按潜在通路靶点分类

通过计算机虚拟筛选技术,基于已知活性分子类似物分析和靶点docking分析,并经过药化性质过滤器过滤,最终从160万小分子中精心挑选而出的靶点库。我们既有针对常见靶点类型的靶点库,如GPCR库、NF-κb库,也有针对蛋白-蛋白相互作用(PPI)等特殊靶点的化合物库。陶素生化提供行业内常见的靶点库类型,并可根据客户需求提供专业的化合物库定制服务。

PI3K/Akt/mTOR Focused Library
LF5900 PI3K/Akt/mTOR靶向库
4400 compounds
Nucleic acid ligands
DP4400 核酸配体
9000 compounds
Akt-Targeted Library
DP3200 Akt靶向库
12000 compounds
PRMT Library
DP1800 PRMT靶向库
31000 compounds
ROCK Targeted Library
LF5200 ROCK靶向库
1360 compounds
Aspartic Protease Screening Libraries
LF6300 天冬氨酸蛋白酶筛选库
1400 compounds
Aquaporin Screening Library
LF2100 水通道蛋白筛选库
2000 compounds
CXCR4-Targeted Library
DP4000 CXCR4靶向库
11000 compounds
Phosphatase Inhibitors
DP3100 磷酸酶抑制剂筛选库
15000 compounds
Fibroblast Growth Factor Receptor 1 Tyrosine Kinase Targeted Library
LF4800 FGFR1酪氨酸激酶靶向库
646 compounds
STING Targeted Library
LF6900 STING靶向库
1600 compounds
Matrix Metalloproteinase Focused Library
LF5700 基质金属蛋白酶靶向库
2000 compounds
Cysteine Protease Focused Library
LF6500 半胱氨酸蛋白酶靶向库
3700 compounds
BRD4 targeted library
DP5300 BRD4靶向库
5000 compounds
Lipid Metabolism Library
DD5300 脂质代谢库
9000 compounds
Autophagy-Targeted Library
DP2800 自噬靶向库
17000 compounds
Glucocorticoid receptors Library
DP5100 糖皮质激素受体库
5000 compounds
Allosteric GPCR Library
EN1600 变构GPCR调节剂库
14400 compounds
Type II Kinase Inhibitors Library
DP4900 II型激酶抑制剂库
8000 compounds
Protease Targeted Library
LF6600 蛋白酶靶向库
5700 compounds
Histone Deacetylases (HDAC) Targeted Library
DD5000 HDAC筛选库
9500 compounds
Aurora A Kinase Targeted Library
LF4200 Aurora A激酶靶向库
590 compounds
Hinge Binders Library
EN2600 激酶ATP位点结合剂筛选库
24000 compounds
ERK5 (MAPK7) Kinase Targeted Library
LF4700 ERK5(MAPK7)靶向库
900 compounds
NR-Focused Library
DP6000 核受体靶向库
1700 compounds
Protein-Protein Interaction Library
EN3800 蛋白相互作用库
40640 compounds
Developmental Pathway (Hh/Wnt) Set
DP5800 Hh/Wnt 通路靶向库
2000 compounds
3CLpro Library
DD4200 3CLpro抑制剂筛选库
4792 compounds
Library of Small Molecule Inhibitors of beta-Catenin Signaling
DP4700 beta-Catenin通路靶向库
8000 compounds
Lysine-specific demethylase 4A (KDM4A) Targeted Library
LF5500 KDM4A靶向库
2000 compounds
Aurora B Kinase Targeted Library
LF4300 Aurora B激酶靶向库
1000 compounds
Cyclic Ugi PPI Library
DP4200 Cyclic Ugi PPI库
10000 compounds
Aquaporins Library
EN1900 水通道蛋白库
1348 compounds
Kynurenine Pathway Library
EN3200 犬尿氨酸通路库
12304 compounds
HA2 Library
DP5500 HA2库
4000 compounds
DGK Inhibitors Library
DP9200 DGK抑制剂库
12000 compounds
ALK Tyrosine Kinase Focused Library
LF4100 ALK酪氨酸激酶靶向库
2500 compounds
P24-Targeted Library
DP3600 P24靶向库
12000 compounds
GPCR Library
EN2500 GPCR库
54080 compounds
Kinase Targeted Library by Docking
LF3800 激酶靶向库-基于分子对接
13000 compounds
Adenosine Receptors Targeted Library
DP2400 腺苷受体靶向库
21000 compounds
Kinase Library
EN3100 激酶库
65200 compounds
DNMT-Focused Library
DP1600 DNMT靶向库
38000 compounds
