Androgen Receptor antagonist kit 包含雄激素受体拮抗剂,雄激素受体属于核受体超家族中的类固醇受体,与雄激素结合后,激活第二信使信号通路,调控靶基因的转录和翻译,从而影响生殖、骨骼肌、心血管、神经、免疫、造血系统的发育和稳态维持等方面。TargetMol 为您提供43种精选雄激素受体拮抗剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0272 | Nilutamide | 63612-50-0 | 317.22 | 10mM | Androgen Receptor |
T0380 | Bicalutamide | 90357-06-5 | 430.37 | 10mM | Androgen Receptor; Autophagy |
T0489 | Flutamide | 13311-84-7 | 276.21 | 10mM | Androgen Receptor |
T1167 | Cyproterone acetate | 427-51-0 | 416.94 | 10mM | Androgen Receptor |
T1541 | Drospirenone | 67392-87-4 | 366.49 | 10mM | Androgen Receptor; COX; Estrogen/progestogen Receptor; Glucocorticoid Receptor; progesterone receptor |
T1596 | Chlormadinone acetate | 302-22-7 | 404.93 | 10mM | Androgen Receptor; progesterone receptor |
T2236 | RU 58841 | 154992-24-2 | 369.34 | 10mM | Androgen Receptor |
T2339 | Apalutamide | 956104-40-8 | 477.43 | 10mM | Androgen Receptor; GABA Receptor |
T2895 | Lupeol | 545-47-1 | 426.73 | 10mM | Akt; Androgen Receptor; Apoptosis |
T2991 | 3,3'-Diindolylmethane | 1968-05-4 | 246.31 | 10mM | Androgen Receptor; Autophagy |
T3357 | Clascoterone | 19608-29-8 | 402.52 | 10mM | Androgen Receptor |
T3393 | Triptophenolide | 74285-86-2 | 312.4 | 10mM | Androgen Receptor |
T6002 | Enzalutamide | 915087-33-1 | 464.44 | 10mM | Androgen Receptor; Autophagy |
T6400 | AZD3514 | 1240299-33-5 | 519.56 | 10mM | Androgen Receptor |
T6509 | Galeterone | 851983-85-2 | 388.55 | 10mM | Androgen Receptor; P450 |
T6829 | EPI-001 | 227947-06-0 | 394.89 | 10mM | Androgen Receptor; Apoptosis; PPAR |
T6889 | MI-136 | 1628316-74-4 | 470.51 | 10mM | Androgen Receptor; Apoptosis; Epigenetic Reader Domain |
T6915 | Darolutamide | 1297538-32-9 | 398.85 | 10mM | Androgen Receptor |
T7440 | p,p'-DDE | 72-55-9 | 318 | 10mM | Androgen Receptor; Drug Metabolite |
T7690 | 2-hydroxy Flutamide | 52806-53-8 | 292.21 | 10mM | Androgen Receptor |
T8592 | CTK8A3536 | 926228-58-2 | 276.35 | 10mM | Androgen Receptor |
T13273 | UT-34 | 2168525-92-4 | 356.27 | 10mM | Androgen Receptor |
TQ0209 | Ailanthone | 981-15-7 | 376.4 | 10mM | Androgen Receptor |
TQ0214 | Dimethylcurcumin | 52328-98-0 | 396.43 | 10mM | Androgen Receptor |
T19450 | N-desmethyl Enzalutamide | 1242137-16-1 | 450.41 | 10mM | Androgen Receptor |
TCS1372 | Atraric acid | 4707-47-5 | 196.2 | 10mM | Androgen Receptor; phosphatase |
T8933 | JNJ-63576253 free base | 2110426-27-0 | 502.51 | 10mM | Androgen Receptor |
T22263 | Bavdegalutamide | 2222112-77-6 | 812.29 | 10mM | Androgen Receptor |
T12323 | ORM-15341 | 1297537-33-7 | 396.83 | 10mM | Androgen Receptor |
T14008 | 2,2,5,7,8-Pentamethyl-6-Chromanol | 950-99-2 | 220.31 | 10mM | Androgen Receptor |
T13272 | UT-155 | 2031161-35-8 | 405.35 | 10mM | Androgen Receptor |
T15445 | Proxalutamide | 1398046-21-3 | 517.5 | 10mM | Androgen Receptor; SARS-CoV |
T9246 | JNJ-63576253 | 2110428-64-1 | 538.97 | 10mM | Androgen Receptor |
T10359 | AR antagonist 1 | 1818885-54-9 | 278.78 | 10mM | Androgen Receptor; Ligand for E3 Ligase; Ligands for Target Protein for PROTAC |
T12146 | N-Desmethyl-Apalutamide | 1332391-11-3 | 463.41 | 10mM | Androgen Receptor; P450 |
T9179 | CLP-3094 | 312749-73-8 | 304.8 | 10mM | Androgen Receptor |
T14116 | ACP-105 | 899821-23-9 | 290.79 | 10mM | Androgen Receptor |
T12928 | SK33 | 1928724-23-5 | 500.31 | 10mM | Androgen Receptor |
T29111 | VPC-13566 | 218464-59-6 | 258.32 | 10mM | Androgen Receptor |
T20625 | Prochloraz | 67747-09-5 | 376.67 | 10mM | AhR; Androgen Receptor; Antifungal; Estrogen Receptor/ERR |
T24943 | VPC-14228 | 19983-28-9 | 246.33 | 10mM | Androgen Receptor |
T39695 | ARD-2128 | 2222111-87-5 | 820.38 | 10mM | Androgen Receptor |
T21740 | RD162 | 915087-27-3 | 476.45 | 10mM | Androgen Receptor |