||Dantrolene sodium salt
||Dantrolene is a skeletal muscle relaxant and can interfere with excitation-contraction coupling in the muscle fiber. It is used for the treatment of spasticity and other neuromuscu
||Diltiazem Hydrochloride is a benzothiazepine calcium channel blocking agent with vasodilating action due to its antagonism of the actions of CALCIUM ion on membrane functions.
||Nitrendipine is a calcium channel blocker with marked vasodilator action. It is an effective antihypertensive agent and differs from other calcium channel blockers in that it does
||Azelnidipine is a dihydropyridine used as calcium channel blocker.
||Felodipine is a longlasting 1,4-dihydropyridine calcium channel repressor.
||Nisoldipine is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent.
||Levetiracetam is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onset seizures. Levetiracetam has been li
||Manidipine dihydrochloride is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).
||Ranolazine(RS-43285), an antianginal agent, can treat arrhythmia via a novel mechanism of action (inhibition of the late phase of the inward sodium current), and do not affect bloo
||Amlodipine Besylate is a long-lasting calcium channel blocker.
||Zonisamide, a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures. It may inhibit a carbonic anhydrase although this is
||Trimethadione is a dione-type anticonvulsant with antiepileptic activity.
||Fendiline is a non-selective blocker of calcium channel.
||Nimodipine, a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.
||Cilnidipine(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.
||Gabapentin is a GABA analogue, used to treat seizures and neuropathic pain.
||Ethosuximide is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied by other types of seizures.
||Flunarizine is a selective calcium entry blocker with calmodulin binding properties and histamine H1 blocking activity. Flunarizine hydrochloride is effective in the prophylaxis of
||Cinnarizine is a piperazine derivative having histamine H1-receptor and calcium-channel blocking activity with vasodilating and antiemetic properties but it induces PARKINSONIAN DI
||Isradipine is a dihydropyridine calcium channel blockers with antihypertensive and vasodilator activities. Isradipine blocks the calcium entry through the calcium ion channels of c
||Clevidipine is a dihydropyridine L-type calcium channel blocker that is selective for vascular smooth muscle and is indicated for blood pressure reduction when oral therapy is not
||Verapamil hydrochloride is a calcium channel blocker that is a class IV anti-arrhythmia agent.
||Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
||Nifedipine is a dihydropyridine calcium channel blocking agent. Nifedipine inhibits the transmembrane influx of extracellular calcium ions into myocardial and vascular smooth muscl
||Trimebutine maleate is a weak mu-opioid agonist and has antimuscarinic effects. Trimebutine is an agonist of peripheral mu, delta, and kappa opiate receptors served as a spasmolyti
||Nicardipine Hydrochloride is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nicardipine (Nifedipine
||An anticonvulsant that is the active metabolite of TRIMETHADIONE.
||Amlodipine is a synthetic dihydropyridine and a calcium channel blocker with antihypertensive and antianginal properties.
||Nilvadipine, a calcium channel blocker (CCB), is utilized for treatment of hypertension.
||Praziquantel increases the permeability of the tegument of susceptible worms, resulting in an influx and increase in intra-tegumental calcium leading to rapid contractions and para
||Lacidipine is a lipophilic dihydropyridine calcium antagonist with an intrinsically slow onset of activity. Due to its long duration of action, lacidipine does not lead to reflex t
||Otilonium Bromide, an antimuscarinic, is utilized as a spasmolytic agent.
||Levamlodipine belongs to the dihydropyridine group of calcium channel blockers. Levamlodipine, also known as S-amlodipine, is a pharmacologically active enantiomer of amlodipine, a
||Strontium ranelate, a strontium (II) salt of the ranelic acid, is a medication for osteoporosis. Studies indicate it can also slow the course of osteoarthritis of the knee. The dru
||NPS-2143 is a novel potent and selective antagonist of Ca(2+) receptor.
||Efonidipine(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.
||Lercanidipine is a calcium channel blocker of the dihydropyridine class.
||1-Ethyl-2-benzimidazolinone is a calium channel agonist.
||Tetrandrine is a natural, bis-benzylisoquinoline alkaloid isolated from the root of the plant. Tetrandrine non-selectively inhibits calcium channel activity and induces G1 blockade
||Phenylalanine is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.
||(±)-trans-ACPD is an equimolecular mixture of (1S,3R)- and (1R,3S)-ACPD. (±)-trans-ACPD is a selective agonist of the mGluR (metabotropic glutamate receptor); active at the group
||SEA0400 is a selective inhibitor of the Na+/Ca2+ exchanger.
||NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).
||ABT-639 is a potent and selective T-type calcium channel blocker.
||(S)-Amlodipine Besylate (103129-82-4(free base))
||Levamlodipine, also known as S-amlodipine, is a pharmacologically active enantiomer of amlodipine, an antihypertensive and anti-anginal medication. Levamlodipine belongs to the dih
||Fantofarone is a highly potent Calcium Channel antagonist.
||Addition of the Rhamnose-rich polysaccharide, RROP-1, to normal human dermal fibroblasts (NHDFs) and human endothelial cells produced a dose-dependent stimulation of the calcium-si
||Aranidipine (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.
||Bepridil is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels.
||MK-8998 as potent inhibitors of T-type calcium channels.
||Barnidipine is a dihydropyridine calcium channel blocker that has an IC50 value of 0.35 nM in potassium-induced tonic contraction of pig coronary artery
||Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
||Lomerizine dihydrochloride is an antagonist of L- and T-type voltage-gated calcium channels used to treat migraine.
||Manidipine, a calcium channel blocker, which is dihydropyridine type. It is utilized
||Ranolazine 2HCl，a calcium uptake inhibitor，is used to treat chronic angina via the sodium/calcium channa.
||Lercanidipine is a calcium channel blocker of the dihydropyridine class.
||Dronedarone is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
||Mirogabalin is a calcium channel blocker with analgesic effects.
||NP118809 is a potent N-type calcium channel blocker(IC50 : 0.11 μM).
||DHBP dibromide is calcium release and a muscle relaxant inhibitor.
||CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).
||Barnidipine is a calcium channel blocker.
||Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.
||1. Pulegone has cytotoxicity followed by regenerative cell proliferation is the MOA for Pulegone-induced urothelial tumors in female rats. 2. Pulegone induces a verapamil-sensitive
||(S)-(-)-Bay K 8644
||(S)-(-)-Bay-K-8644 is an agonist of L-type Ca2+ channel. It activates Ba2+ currents (IBa) (EC50: 32 nM).
||(R)-(+)-Bay K 8644
||(R)-(+)-Bay K 8644 is a calcium channel inhibitor. It inhibits Ba2+ currents (IBa) (IC50: 975 nM).
||Mibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s: 2.7 μM and 18.6 μM for T-type and L-type currents).
||Thapsigargin is a microsomal Ca2+-ATPase inhibitor and Endoplasmic Reticulum stress-inducing agent.