted from multi-resistant bacteria including methicillin-resistant
T0418 Allylthiourea Allylthiourea, a metabolic inhibitor, specifically suppresses ammonia oxidation.
T0751 Furazolidone Furazolidone, a nitrofuran derivative, inhibits AML1-ETO transformed cells with IC50 value of 12.7 μM. It is antibacterial and antiprotozoal activity,
T0821 Iproniazid Phosphate Iproniazid is a non-selective, irreversible monoamine oxidase inhibitor (MAOI).
T0966 Sennoside A Sennoside A, a kind of irritant laxative isolated from rhei rhizome, causes purgative actions in the intestine.
T10079 MAO-IN-1 MAO-IN-1 is an inhibitor of monoamine oxidase B (MAO B; IC50: 20 nM).
T10146 4-Hydroxyderricin 4-Hydroxyderricin, the major active ingredients of Angelica keiskei Koidzumi, is a potent selective MAO-B inhibitor (IC50: 3.43 μM). It also mildly inhibits DBH (dopamine β-hydro
T1025 Tranylcypromine (2-PCPA) hydrochloride Tranylcypromine Hydrochloride, a monoamine oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and atypical depression. It is a propylamine fo
T10617 Brofaromine Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).
T1117 Clorgyline hydrochloride Clorgyline hydrochloride, a white powder, is served as monoamine oxidase inhibitor.
T1119 Rasagiline Rasagiline is an inhibitor of monamine oxidase used as adjunctive therapy in combination with levodopa and carbidopa in the management of Parkinsons disease.
T1455 Nialamide Nialamide is an MAO inhibitor that is used as an antidepressive agent.
T15010 CR4056 CR4056 is a selective inhibitor of human recombinant MAO-A (IC50: 202.7 nM) and a ligand of the imidazoline-2 receptor (I2R) (IC50: 596 nM).
T15023 CX-157 CX-157 is a reversible monoamine oxidase-A (MAO-A) inhibitor (EC50:19.3 ng/mL).
T1549 Raloxifene hydrochloride Raloxifene hydrochloride is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women. It has estrogen agonist effects o
T1578 Pargyline hydrochloride Pargyline hydrochloride is an irreversible monoamine oxidase(MAO) inhibitor with antihypertensive properties.
T1613 Hydralazine hydrochloride Hydralazine Hydrochloride is the hydrochloride salt of hydralazine, a phthalazine derivative with antihypertensive and potential antineoplastic activities. Hydralazine alters intra
T16770 Ro 41-1049 hydrochloride Ro 41-1049 hydrochloride is a reversible and selective inhibitor of monoamine oxidase-A (Kd: 16.5 and 64.4 nM, respectively).
T1711 Harmine Harmine is an alkaloid isolated from seeds of Peganum harmala.
T1747 Torezolid Tedizolid is an Oxazolidinone Antibacterial. The mechanism of action of tedizolid is as a Breast Cancer Resistance Protein Inhibitor.
T2741 Glycyrrhizin Glycyrrhizic acid is a triterpenoid saponinl with anti-tumor and anti-diabetic activities.
T2765 Rosmarinic acid Rosmarinic acid has shown to contain antioxidant, anti-inflammatory and antimicrobial activities. Possesses promising physiological actions related to cognitive performance, Alzhei
T2900 Paeonol Paeonol is an active extraction from Paeonia suffruticosa. Paeonol inhibits MAO-A and MAO-B with IC50 of 54.6 μM and 42.5 μM, respectively.
T3095 Tyramine Tyramine is an indirect sympathomimetic that occurs naturally in cheese and other foods. Tyramine does not directly activate adrenergic receptors, but it can serve as a substrate f
T3596 TB5 TB5 is a potent, selective and reversible inhibitor of hMAO-B.
T3933 Jatrorrhizine Jatrorrhizine is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species. It was found to have antimicrobial and antifungal activity. It binds and
T5050 Selegiline hydrochloride Selegiline hydrochloride is a selective, reversible inhibitor of MAO-B (Ki = 0.091 μM) over MAO-A (Ki = 9.06 μM). Monoamine oxidase (MAO) inhibitors have utility in ameliorating
T5053 Eprobemide Eprobemide is a non-competitive reversible inhibitor of monoamine oxidase A (MAO-A).
T5323 MD 69276 MD 69276 (Toloxatone) is a reversible monoamine oxidase A (MAOA) inhibitor.
T5470 LAZABEMIDE LAZABEMIDE(Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively).
