Potassium Channel inhibitor kit 包含钾离子通道抑制剂,可以抑制平滑肌细胞、神经瘤细胞以及肝细胞膜上低电的钾通道,也可以扩张冠状动脉血管,增加冠状动脉的血流量,减少心肌的耗氧量、减慢心率,治疗室上性的房颤以及心动过速,还可以增加钙的流入,增加肌纤维收缩力,从而治疗肌无力等疾病。TargetMol 为您提供68种精选钾离子通道抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0038 | Doxapram hydrochloride hydrate | 7081-53-0 | 432.99 | 10mM | Potassium Channel |
T0127 | Glimepiride | 93479-97-1 | 490.62 | 10mM | Potassium Channel |
T0249 | N-Acetylprocainamide | 32795-44-1 | 277.36 | 10mM | Drug Metabolite; Potassium Channel; Sodium Channel |
T0266 | Quinidine hydrochloride monohydrate | 6151-40-2 | 378.89 | 10mM | Parasite; Potassium Channel; Sodium Channel |
T0451 | Minoxidil | 38304-91-5 | 209.25 | 10mM | COX; Potassium Channel |
T0690 | Quinine | 130-95-0 | 324.42 | 10mM | Parasite; Platelet aggregation; Potassium Channel |
T0723 | Cloperastine hydrochloride | 14984-68-0 | 366.33 | 10mM | 5-HT Receptor; Potassium Channel |
T0816 | Acetohexamide | 968-81-0 | 324.4 | 10mM | NADPH; Potassium Channel |
T0860 | Mefloquine hydrochloride | 51773-92-3 | 414.77 | 10mM | Autophagy; Parasite; Potassium Channel; Reactive Oxygen Species; SARS-CoV |
T0979 | Dequalinium chloride | 522-51-0 | 527.59 | 10mM | PKC; Potassium Channel |
T1073 | Dronedarone hydrochloride | 141625-93-6 | 593.22 | 10mM | Adrenergic Receptor; Autophagy; Calcium Channel; Potassium Channel; Sodium Channel |
T1384 | Chlorpromazine hydrochloride | 69-09-0 | 355.32 | 10mM | 5-HT Receptor; Autophagy; Dopamine Receptor; Potassium Channel; Sodium Channel |
T1496 | Amiodarone hydrochloride | 19774-82-4 | 681.78 | 10mM | Adrenergic Receptor; Autophagy; Potassium Channel |
T1527 | Gliclazide | 21187-98-4 | 323.42 | 10mM | Potassium Channel |
T1530 | Mitiglinide calcium hydrate | 207844-01-7 | 704.91 | 10mM | Potassium Channel |
T1634 | Glibenclamide | 10238-21-8 | 494.01 | 10mM | Autophagy; CFTR; Mitochondrial Metabolism; P-gp; Potassium Channel |
T1674 | Nateglinide | 105816-04-4 | 317.42 | 10mM | Potassium Channel; PPAR; Proteasome |
T1752 | NS6180 | 353262-04-1 | 323.33 | 10mM | Potassium Channel |
T2712 | Nifekalant hydrochloride | 130656-51-8 | 441.91 | 10mM | Potassium Channel |
T2996 | Tetrandrine | 518-34-3 | 622.77 | 10mM | Calcium Channel; Potassium Channel |
T3528 | Senicapoc | 289656-45-7 | 323.11 | 10mM | Potassium Channel |
T3557 | GAL-021 | 1380341-99-0 | 254.33 | 10mM | Potassium Channel |
T3574 | Sematilide hydrochloride | 101526-62-9 | 349.87 | 10mM | Potassium Channel |
T4316 | ML365 | 947914-18-3 | 360.41 | 10mM | Potassium Channel |
T6186 | TRAM-34 | 289905-88-0 | 344.84 | 10mM | IκB/IKK; Potassium Channel |
T6476 | Dofetilide | 115256-11-6 | 441.56 | 10mM | Potassium Channel |
T6592 | ML133 hydrochloride | 1222781-70-5 | 313.82 | 10mM | Potassium Channel |
T3S0081 | Oxypeucedanin | 737-52-0 | 286.28 | 10mM | Potassium Channel |
T3S1873 | Talatisamine | 20501-56-8 | 421.57 | 10mM | Potassium Channel |
T5585 | AM-92016 hydrochloride | 133229-11-5 | 483.84 | 10mM | Potassium Channel |
