T4240
|
3',4',7-Trimethoxyflavan
|
3',4',7-Trimethoxyflavan 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T4240,CAS号为 116384-26-0。
|
TN2868
|
3',4',7,8-Tetrahydroxyflavone
|
3',4',7,8-Tetrahydroxyflavone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2868,CAS号为 3440-24-2。
|
TN4987
|
Semialactone
|
Semialactone shows inhibitory activities on human acyl-CoA:cholesterol acyltransferase(hACAT)1 with IC50 values of 79.1 uM and on human hACAT2 with IC50 values of 76.9 uM, it may be effective in the prevention and treatment of hypercholesterolemia or athe
|
TN4585
|
Moronic acid
|
Moronic acid shows oral therapeutic efficacy in HSV-infected mice and possessed novel anti-HSV activity. It also shows significant anti-HIV activity (EC(50) 186) and was modified to develop more potent anti-AIDS agents. Moronic acid is a new structural lead for anti-EBV drug development, can substantially reduce the numbers of EBV particles produced by the cells after lytic induction. Morolic and moronic acids have shown sustained antidiabetic and antihyperglycemic action possibly mediated by an insulin sensitization with consequent changes of glucose, cholesterol and triglycerides, in part mediated by inhibition of 11β-HSD 1 as indicated by in vitro.
|
TN4584
|
Morolic acid
|
Morolic acid and moronic acid have shown sustained antidiabetic and antihyperglycemic action possibly mediated by an insulin sensitization with consequent changes of glucose, cholesterol and triglycerides, in part mediated by inhibition of 11β-HSD 1. Moro
|
TN4911
|
Rhuscholide A
|
Rhuscholide A possesses significant anti-HIV-1 activity with an EC50 value of 1.62 microM and a therapeutic index (TI) of 42.40.
|
T8290
|
3,5-DIHYDROXY-4-METHOXYBENZOIC ACID
|
3,5-DIHYDROXY-4-METHOXYBENZOIC ACID 是一种天然存在的酚类化合物,存在于各种植物和动物中,具有抗氧化、抗炎、抗菌和抗肿瘤的活性。
|
T0801
|
Tannic acid
|
Tannic acid (Gallotannic acid) 是新型hERG 通道阻塞剂,IC50为 3.4 μM。
|
T5120
|
Rhamnose
|
alpha-L-Rhamnose (6-Deoxy-L-mannose) 是存在植物和细菌中的一种单糖。Rhamnose- 免疫原连接物能被用于免疫疗法。Rhamnose 能通过胞外途径穿过上皮细胞,能够作为肠吸收的标志。
|
TN1237
|
3-O-Methylgallic acid
|
3-O-Methylgallic acid (3,4-Dihydroxy-5-methoxybenzoic acid) 是一种花青素代谢产物,具有强大的抗氧化能力。它还诱导细胞凋亡并具有抗癌作用,可抑制 Caco-2 细胞增殖,IC50值为 24.1 μM。
|
T3040
|
Gallein
|
Gallein (Mordant violet 25) 是 G 蛋白 βγ 亚基信号抑制剂,能够干扰 Gβγ 亚基与 PI3Kγ 的相互作用。它可用作红色染料,酸碱指示剂和磷酸盐的检测试剂,具有抗肿瘤作用。
|
TN2244
|
Sulfuretin
|
Sulfuretin 是竞争性单酚酶和二酚酶活性抑制剂,IC50=13.64 μM。它通过抑制NF-κB 通路来抑制炎症反应。 它可用于过敏性气道炎症的研究。它减少氧化应激、血小板聚集和诱变。
|