Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Medrysone (6α-Methyl-11β-hydroxyprogesterone) 是局部合成的糖皮质激素,具有代谢、抗炎和抗过敏特性,有潜力用于眼科的眼炎症研究。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
25 mg | ¥ 148 | 现货 | ||
50 mg | ¥ 256 | 现货 | ||
100 mg | ¥ 490 | 现货 | ||
200 mg | ¥ 960 | 现货 |
产品描述 | Medrysone (6α-Methyl-11β-hydroxyprogesterone) is a topical, synthetic glucocorticoid with metabolic, anti-inflammatory and anti-allergic properties. Medrysone exerts its effect by interacting with specific intracellular glucocorticoid receptors and subsequently binds to DNA to modify gene expression. This results in an induction of the synthesis of certain anti-inflammatory proteins while inhibiting the synthesis of certain inflammatory mediators. Consequently, an overall reduction in chronic inflammation and autoimmune reactions is accomplished. |
别名 | Gimeracil, 6α-Methyl-11β-hydroxyprogesterone, 6A-甲基-11B-羟孕酮, 甲羟松 |
分子量 | 344.49 |
分子式 | C22H32O3 |
CAS No. | 2668-66-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 200.3 mM
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 2.9028 mL | 14.5142 mL | 29.0284 mL | 72.571 mL |
5 mM | 0.5806 mL | 2.9028 mL | 5.8057 mL | 14.5142 mL | |
10 mM | 0.2903 mL | 1.4514 mL | 2.9028 mL | 7.2571 mL | |
20 mM | 0.1451 mL | 0.7257 mL | 1.4514 mL | 3.6286 mL | |
50 mM | 0.0581 mL | 0.2903 mL | 0.5806 mL | 1.4514 mL | |
100 mM | 0.029 mL | 0.1451 mL | 0.2903 mL | 0.7257 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
Medrysone 2668-66-8 Endocrinology/Hormones Others Glucocorticoid Receptor inhibit Gimeracil 6α-Methyl-11β-hydroxyprogesterone 6A-甲基-11B-羟孕酮 6a-Methyl-11b-hydroxyprogesterone 6alpha-Methyl-11beta-hydroxyprogesterone HMS Inhibitor 甲羟松 inhibitor