经典已知活性库

Bioactive Compound Library
产品编号 L4000
  库化合物信息   Excel SDF

经典已知活性库是8829个具有生物活性,能引起细胞、组织甚至个体生物学反应的化合物的集合。包括了正在进行临床前研究的药物分子,临床期的药物分子和已经上市的药物。靶点明确,信息全面,非常适合完成药物功能重定位、小分子诱导细胞分化以及机制研究中蛋白靶点确认等科研工作。

由于活性明确,靶点已知,很多科学家会从已知活性库中选择可以用于细胞诱导分化的小分子,通过单一或几个小分子的联合作用,选择出将各种体细胞诱导成为诱导多能干细胞,神经前体细胞,心肌细胞等,甚至还有使用小分子组合在体内完成诱导分化的成功尝试。

为了保证客户的最佳使用效果,我们把已知活性库中需要现配现用的多肽以及其他药物分子以干粉形式提供(设置为PartB),尽可能增加新的药物筛选机会,增加成功筛选到目标分子的几率。

包含L4000已知活性库在内,陶术生物可以提供多达4万种生物活性已知的小分子化合物,可以满足您在各个阶段的科研工作需要,欢迎随时和我们联系。

经典已知活性库
规格 价格/RMB
100 μL * 10 mM (in DMSO) 598294.00
250 μL * 10 mM (in DMSO) 912129.00
1 mg 912129.00
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产品描述

  • 8829个已知活性化合物的集合,可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认;
  • 所有化合物都有相应的靶点信息的描述,靶点信息已知;
  • 是老药新用、细胞诱导靶点筛选的有效工具;
  • 涵盖多个疾病研究领域,如癌症、代谢、免疫和心血管系统等;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • 结构多样,药效显著,可渗透细胞;
  • NMR、HPLC/ LCMS多重检测,保证产品结构准确,纯度高,保障实验顺利进行。

化合物库定制

我们的化合物库可以灵活定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L4000)

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Vasopressin Receptor (11)
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Endothelin Receptor (11)
HIF/HIF Prolyl-Hydroxylase (11)
Hydroxylase (10)
Liver X Receptor (10)
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Kinesin (10)
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Melanocortin Receptor (10)
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Histone Acetyltransferase (8)
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PAI-1 (7)
Monocarboxylate transporter (7)
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IRE1 (6)
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化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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