Estrogen Receptor inhibitor kit 包含雌激素受体抑制剂,雌激素受体主要通过调节特异性靶基因的转录或第二信使系统发挥间接的转录调控功能而发挥作用,参与了对骨组织、生殖系统和神经系统诸如学习、记忆、认知等多种功能的调节。TargetMol 为您提供45种精选雌激素受体抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0168 | Estradiol (cypionate) | 313-06-4 | 396.58 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T1102 | Mifepristone | 84371-65-3 | 429.6 | 10mM | Autophagy; Estrogen/progestogen Receptor; Glucocorticoid Receptor; NO Synthase; progesterone receptor |
T1193 | Clomiphene citrate | 50-41-9 | 598.1 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T1549 | Raloxifene hydrochloride | 82640-04-8 | 510.04 | 10mM | Autophagy; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; MAO |
T1571 | Estriol | 50-27-1 | 288.39 | 10mM | Endogenous Metabolite; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; MRP |
T2177 | Kaempferol | 520-18-3 | 286.23 | 10mM | Apoptosis; Autophagy; Endogenous Metabolite; Estrogen Receptor/ERR; Estrogen/progestogen Receptor; HIV Protease; Mitophagy; Parasite |
T2527 | Ulipristal acetate | 126784-99-4 | 475.62 | 10mM | Autophagy; Estrogen/progestogen Receptor; progesterone receptor |
T2544 | Bazedoxifene acetate | 198481-33-3 | 530.67 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T2569 | Chlorotrianisene | 569-57-3 | 380.86 | 10mM | COX; Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T2837 | Chrysin | 480-40-0 | 254.24 | 10mM | Antioxidant; Estrogen Receptor/ERR |
T2882 | Genistin | 529-59-9 | 432.37 | 10mM | Apoptosis; Estrogen Receptor/ERR |
T3717 | Hinokitiol | 499-44-5 | 164.2 | 10mM | DNA Methyltransferase; Estrogen/progestogen Receptor; Virus Protease; Nrf2 |
T3840 | Dihydroresveratrol | 58436-28-5 | 230.3 | 10mM | Estrogen Receptor/ERR |
T3855 | Tracheloside | 33464-71-0 | 550.56 | 10mM | Estrogen Receptor/ERR; Phosphorylase |
T3975 | AZD9496 | 1639042-08-2 | 442.47 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T4388 | PHTPP | 805239-56-9 | 423.32 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T4420 | 4-Hydroxytamoxifen | 68047-06-3 | 387.51 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T6491 | (-)-(S)-Equol | 531-95-3 | 242.27 | 10mM | Endogenous Metabolite; Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T6713 | Ulipristal | 159811-51-5 | 433.58 | 10mM | Estrogen/progestogen Receptor; progesterone receptor |
T6743 | (E/Z)-4-Hydroxytamoxifen | 68392-35-8 | 387.51 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T5S0543 | Isocurcumenol | 24063-71-6 | 234.33 | 10mM | Apoptosis; Estrogen Receptor/ERR; Reductase |
T5118 | Brilanestrant | 1365888-06-7 | 446.9 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T5633 | H3B-5942 | 2052128-15-9 | 494.63 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T7389 | G15 | 1161002-05-6 | 370.24 | 10mM | Estrogen Receptor/ERR |
T7313 | Enclomiphene citrate | 7599-79-3 | 598.08 | 10mM | Estrogen Receptor/ERR |
T7839 | Lasofoxifene Tartrate | 190791-29-8 | 563.64 | 10mM | Estrogen Receptor/ERR |
T12832 | Amcenestrant | 2114339-57-8 | 554.48 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
TQ0295 | Coumestrol | 479-13-0 | 268.2 | 10mM | Estrogen Receptor/ERR |
T8984 | FLTX1 | 1481401-71-1 | 520.6 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T15249 | Estrogen receptor modulator 1 | 63676-22-2 | 242.29 | 10mM | Estrogen Receptor/ERR |
T11399 | Giredestrant | 1953133-47-5 | 522.55 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T5348 | SNG-1153 | 1446712-19-1 | 406.35 | 10mM | Estrogen/progestogen Receptor |
T15191 | PROTAC ERRα ligand 1 | 1264754-13-3 | 420.36 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T13674 | Elacestrant | 722533-56-4 | 458.63 | 10mM | Estrogen Receptor/ERR; Estrogen/progestogen Receptor |
T21387L | Nafoxidine | 1845-11-0 | 425.56 | 10mM | Estrogen Receptor/ERR |
T13675 | Elacestrant dihydrochloride | 1349723-93-8 | 531.56 | 10mM | Estrogen/progestogen Receptor |
T20625 | Prochloraz | 67747-09-5 | 376.67 | 10mM | AhR; Androgen Receptor; Antifungal; Estrogen Receptor/ERR |
T39710 | ARV-471 | 2229711-68-4 | 723.9 | 10mM | Estrogen Receptor/ERR |
T21897L | MPP hydrochloride | T21897L | 506.04 | 10mM | Estrogen Receptor/ERR |
T10239 | Acolbifene | 182167-02-8 | 457.56 | 10mM | Estrogen Receptor/ERR |
T12482 | Pipendoxifene hydrochloride | 245124-69-0 | 493.04 | 10mM | Estrogen Receptor/ERR |
T17252 | WAY-204688 | 796854-35-8 | 556.62 | 10mM | Estrogen/progestogen Receptor;NF-κB |
T15788 | LSZ-102 | 2135600-76-7 | 470.46 | 10mM | Estrogen Receptor/ERR |
T12654 | (Rac)-Acolbifene | 151533-34-5 | 457.56 | 10mM | Estrogen Receptor/ERR |
T11230 | ERRα antagonist-1 | 1072145-33-5 | 377.53 | 10mM | Estrogen/progestogen Receptor |