Protein Kinases Inhibitors Library
DP1700 蛋白激酶抑制剂库
38000 compounds
Ligase Focused Screening Library
LF5400 连接酶靶向库
3900 compounds
Calcium Channels Library
DP3900 钙离子通道库
11000 compounds
Epigenetic Screening Libraries
LF2900 表观遗传筛选库
11500 compounds
ATPase Focused Library
LF2200 ATP酶靶向库
8800 compounds
Chelator Focused Library
LF5600 螯合剂靶向库
5700 compounds
PI3K-Targeted Library
DP2900 PI3K靶向库
19000 compounds
Phosphatase Screening Library
LF6100 磷酸酶筛选库
2700 compounds
Lipoxygenase Library
EN3400 脂氧合酶靶向库
1388 compounds
ACE2 Library
DD4300 ACE2抑制剂筛选库
3051 compounds
Vascular Endothelial Growth Factor Receptor Kinase 2 (VGFR-2) Focused Library
LF5300 VEGFR2靶向库
1000 compounds
MDM2 focused Library
DP7690 MDM2靶向库
6500 compounds
Tubulin Library
EN4200 微管靶向库
3452 compounds
Beta 2 Adrenoligands Library
DP2500 β2肾上腺素库
20000 compounds
GP-120 & GP-41 Libraries
DP2600 GP-120 & GP-41库
20000 compounds
Chelators targeting matrix metalloproteinases Library
DD4800 螯合剂靶向基质金属蛋白酶文库
9300 compounds
MDM2-p53 interaction inhibitors Library
DP2300 MDM2-p53相互作用抑制剂库
23000 compounds
DNA-encoded (DEL) Reagents and Building Blocks
LF2800 DNA编码化合物库
70000 compounds
GPCR Target Platform Library
DP1500 GPCR靶向库
40000 compounds
JAK/STAT pathway modulators
EN3000 JAK/STAT通路调节剂库
1392 compounds
DNA Library
EN2200 DNA稳定蛋白靶向库
5530 compounds
SH2 Library
DP3700 SH2库
12000 compounds
Lipid GPCR Library
EN3300 脂GPCR靶向库
5440 compounds
Polymerase Library
DP5200 聚合酶靶向库
5500 compounds
Allosteric Kinase Library
EN1700 变构激酶库
4800 compounds
Serine Protease Screening Libraries
LF6700 丝氨酸蛋白酶筛选库
5400 compounds
3-Phosphoinositide-Dependent Kinase-1 (PDK1) Targeted Library
LF4000 PDK1靶向库
760 compounds
Sodium Ion Channel Library
EN4100 钠离子通道库
5440 compounds
Hsp90-Targeted Library
DP3500 Hsp90靶向库
13000 compounds
Epigenetics Library
EN2300 表观遗传靶向库
9352 compounds
Targeted Diversity Library
DP1400 靶点多样性库
45000 compounds
MEF2-HDAC (class II) Modulators Library
DP5000 MEF2-HDAC(II类)调节剂库
6000 compounds
Proline Kinase Library
DP5900 脯氨酸激酶库
2000 compounds
Cyclin-dependent Kinases 2 (CDK2) Focused Library
LF4600 CDK2靶向库
400 compounds
Peptidomimetic Compound Library
LF6000 拟肽化合物库
5800 compounds
NFkb-Regulators Library
DP4500 NFkb调节剂库
9000 compounds
SH2 PTB Focused Library
DP4600 SH2 PTB靶向库
7000 compounds
IDO Targeted Library
EN2700 IDO靶向库
5502 compounds
MCL1 Targeted Library Selection
DD4600 MCL1靶向库
12000 compounds
c-AMP Dependent Protein Kinase (PKA) Targeted Library
LF4400 PKA靶向库
730 compounds
G9a-Inhibitors Library
DP3400 G9a抑制剂库
13000 compounds
N-methyl-D-aspartate (NMDA) Receptor Screening Library
LF3500 NMDA受体筛选库
1000 compounds
PTPN-targeted Library
DD5200 非受体型蛋白酪氨酸磷酸酶靶向库
33000 compounds
Aurora A-B Kinases Library
DP4300 Aurora A-B激酶库
10000 compounds
Cysteine Targeted Covalent Library
DD5700 半胱氨酸靶向共价库
39301 compounds
Kinase Screening Library