T5648 Purpurin Purpurin was a reversible and competitive inhibitor of MAO-A with a Ki value of 0.422μM. it exhibits anti-angiogenic, antifungal, antibiotic, and antioxidative activities.
T5676 (Z)-SU4312 (Z)-SU4312 is a inhibitor of MAO-B and NOS(IC50 value of 0.2 μM, 19.0μM,respectively).
T5678 N-(2-Aminoethyl)-5-chlor-2-pyridincarbox N-(2-Aminoethyl)-5-chlor-2-pyridincarbox is a reversible and selective mao-b inhibitor(Ki:7.9nM).
T5887 3,4-Dihydro-7-hydroxy-2(1H)-quinolinone 3,4-Dihydro-7-hydroxy-2(1H)-quinolinone (7-​Hydroxy-​3,​4-​dihydro-​2(1H)​-​quinolinone) is a weak MAO-A inhibitor(with an IC50 of 183 μM) .
T6651 Safinamide mesylate Safinamide Mesylate, a mesylate salt of Safinamide, can reversibly and specifically inhibit MAO-B (IC50: 98 nM), has 5918-fold selectivity against MAO-A.
T6862 Isatin Isatin is an endogenous MAO inhibitor.
T6962 Rasagiline Mesylate Rasagiline Mesylate is a novel MAO-B inhibitor, which can treat idiopathic Parkinson's disease.
T7048 1,4-Naphthoquinone 1, 4-Naphthoquinone was used as a potential inhibitor of monoamine oxidase and DNA topoisomerase activities[2]. It was also used to inhibit the acetyltransferase activity[1].
T7942 Tranylcypromine (hemisulfate) Tranylcypromine is an inhibitor of monoamine oxidase (MAO) and lysine-specific demethylase 1 (LSD1)  with a rapid onset of activity.
T8589 Amiflamine Amiflamine is an inhibitor of reversible MAO-A.
T8849 PF-9601N PF-9601N showed high potency and selectivity as a MAO-BI (monoamine oxidase type B inhibitor) and also demonstrated remarkable neuroprotective properties in several in vivo and cel
T8907 Minaprine dihydrochloride Minaprine dihydrochloride is a reversible MAO-A inhibitor; It weakly inhibit acetylcholinesterase. Minaprine dihydrochloride is an antidepressant for treatment of depression.
TMS1743 Salvigenin Salvigenin is a potent hMAO-A inhibitor, has neuroprotective, antitumor and immunomodulatory effects.
TN1099 Dihydroevocarpine Dihydroevocarpine shows potent anti-Helicobacter pylori activity with the minimum inhibitory concentration (MIC) value of 10-20 microg/ml. Dihydroevocarpine is a moderate modulator
TN1120 Osthenol Osthenol is a natural product, and is selective, reversible, and competitive human monoamine oxidase-A (hMAO-A) inhibitor (Ki=0.26 µM).It shows antitumor-promoting activity, it al
TN1705 Glycyrrhisoflavone Glycyrrhisoflavone is a tyrosinase inhibitor, it also shows inhibitory effects on monoamine oxidase.
TN2553 1-Methyl-2-undecylquinolin-4(1H)-one 1-Methyl-2-undecyl-4(1H)-quinolone, and dihydroevocarpine should also be served as the chemical markers together with evodiamine for the quality control of Evodia rutaecarpa (Juss.
TN2790 2'-O-Methylperlatolic acid 2'-O-Methylperlatolic acid and confluentic acid are monoamine oxidase B inhibitors in a Brazilian plant, Himatanthus sucuuba.
TN3024 4'-Demethyleucomin
TN3116 5-Hydroxy-1-methoxyxanthone 5-Hydroxy-1-methoxyxanthone, 1,5-dihydroxyxanthone and 6-deoxyjacareubin are all antifungal against Cladosporium cucumerinum, while they show differing degrees of inhibition of mon
TN3294 8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate 8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes.
TN3300 8alpha-Tigloyloxyhirsutinolide 13-O-acetate 8alpha-Tigloyloxyhirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes. 8alpha-Tigloyloxyhirsutinolide 13-O-acetate has anti-cancer activit
TN3726 Cudraflavone B Cudraflavone B has anti-proliferative activity, mouse brain monoamine oxidase (MAO) inhibitory effects, apoptotic actions in human gastric carcinoma cells and mouse melanoma cells,
TN3918 Echitovenidine Echitovenidine shows monoamine oxidase inhibitor activity.
TN4137 Glicoricone Glicoricone acts as a partial estrogen antagonist. Glicoricone inhibited the monoamine oxidase with the IC50 values of 6.0 x 10(-5)-1.4 x 10(-4) M.
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