单克隆抗体是由单个B 淋巴细胞克隆所分泌的抗体,由于B 淋巴细胞只能产生一种专有的、针对一种抗原决定簇的抗体,所以具有理化性质高度专一、生物活性单一、与抗原结合特异性强等特点。因此,它也被形象地被称为“生物导弹”, 现有的抗体药物大多属于此类抗体。近年来,单克隆抗体药物迅速发展,并逐渐成为生物医药领域发展的主要方向。
TargetMol可为您提供 xnum 多种抗体抑制剂,满足您的实验需求。TargetMol始终致力于服务“科研人员”,将热门的研究报道和产品推送给各位科研人员。
Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T9920 | Evolocumab
依洛尤单抗
|
1256937-27-5 | 98% |
Evolocumab
|
Evolocumab 是人源化单克隆抗体PCSK9的抑制剂。它与循环的 PCSK9 蛋白结合,使得PCSK9与 LDLR 结合受到抑制。它可用研究于高胆固醇血症以及动脉粥样硬化性心血管疾病的研究。 | ||||
T78269 | RMP1-14
抗体RMP1-14
|
98% |
RMP1-14
|
|
RMP1-14 是一种 IgG1 样免疫球蛋白抗小鼠 PD-1 抗体,可阻断 PD-1/PD-L1 信号传导。 | ||||
T36653 | Anti-SARS-80R mAb
Anti-SARS-80R mAb
|
98% |
Anti-SARS-80R mAb
|
|
Anti-SARS-80R mAb (SARS-80R) is a human IgG1 monoclonal antibody that is derived from CHO cells. Its main function is to selectively bind to the Spike (S1) prote... | ||||
T36654 | Anti-SARS-CoV-2 Spike mAb (CR3022)
Anti-SARS-CoV-2 Spike mAb (CR3022)
|
98% |
Anti-SARS-CoV-2 Spike mAb (CR3022)
|
|
Anti-SARS-CoV-2 Spike mAb (CR3022) is a human monoclonal IgG1 antibody derived from CHO cells. It specifically targets the S1 domain of the Spike protein in both... | ||||
T9923 | Nimotuzumab
尼妥珠单抗
|
828933-51-3 | 98% |
|
Nimotuzumab 是一种针对表皮生长因子受体 EGFR 的人源化治疗性单克隆抗体。 | ||||
T36651 | Anti-MERS-2E6 mAb
Anti-MERS-2E6 mAb
|
98% |
Anti-MERS-2E6 mAb
|
|
Anti-MERS-2E6 mAb (MERS-2E6), a human IgG1 neutralizing antibody, is expressed in CHO cells. It effectively competes with the virus Spike protein for binding to ... | ||||
T36655 | Anti-Spike-RBD mAb
Anti-Spike-RBD mAb
|
98% |
Anti-Spike-RBD mAb
|
|
Anti-Spike-RBD mAb is a CHO cell derived human monoclonal IgG1 antibody. Blocking the interaction of spike protein and ACE2 is a potential therapeutic approach f... | ||||
T9922 | Matuzumab
马妥珠单抗
|
339186-68-4 | 98% |
Matuzumab
|
Matuzumab 是一种用于癌症治疗的人源化单克隆抗体。它对 EGFR 具有高亲和力,通常与恶性肿瘤中血管的生长有关,从而促进肿瘤的生长和存活。 | ||||
T35389 | Sarilumab (anti-IL-6Rα)
Sarilumab (anti-IL-6Rα)
|
98% |
Sarilumab (anti-IL-6Rα)
|
|
Sarilumab (anti-IL-6Rα)是人源anti-IL-6Rα单克隆抗体,与膜结合的和可溶性的IL-6Rα以高亲和力结合。MW: 144.13 KD。 | ||||
T36656 | Anti-Spike-RBD Single Domain mAb
Anti-Spike-RBD Single Domain mAb
|
98% |
Anti-Spike-RBD Single Domain mAb
|
|
The Anti-Spike-RBD Single Domain mAb is a monoclonal antibody derived from CHO cells in Alpaca. It is composed of VHH-huFc and exhibits a strong affinity for the... | ||||
T12706 | Reslizumab
化合物 T12706
|
241473-69-8 | 98% |
|
Reslizumab is humanized monoclonal antibodies that target interleukin-5 (IL-5) for the treatment of eosinophilic asthma. | ||||
T9931 | Meplazumab
化合物meplazumab
|
2413715-21-4 | 98% |
meplazumab
|
meplazumab 是一种人源化抗 CD147 抗体,作为 COVID-19 肺炎患者的附加疗法。 | ||||
T36652 | Anti-MERS-3A1 mAb
Anti-MERS-3A1 mAb
|
98% |
Anti-MERS-3A1 mAb
|
|
Anti-MERS-3A1 mAb (MERS-3A1) is a high-affinity human monoclonal IgG1 antibody derived from CHO cells. It effectively inhibits the interaction between the MERS-C... | ||||
T35396 | Spartalizumab (anti-PD-1)
Spartalizumab (anti-PD-1)
|
98% |
Spartalizumab (anti-PD-1)
|
|
Spartalizumab (anti-PD-1)是一种针对PD-1的人源IgG4抗体,抑制PD-L1和PD-L2与PD-1的结合。PDR001可与PD-1以高亲和力结合,抑制其生物活性;MW: 145.8 KD。 | ||||
T9921 | Infliximab
英夫利昔单抗
|
170277-31-3 | 99.70% |
|
Infliximab 是一种与 TNF-α特异性结合的嵌合单克隆 IgG1 抗体,可阻止 TNF-α与 TNFR1和 TNFR2 的相互作用,用于治疗克罗恩病和类风湿性关节炎。 | ||||
T9906 | Ipilimumab
伊匹单抗
|
477202-00-9 | 99.60% |
|
Ipilimumab 是全人类单克隆抗体 IgG1κ,能够抗 CTLA-4。其中CTLA-4是一种由活化的 T 细胞产生的免疫抑制分子。 | ||||
T9911 | Tocilizumab
托珠单抗
|
375823-41-9 | 99.50% |
|
Tocilizumab 是抗人白细胞介素-6 受体 (IL-6R) 的中和抗体,能够阻碍 IL-6 与 IL-6R 的结合,进而抑制经典和反式信号。它可用于研究类风湿性关节炎,对重症 COVID-19 冠状病毒病方面的研究具有显著效果。 | ||||
T9930 | Secukinumab
苏金单抗
|
875356-43-7 | 99.10% |
Secukinumab
|
Secukinumab 是一种完全人源化的单克隆抗 IL-17A 抗体,是一个被美国食品和药物管理局批准用于治疗中度至重度斑块型银屑病的抗体。 | ||||
T9905 | Cetuximab
西妥昔单抗
|
205923-56-4 | 98.60% |
|
Cetuximab 是一种单克隆抗体,是一种表皮生长因子受体(EGFR)抑制剂。它具有高效的抗肿瘤作用,通过 SPR 方法测得其对EGFR 的Kd 值为 0.201 nM。 | ||||
T37535 | Camrelizumab
卡瑞利珠单抗
|
1798286-48-2 | 98.6% |
|
Camrelizumab (SHR-1210) 是一种具有高亲和力且针对 PD-1的人源 IgG4-κ单克隆抗体。Camrelizumab 与 PD-1 的结合亲和力高达 3 nM,对 PD-1/PD-L1具有抑制作用, IC50 为 0.70 nM。Camrelizumab 具有抗肿瘤活性和耐受性,可用于研究包括 NS... |