T2382 | Vemurafenib |
Vemurafenib (PLX4032) is a novel and potent B-Raf (V600E) inhibitor (IC50: 31 nM). |
T2641 | KRCA0008 | KRCA-0008 is an effective and specific ALK/Ack1 inhibitor (IC50: 12/4 nM); displays drug-like properties without hERG liability. |
T5092 | AIM100 | AIM-100 is a Ack1 inhibitor (IC50: 24 nM). |