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"Perphenazine" 的搜索结果

相关产品

目录号	产品详情		靶点
T1090	Perphenazine	Perphenazin,Trilafon,Etaperazine,奋乃静	CaMK Dopamine Receptor 5-HT Receptor Adrenergic Receptor Histamine Receptor
T1090	Perphenazine 是吩噻嗪衍生物和多巴胺拮抗剂，具有止吐和抗精神病特性。它能够抑制5-HT2A 受体，α1A 肾上腺素能受体，多巴胺D2、D3、D2L 受体，以及组胺H1受体，对应的Ki 值分别为5.6、10、0.765、0.13、3.4 和 8 nM。
T69381	Dechloro perphenazine
T69381	Dechloro perphenazine is the dechlorinated analogue of Perphenazine (P291100), an D2 dopamine receptor antagonist; α-adrenergic receptor antagonist and σ-receptor agonist.
T63115	Perphenazine dihydrochloride
T63115	Perphenazine dihydrochloride 是一种口服具有活力的多巴胺受体 (dopamine receptor) 和组胺-1 受体 (histamine-1 receptor) 拮抗剂，作用于 D2 (Ki: 0.56 nM)、D3 (Ki: 0.43 nM)、5-HT2A (Ki: 0.6 nM)。Perphenazine dihydrochloride 也能够结合 Alpha-1A 肾上腺素受体。Perphenazine dihydrochloride 能够诱导细胞凋亡，并抑制癌细胞增殖。Perphenazine dihydrochloride 能够用于研究精神疾病、癌症、炎症。
T12411	Perphenazine D8 Dihydrochloride		Others
T12411	Perphenazine D8 Dihydrochloride is the deuterium labeled Perphenazine, which is an antipsychotic drug.		Others
T26834	BL-1020 Mesylate	Perphenazine GABA ester,CYP-1020,AN-168,BL 1020,BL1020
T26834	BL-1020 is a GABA A receptor agonist and dopamine receptor antagonist. BL-1020 is an ester of GABA and perphenazine, and pharmacologically it acts as a GABA agonist and D2 antagonist. BL-1020 has shown pro-cognitive effects in the trials.