Endothelin Receptor antagonist kit 包含内皮素受体拮抗剂,内皮素具有强烈缩血管作用,诱导血管生成、促分化、促细胞有丝分裂和类细胞生长因子。内皮素还有强大的正性肌力作用,反射性引起心率抑制,造成心肌供血不足.而且还可诱发心肌细胞糖超载,心律失常以及心肌能量代谢障碍。内皮素受体拮抗剂常用于心绞痛、AMI、心肌1/R 损伤、缺血性心脏病的防治研究。TargetMol 为您提供18种精选内皮素受体拮抗剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0750 | Sulfisoxazole | 127-69-5 | 267.31 | 10mM | Antibacterial; Antibiotic; Autophagy; Endothelin Receptor |
T1655 | Ambrisentan | 177036-94-1 | 378.42 | 10mM | Endothelin Receptor |
T2561 | Macitentan | 441798-33-0 | 588.27 | 10mM | Apoptosis; Endothelin Receptor |
T3194 | Ro 46-2005 | 150725-87-4 | 473.54 | 10mM | Endothelin Receptor |
T3474 | RO 46-8443 | 175556-12-4 | 609.69 | 10mM | Endothelin Receptor |
T6264 | Bosentan | 147536-97-8 | 551.61 | 10mM | Endothelin Receptor |
T6265 | Bosentan (hydrate) | 157212-55-0 | 569.63 | 10mM | Endothelin Receptor |
T6672 | Sitaxsentan sodium | 210421-74-2 | 476.89 | 10mM | Endothelin Receptor |
T6792 | BQ-123 | 136553-81-6 | 610.7 | 10mM | Endothelin Receptor |
T5458 | Darusentan | 171714-84-4 | 410.43 | 10mM | Endothelin Receptor |
T7817 | Aprocitentan | 1103522-45-7 | 546.19 | 10mM | Endothelin Receptor |
T5355 | Sparsentan | 254740-64-2 | 592.8 | 10mM | Endothelin Receptor; RAAS |
T21790 | BMS 182874 hydrochloride | 1215703-04-0 | 381.88 | 10mM | Endothelin Receptor |
TQ0259 | Atrasentan | 173937-91-2 | 510.62 | 10mM | Endothelin Receptor |
TQ0282 | Avosentan | 290815-26-8 | 479.51 | 10mM | Endothelin Receptor |
TQ0270 | Atrasentan hydrochloride | 195733-43-8 | 547.08 | 10mM | Endothelin Receptor |
TP1219 | Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate | 1366000-58-9 | 3140.5 | 10mM | Endothelin Receptor |
T15596 | IRL 2500 | 169545-27-1 | 573.68 | 10mM | Endothelin Receptor |