首页 GPCR/G Protein Histamine Receptor Bavisant
Bavisant
编号 TQ0046     别名: JNJ-31001074
CAS 929622-08-2     分子式 C19H27N3O2     分子量 329.44
靶点:
Bavisant (JNJ-31001074) is a selective and orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition.
选择批次  
纯度 98.00%
规格 库存 单价 数量
10 mg 待询 3200.00
25 mg 待询 6100.00
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生物活性

产品描述

Bavisant (JNJ-31001074) is a selective and orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition.

靶点活性

体外活性

体内活性

Mean change from baseline in the total ADHD-RS-IV score at day 42 (primary efficacy endpoint) was -8.8 in the placebo group versus -9.3, -11.2 and -12.2 in the bavisant 1 mg/day, 3 mg/day and 10 mg/day groups, respectively; the change in the 10 mg/day group was not statistically superior to placebo, and hence statistical comparisons of the 1 mg/day and 3 mg/day groups with placebo based on a step-down closed testing procedure were not performed.

化学信息

分子量

329.44

分子式

C19H27N3O2

CAS

929622-08-2

溶解度

DMSO: Soluble

( < 1 mg/ml refers to the product slightly soluble or insoluble )

储存条件

store at -80°C

备注

For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

配制溶液

1 mg 5 mg 10 mg
1 mM 3.035 ml 15.177 ml 30.355 ml
5 mM 0.607 ml 3.035 ml 6.071 ml
10 mM 0.304 ml 1.518 ml 3.035 ml
50 mM 0.061 ml 0.304 ml 0.607 ml
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