Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T0246L | Betahistine mesylate
甲磺酸倍他司汀
|
54856-23-4 | 99.83% |
|
Betahistine mesylate (Extovyl) 是可口服的组胺 H1 受体激动剂和 H3 受体的拮抗剂,可用作血管扩张剂,用于类风湿性关节炎的研究。 | ||||
T13566 | Bamirastine
巴麦斯汀
|
215529-47-8 | 96.68% |
|
Bamirastine 抑制配体结合到重组人组胺 H1 受体 (rhH1R),IC50 值为 17.3 nM。Bamirastine 对过敏性皮肤炎症有抑制作用。 | ||||
T61213 | PF-03654764
化合物PF-03654764
|
935840-35-0 | 100% |
|
PF-03654764 是一种具有口服活性、高效性和选择性的组胺 H3 受体拮抗剂,对人 H3 和大鼠 H3 具有抑制作用, Ki 值分别为 1.2 nM 和 7.9 nM。PF-03654764 常与 Fexofenadine 一起联合用药来治疗过敏性鼻炎。 | ||||
TN3699 | Corchoionoside C
化合物 TN3699
|
185414-25-9 | 98% |
|
Corchoionoside C has antioxidant activity, shows strong scavenging activities on DPPH radical, it also shows weak antifungal activity. Corchoionosides A, B, and ... | ||||
T10770 | Cetirizine D8
化合物 T10770
|
774596-22-4 | 98% |
|
Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist. | ||||
T77715 | H4R antagonist 3
H4R拮抗剂3
|
1003091-20-0 | 98% |
|
H4R antagonist 3 是一种新型组胺-4受体 (H4R)拮抗剂,EC50 <10 mM。H4R antagonist 3 具有潜在的炎性活性,可用于研究自身免疫性、过敏性和眼部疾病。 | ||||
T78126 | Dothiepin
度硫平
|
113-53-1 | 98% |
|
Dothiepin(Dosulepin; Dothep)是一种具备镇静/抗焦虑作用的抗抑郁药物。该化合物主要通过抑制去甲肾上腺素的再摄取,而非血清素,以增强去肾上腺素能神经传递。同时,Dothiepin作为组胺H1受体的拮抗剂,具备显著的镇痛活性,适用于治疗心因性面部疼痛、特发性纤维肌痛综合征或类风湿关节炎,并且不具有心... | ||||
T79786 | H4R antagonist 2
化合物 H4R antagonist 2
|
1148115-99-4 | 98% |
|
H4R antagonist 2 是Furo[3,2-d]嘧啶衍生的有效H4R拮抗剂,主要用于类风湿性关节炎的研究。 | ||||
T80645 | 4-Methylhistamine
化合物 4-Methylhistamine
|
36507-31-0 | 98% |
|
4-Methylhistamine 作为一种有效的组胺 4 受体 (H4R) 激动剂,显示出在研究免疫相关疾病,如癌症和自身免疫性疾病方面的应用潜力。 | ||||
T11729 | JTE-952
化合物 T11729
|
1255303-54-8 | 98% |
|
JTE-952 is a oral, potent active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), wit... | ||||
T15590 | Iodophenpropit dihydrobromide
化合物 T15590
|
145196-87-8 | 98% |
|
Iodophenpropit dihydrobromide is an effective and selective antagonist of the histamine H3 receptor. The binding of [125I]Iodophenpropit is readily reversible, s... | ||||
TN3483 | Bakkenolide D
化合物 TN3483
|
18456-03-6 | 98% |
|
Bakkenolide D has anti-allergic effect, it and bakkenolide D demonstrates inhibitory effect on the trachea contraction induced by histamine in vitro, they have o... | ||||
T12630 | (R)-(-)-α-Methylhistamine dihydrobromide
(R)(−)-α-甲基组胺 二盐酸盐
|
868698-49-1 | 98% |
|
(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM). | ||||
TN2155 | Rhodiocyanoside A
化合物Rhodiocyanoside A
|
168433-86-1 | 98% |
|
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP ... | ||||
T11088 | Doxepin D3 Hydrochloride
化合物 T11088
|
347840-07-7 | 98% |
|
Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin... | ||||
T15722 | Lavoltidine
化合物 T15722
|
76956-02-0 | 98% |
|
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hyperg... | ||||
T17118 | Toreforant
化合物 T17118
|
952494-46-1 | 98% |
|
Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM). | ||||
T12416 | PF-03654746 Tosylate
化合物 T12416
|
1039399-17-1 | 98% |
|
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration. | ||||
T12703 | ReN-1869 hydrochloride
化合物 T12703
|
170149-76-5 | 98% |
|
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor. | ||||
T19443L | N-Acetylhistamine acetate
化合物N-Acetylhistamine acetate
|
98% |
|
|
N-Acetylhistamine acetate 是一种组胺代谢物。 它可用作过敏反应的组氨酸代谢的潜在生物标志物。 |