GABA Receptor inhibitor kit 包含γ-氨基丁酸GABA 受体抑制剂,GABA 受体能识别并结合GABA,导致细胞膜离子通透性变化,GABA 是脊椎动物中枢神经系统中的主要抑制性神经递质。GABA 受体抑制剂可以升高血压,具有中枢神经系统兴奋作用,促进学习与记忆功能。TargetMol 为您提供39种精选GABA 受体抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0128 | Vigabatrin | 60643-86-9 | 129.16 | 10mM | ABC; GABA Receptor |
T0349 | Riluzole | 1744-22-5 | 234.2 | 10mM | GABA Receptor; NMDAR; Sodium Channel |
T1240 | Flumazenil | 78755-81-4 | 303.29 | 10mM | GABA Receptor |
T1396 | Bemegride | 64-65-3 | 155.19 | 10mM | GABA Receptor |
T2196 | Fipronil | 120068-37-3 | 437.15 | 10mM | GABA Receptor; GluCls; P450 |
T2407 | Tiagabine | 115103-54-3 | 375.55 | 10mM | GABA Receptor |
T2749 | Ginkgolide A | 15291-75-5 | 408.4 | 10mM | Endogenous Metabolite; GABA Receptor |
T2850 | Bicuculline | 485-49-4 | 367.36 | 10mM | GABA Receptor |
T2998 | Dihydromyricetin | 27200-12-0 | 320.25 | 10mM | Autophagy; DNA/RNA Synthesis; GABA Receptor; Influenza Virus; mTOR |
T3644 | U93631 | 152273-12-6 | 299.37 | 10mM | GABA Receptor |
T3698 | alpha-Asarone | 2883-98-9 | 208.3 | 10mM | GABA Receptor; HMG-CoA Reductase; P450 |
T4363 | CGP52432 | 139667-74-6 | 384.23 | 10mM | GABA Receptor |
T4440 | Saclofen | 125464-42-8 | 249.71 | 10mM | GABA Receptor |
T7000 | Tiagabine hydrochloride | 145821-59-6 | 412.01 | 10mM | GABA Receptor |
T2S1464 | Thiocolchicoside | 602-41-5 | 563.61 | 10mM | GABA Receptor |
T2S1814 | p-Hydroxybenzaldehyde | 123-08-0 | 122.12 | 10mM | Endogenous Metabolite; GABA Receptor; transaminase |
T5S1882 | Songorine | 509-24-0 | 357.49 | 10mM | GABA Receptor |
T5330 | Fluralaner | 864731-61-3 | 556.29 | 10mM | GABA Receptor; Parasite |
T5880 | Aminooxyacetic acid hemihydrochloride | 2921-14-4 | 109.3 | 10mM | GABA Receptor |
T7622 | Gabazine | 104104-50-9 | 368.23 | 10mM | GABA Receptor |
T7557 | Guvacine hydrochloride | 6027-91-4 | 163.6 | 10mM | GABA Receptor |
T7793 | 6-(4-Methoxyphenyl)-3-pyridazinamine | 4776-87-8 | 201.22 | 10mM | GABA Receptor |
T8193 | α-Thujone | 546-80-5 | 152.23 | 10mM | AChR; Apoptosis; Autophagy; GABA Receptor; Parasite; Reactive Oxygen Species |
T8268 | 6,2'-Dihydroxyflavone | 92439-20-8 | 254.24 | 10mM | GABA Receptor |
T3S2100 | (-)-Securinine | 5610-40-2 | 217.26 | 10mM | GABA Receptor |
T8162 | Cannabidivarin | 24274-48-4 | 286.4 | 10mM | GABA Receptor |
T8568 | Suritozole | 110623-33-1 | 223.27 | 10mM | GABA Receptor |
T11307 | Fluxametamide | 928783-29-3 | 474.26 | 10mM | GABA Receptor |
T8971 | Imidazenil | 151271-08-8 | 399.2 | 10mM | GABA Receptor |
T13536 | Afoxolaner | 1093861-60-9 | 625.87 | 10mM | Chloride channel; GABA Receptor; Parasite |
T15775 | Lotilaner | 1369852-71-0 | 596.76 | 10mM | GABA Receptor; Parasite |
TQ0040 | ONO-8590580 | 1802661-73-9 | 376.43 | 10mM | GABA Receptor |
T10618 | Broflanilide | 1207727-04-5 | 663.28 | 10mM | GABA Receptor |
T12930 | SKF89976A hydrochloride | 85375-15-1 | 371.9 | 10mM | GABA Receptor |
T23339 | SCS | 3232-36-8 | 256.26 | 10mM | GABA Receptor |
T37190 | L-Allylglycine | 16338-48-0 | 115.13 | 10mM | Dehydrogenase; GABA Receptor |
T24540 | NO-711ME | 127586-66-7 | 364.44 | 10mM | GABA Receptor |
T21793 | CGP 35348 | 123690-79-9 | 225.22 | 10mM | GABA Receptor |
T11137 | (E)-GABAB receptor antagonist 1 | 1611483-29-4 | 304.38 | 10mM | GABA Receptor |