LF3700 激酶筛选库
3000 compounds
Glutamate Receptor Focused Library
LF3000 谷氨酸受体靶向库
4600 compounds
Focused Epigenetics Set
DP1900 表观遗传筛选库
30431 compounds
Kinase Focused Library
LF3600 激酶靶向库
32000 compounds
RNA Library
EN3900 RNA靶向库
15520 compounds
Alpha-Helix Mimetics Library
DP3580 α螺旋模拟物库
24737 compounds
Phosphatidylinositol 3-Kinase (PI3K) Targeted Library
LF5100 PI3K靶向库
939 compounds
Cytochrome Inhibitor Library
LF2400 细胞色素酶抑制剂库
1900 compounds
Ion Channels Focused Library
DD4900 离子通道筛选库
26000 compounds
RNA-Protein Interaction Inhibitors Library
DD5600 RNA-蛋白相互作用抑制剂筛选库
2111 compounds
Hormone-related Focused Library
LF3400 激素相关靶向库
750 compounds
INTEGRIN Receptors Targeted library
DP5700 整合素受体靶向库
2000 compounds
Arginase Targeted Library
DD4700 精氨酸酶靶向库
2000 compounds
DNA and RNA Polymerase Screening Libraries
LF2700 DNA与RNA聚合酶筛选库
18234 compounds
Hedgehog Pathway Library
DP4100 Hedgehog通路靶向库
11000 compounds
GPCR Targeted Library by Receptor-based Approach
LF3200 GPCR靶向库-基于受体
8500 compounds
Recognition Elements PPI Library
DP2000 识别元件PPI库
26000 compounds
Deubiquitinase Screening Libraries
LF2600 去泛素化酶筛选库
3300 compounds
Phosphodiesterase (PDE10) Targeted Library
LF6200 PDE10靶向库
1450 compounds
Molecular Chaperones Library
EN3500 分子伴侣靶向库
2468 compounds
RNA Focused Library
LF6800 RNA靶向库
4400 compounds
Serine Hydrolase Library
EN4000 丝氨酸水解酶库
12560 compounds
Degrader Building Blocks for Targeted Protein Degradation
LF2500 靶向蛋白质降解的降解砌块库
1700 compounds
PPI CDI Library
DP1000 PPI计算机辅助药物设计库
230000 compounds
Eccentric PPI Library
DP3300 Eccentric PPI库
13000 compounds
Monoamine Transporters Library
DP4800 单胺转运蛋白库
8000 compounds
Ligand-Gated Ion Channels Library
DP5600 配体门离子通道库
4000 compounds
c-Met (HGFR) Kinase Targeted Library
LF4500 c-Met(HGFR)激酶靶向库
1100 compounds
PPI Helix Turn 3D-Mimetics Library
DP2200 PPI螺旋转角3D模拟物库
74000 compounds
Tyrosine Kinase Screening Library
LF3900 酪氨酸激酶筛选库
5700 compounds
PLpro Library
DD4100 抗PLpro抑制剂筛选库
6442 compounds
KRAS-Targeted Library
DP3800 KRAS靶向库
11000 compounds
Apoptotic Library
DP1200 凋亡靶向库
54000 compounds
Caspase Targeted Library
LF6400 Caspase靶向库
2800 compounds
Nuclear Receptor Screening Libraries
LF5800 核受体筛选库
11000 compounds
Calcium Ion Channel Library
EN2100 钙离子通道库
10560 compounds
Allosteric Kinases Inhibitors Library
DP2100 变构激酶抑制剂库
26000 compounds
Helicase Focused Library
LF3300 预制解旋酶靶向库
2745 compounds
GPCR Focused Screening Library by 2D Similarity
LF3100 GPCR靶向库-基于2D相似性
7600 compounds
BACE Library
EN2000 BACE靶向库
7171 compounds
Janus Kinase (JAK) Targeted Library
LF4900 JAK靶向库
600 compounds
Veterinary Focused Library
LF7000 兽药靶向库
238 compounds
GSK3β-Targeted Library
DP5400 GSK3β靶向库
5000 compounds
p38 Mitogen-activated Protein (MAP) Kinase Focused Library
LF5000 p38 MAP激酶靶向库
1100 compounds
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