Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
TCS2185 | Yohimbine
育亨宾
|
146-48-5 |
|
|
Yohimbine 是一种有效的、相对非选择性的α2 - 肾上腺素能受体拮抗剂,IC50=0.6μM。 | ||||
T1769 | Pardoprunox
帕多芦诺
|
269718-84-5 |
|
|
Pardoprunox (SLV-308) 是多巴胺受体D2、D3部分激动剂和5-HT1A 激动剂,pEC50分别为 8、9.2 和 6.3。 | ||||
TN4882 | Quinine HCl
化合物 TN4882
|
130-89-2 | 98% |
|
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses. | ||||
T5450 | DL-071-IT
化合物DL-071-IT
|
55104-39-7 | 98% |
|
DL-071-IT (Afurolol Hydrochloride) 是一种有效的非选择性β-肾上腺素受体拮抗剂。 DL-071-IT 表现出内在的拟交感神经活性和弱的膜稳定活性。 | ||||
T13470 | (±)-Levomepromazine-d6
化合物 T13470
|
1189805-51-3 | 98% |
|
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor. | ||||
T78567 | Moprolol
化合物 Moprolol
|
5741-22-0 | 98% |
|
Moprolol ((±)-Moprolol)为β-肾上腺素能受体阻滞剂,主要应用于原发性高血压研究。 | ||||
T79641 | (±)-N-Methylcoclaurine
化合物 (±)-N-Methylcoclaurine
|
1472-62-4 | 98% |
|
(±)-N-Methylcoclaurine为选择性α2-肾上腺素受体拮抗剂。 | ||||
T80175 | Conopeptide rho-TIA
化合物 Conopeptide rho-TIA
|
381725-58-2 | 98% |
|
Conopeptide rho-TIA为从掠食性海螺Conus tulipa毒液中提炼的多肽,对人类α1B-Adrenergic Receptor呈现非竞争性抑制作用,同时对α1A-Adrenergic Receptor和α1D-Adrenergic Receptor表现出竞争性抑制。Conopeptide rho-TI... | ||||
T80477 | Muscarinic toxin 3
化合物 Muscarinic toxin 3
|
873336-87-9 | 98% |
|
Muscarinic toxin 3 (MT3) 是高效的非竞争性mAChR及adrenoceptors拮抗剂,对M1、M4、α1A、α1B、α1D、α2A、α2B、α2C受体展示出不同程度的选择性,其pIC50值分别为6.71、8.79、8.86、7.57、8.13、8.49、6.5、7.29。该化合物具有显著的肾上腺... | ||||
TN1797 | Isorhoifolin
异野漆树苷
|
552-57-8 | 98% |
|
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f... | ||||
T81798 | Mibenratide TFA
化合物 Mibenratide TFA
|
98% |
|
|
Mibenratide TFA,一种小环肽及肾上腺素能 β1 受体 (adrenergic β1 receptor) 拮抗剂,适用于心力衰竭研究。 | ||||
T15042 | D2343
化合物 T15042
|
72734-63-5 | 98% |
|
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor. | ||||
T6663 | Scopine hydrochloride
盐酸东莨菪醇
|
85700-55-6 | 98% |
|
Scopine hydrochloride (6,7-Epoxytropine hydrochloride) 是一种 Anisodine 的代谢物。 | ||||
T16769 | Ro 363
化合物 T16769
|
74513-77-2 | 98% |
|
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr... | ||||
TN2267 | Tetrahydroalstonine
四氢鸭脚木碱
|
6474-90-4 | 98% |
|
Tetrahydroalstonine 是从 Rhazya stricta 的果实中提取出来的吲哚类生物碱,是一种具有选择性的 α2-肾上腺素受体拮抗剂。Tetrahydroalstonine 在Rauwolfia tetraphylla 中表现出抗精神病活性。 | ||||
TN3368 | Akuammigine
化合物 TN3368
|
642-17-1 | 98% |
|
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p... | ||||
T11786 | KUL-7211 racemate
化合物 T11786
|
911196-40-2 | 98% |
|
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211. | ||||
T12815 | (S)-Terazosin
(S)-特拉唑嗪
|
109351-33-9 | 98% |
|
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with... | ||||
T13285 | Vatinoxan hydrochloride
化合物 T13285
|
130466-38-5 | 98% |
|
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors. | ||||
T11036 | Diacetolol D7
化合物 T11036
|
1346604-19-0 | 98% |
|
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent. |