T2325
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EGFR
HER
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Neratinib (HKI-272) 是一种口服的、不可逆的酪氨酸激酶抑制剂,对 HER2 和 EGFR 的 IC50值分别为 59 和 92 nM。 |
T67385
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EGFR
HER
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Neratinib maleate (HKI-272 maleate) 是一种不可逆且具有口服活性和高选择性的 HER2 和 EGFR 抑制剂,IC50 值分别为 59 nM 和 92 nM。Neratinib maleate具有抗肿瘤活性,可用于治疗消化系统疾病、呼吸系统疾病、泌尿生殖系统疾病和皮肤和肌肉骨骼疾病,可用于研究乳腺癌和前列腺癌。 |
T71387
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Neratinib maleate monohydrate is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity. |
T70829
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Neratinib pyridine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity. |
T70830
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Neratinib dimethylamine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity. |
T70828
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HBY-793 is an HIV-1 proteinase inhibitor. |
T70827
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MDL-102234 is an adenosine A1 receptor antagonist. |