T6978 | Almitrine mesylate | 29608-49-9 | 669.76 | 10mM | Potassium Channel |
T7195 | GSK369796 Dihydrochloride | 1010411-21-8 | 428.78 | 10mM | Parasite; Potassium Channel |
T7198 | E-4031 | 113559-13-0 | 474.44 | 10mM | EGFR; Potassium Channel |
T7505 | Azimilide Dihydrochloride | 149888-94-8 | 530.88 | 10mM | Potassium Channel |
T7538 | Tetraethylammonium chloride | 56-34-8 | 165.7 | 10mM | Potassium Channel |
T7653 | JNJ 303 | 878489-28-2 | 440.98 | 10mM | Potassium Channel |
T7774 | A2793 | 88349-90-0 | 265.7 | 10mM | Potassium Channel |
T7775 | A2764 dihydrochloride | 861038-72-4 | 351.7 | 10mM | Potassium Channel |
T8372 | VU0134992 | 755002-90-5 | 411.38 | 10mM | Potassium Channel |
T15555 | IK1 inhibitor PA-6 | 500715-03-7 | 492.62 | 10mM | Potassium Channel |
T13316 | VU0134992 hydrochloride | 1052515-91-9 | 447.84 | 10mM | Potassium Channel |
T16110 | ML418 | 1928763-08-9 | 377.87 | 10mM | Potassium Channel |
T15758 | Linopirdine | 105431-72-9 | 391.46 | 10mM | Potassium Channel; TRP/TRPV Channel |
T13320 | VU591 hydrochloride | 1315380-70-1 | 404.76 | 10mM | Potassium Channel |
T17262 | XE 991 dihydrochloride | 122955-13-9 | 449.37 | 10mM | Potassium Channel |
T8700 | TKIM | 326921-25-9 | 371.05 | 10mM | Potassium Channel |
T10979 | DCPIB | 82749-70-0 | 427.36 | 10mM | Chloride channel; Potassium Channel |
T8977 | Kv2-IN-A1 | 689297-68-5 | 396.89 | 10mM | Potassium Channel |
T9070 | ASP2905 | 792184-90-8 | 388.4 | 10mM | Potassium Channel |
T22745 | DPO-1 | 43077-30-1 | 340.44 | 10mM | Potassium Channel |
T16347 | NS3623 | 343630-41-1 | 427.18 | 10mM | Potassium Channel |
T13164 | Tipepidine hydrochloride | 1449686-84-3 | 311.89 | 10mM | Dopamine Receptor; Potassium Channel |
TQ0179 | PAP-1 | 870653-45-5 | 350.36 | 10mM | Potassium Channel |
T12256 | NS8593 hydrochloride | 875755-24-1 | 299.8 | 10mM | Potassium Channel |
T20968 | CyPPA | 73029-73-9 | 285.39 | 10mM | Dopamine Receptor; Potassium Channel |
T14982 | Clofilium tosylate | 92953-10-1 | 510.17 | 10mM | Potassium Channel |
T12786 | RY785 | 1393748-80-5 | 392.47 | 10mM | Potassium Channel |
T15385 | Glibornuride | 26944-48-9 | 366.48 | 10mM | Potassium Channel |
T15546 | ICA | 3374-88-7 | 254.31 | 10mM | Parasite; Potassium Channel |
T10435 | Linaprazan | 248919-64-4 | 366.46 | 10mM | Potassium Channel |
T29457L | 5-Hydroxydecanoate sodium | T29457L | 210.25 | 10mM | Potassium Channel |
T17243 | VU0463271 | 1391737-01-1 | 382.5 | 10mM | Potassium Channel |
T26689 | AVE-0118 | 498577-53-0 | 479.57 | 10mM | Potassium Channel |
T60061 | RU-TRAAK-2 | 1210538-56-9 | 335.42 | 10mM | Potassium Channel |
TQ0139 | VU 0240551 | 893990-34-6 | 342.44 | 10mM | Potassium Channel;HER;Calcium Channel |
T12504 | (+)-KCC2 blocker 1 | 1228439-71-1 | 415.5 | 10mM | Potassium Channel |
T23471 | TRAM 39 | 197525-99-8 | 303.79 | 10mM | Potassium Channel |
T30544 | BMS-919373 | 1272353-82-8 | 468.53 | 10mM | Potassium Channel |