首页 GPCR/G Protein 5-HT Receptor Opiranserin
Opiranserin
编号 T16399    
CAS 1441000-45-8     分子式 C21H34N2O5     分子量 394.51
靶点: 5-HT2A Receptor; GlyT2; rP2X3;
Opiranserin is a development as an injectable agent for the treatment of postoperative pain. Opiranserin is a non-opioid and non-NSAID analgesic candidate and is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A) (IC50s: 0.86 and 1.3 μM, respectively). Opiranserin displays antagonistic activity on rP2X3 (IC50=0.87 μM).
选择批次  
纯度 98.00%
规格 库存 单价 数量
1 mg 待询 1300.00
5 mg 待询 2927.00
10 mg 待询 4388.00
25 mg 待询 7898.00
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生物活性

产品描述

Opiranserin is a development as an injectable agent for the treatment of postoperative pain. Opiranserin is a non-opioid and non-NSAID analgesic candidate and is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A) (IC50s: 0.86 and 1.3 μM, respectively). Opiranserin displays antagonistic activity on rP2X3 (IC50=0.87 μM).

靶点活性

5-HT2A Receptor,1.3 μM

GlyT2,0.86 μM

rP2X3,0.87 μM

体外活性

体内活性

化学信息

分子量

394.51

分子式

C21H34N2O5

CAS

1441000-45-8

溶解度

( < 1 mg/ml refers to the product slightly soluble or insoluble )

储存条件

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

备注

For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

配制溶液

1 mg 5 mg 10 mg
1 mM 2.535 ml 12.674 ml 25.348 ml
5 mM 0.507 ml 2.535 ml 5.07 ml
10 mM 0.253 ml 1.267 ml 2.535 ml
50 mM 0.051 ml 0.253 ml 0.507 ml
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