DPP4 inhibitor kit 包含二肽基肽酶4 DPP4抑制剂,常用于2型糖尿病的研究,能够抑制胰高血糖素样肽-1和葡萄糖依赖性促胰岛素分泌多肽(GIP)的灭活,提高其内源性水平,促进胰岛β细胞释放胰岛素,同时抑制胰岛α细胞分泌胰高血糖素,从而提高胰岛素水平,降低血糖,且不易诱发低血糖和增加体重。TargetMol 为您提供22种精选DPP4抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0178 | Saxagliptin hydrate | 945667-22-1 | 333.43 | 10mM | DPP-4; Proteasome |
T0191 | Linagliptin | 668270-12-0 | 472.54 | 10mM | Autophagy; DPP-4; Ferroptosis; Proteasome |
T0242 | Sitagliptin | 486460-32-6 | 407.32 | 10mM | Autophagy; DPP-4; Proteasome |
T1502 | Vildagliptin | 274901-16-5 | 303.4 | 10mM | Apoptosis; DPP-4; Ferroptosis; Proteasome |
T1581 | Picolamine | 3731-52-0 | 108.14 | 10mM | DPP-4 |
T2296 | Trelagliptin succinate | 1029877-94-8 | 475.47 | 10mM | DPP-4; Proteasome |
T2316 | Omarigliptin | 1226781-44-7 | 398.43 | 10mM | DPP-4; Proteasome |
T2401 | Alogliptin Benzoate | 850649-62-6 | 461.51 | 10mM | DPP-4; Ferroptosis; Proteasome |
T4042 | Talabostat mesylate | 150080-09-4 | 310.18 | 10mM | DPP-4; Proteasome |
T6192 | Alogliptin | 850649-61-5 | 339.39 | 10mM | DPP-4; Ferroptosis; Proteasome |
T6203 | Saxagliptin | 361442-04-8 | 315.41 | 10mM | DPP-4; Proteasome |
T6237 | Trelagliptin | 865759-25-7 | 357.38 | 10mM | DPP-4; Proteasome |
T6999 | Teneligliptin hydrobromide | 906093-29-6 | 628.86 | 10mM | DPP-4; Proteasome |
T7369 | Gemigliptin | 911637-19-9 | 489.36 | 10mM | DPP-4; Proteasome |
T7133 | Anagliptin | 739366-20-2 | 383.45 | 10mM | DPP-4; Proteasome |
T16838 | Saikogenin A | 5092-09-1 | 472.7 | 10mM | DPP-4; Proteasome |
T12710 | Retagliptin Phosphate | 1256756-88-3 | 562.36 | 10mM | DPP-4; Proteasome |
T15079 | DBPR108 | 1186426-66-3 | 324.39 | 10mM | DPP-4; Proteasome |
T25340 | Diprotin A | 90614-48-5 | 341.45 | 10mM | DPP-4 |
T11526 | DPP-IV-IN-2 | 136259-18-2 | 378.42 | 10mM | DPP-4 |
T23358 | Sitagliptin phosphate | 654671-78-0 | 505.31 | 10mM | Autophagy; DPP-4 |
TN1418 | Azaleatin | 529-51-1 | 316.26 | 10mM | DPP-4 |