T3753
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Sinapinic Acid
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Sinapinic acid 是从Hydnophytum formicarumJack. 根中分离到的酚类,是HDAC抑制剂,对ACE-I的活性也有抑制作用。它有抗肿瘤活性,诱导肿瘤细胞凋亡,具有抗氧化、抗糖尿病的作用。
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T3717
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Hinokitiol
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Hinokitiol 是从日本扁柏中分离到的一种挥发油成分,可抑制紫外线 B 诱导的角质形成细胞凋亡,可调节雌激素受体信号传导并抑制人乳腺癌细胞的增殖。它具有抗感染、抗氧化及抗肿瘤等活性。
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T4S0181
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Hinokiflavone
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Hinokiflavone是pre-mRNA剪接活性的新型调节剂,通过抑制剪接体装配来阻止pre-mRNA 底物的剪接,特别是阻止 B complex 的形成。它是SUMO protease蛋白酶抑制剂,能够抑制前哨蛋白特异性蛋白酶 1 的活性。
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TN2516
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1,7-Diepi-8,15-cedranediol
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TN3691
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Communic acid
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Communic acid has antibacterial activity, including against mycobacterial. trans-Communic acid has potential to be utilized as anti-wrinkling agents and cosmetic ingredients, as they suppress UVB-induced MMP-1 expression.
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TN4794
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Pinusolidic acid
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Pinusolidic acid shows a potent inhibitory effect on platelet activating factor (PAF) binding to rabbit platelets (IC50 = 2.3 x 10(-5) M, 7.48 +/- 2.11 micrograms/ml).
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TMA0164
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15-Hydroxydehydroabietic acid
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15-Hydroxydehydroabietic acid exhibits a promising alpha-glucosidase inhibitory activity, it also shows significant antibacterial activities.
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TL0014
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Pinusolide
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Pinusolide is a platelet activating factor ( PAF) antagonist, it may prove of therapeutic value in the treatment of hypotension, it has antileukemic potential, and could be used to treat neurodegenerative diseases. Pinusolide attenuates blockade of insuli
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TN3808
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Dehydroheliobuphthalmin
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Dehydroheliobuphthalmin has significant neuroprotective activities against glutamate- induced neurotoxicity.
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TN3260
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8(14),15-Isopimaradien-3-ol
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ent-8(14),15-pimaradien-3beta-ol (8(14),15-Isopimaradien-3-ol) can induce vascular relaxation. It displays high antibacterial activities (MIC values lower than 10 microg /mL for most pathogens).
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TN3261
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8(14),15-Isopimaradiene-3,18-diol
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TN2639
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15-Isopimarene-8,18-diol
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TN4716
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Oplodiol
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Oplodiol exhibits noteworthy anti-plasmodial activity against Plasmodium falciparum strains. Oplodiol has a stimulative effect on significantly proliferation and differentiation of culture osteoblasts; it also shows moderate cytotoxic effects on the human
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TN2641
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15-Methoxypinusolidic acid
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15-Methoxypinusolidic acid has anti-inflammatory effects, it inhibits LPS-induced iNOS expression and NO production, independent on MAPK and NF-kappaB. 15-Methoxypinusolidic acid suppresses adipocyte differentiation through the inhibition of PPARgamma-dep
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TN2645
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16-Hydroxy-8(17),13-labdadien-15,16-olid-19-oic acid
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16-Hydroxy-8(17),13-labdadien-15,16-olid-19-oic acid may show a strong algicidal activity against Raphidocelis subcapitata.
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