首页 GPCR/G Protein Histamine Receptor Astemizole
Astemizole
编号 T1278     别名: Histaminos, Paralergin, Laridal
CAS 68844-77-9     分子式 C28H31FN4O     分子量 458.58
靶点: H1 receptor; Potassium Channel;
Astemizole is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to related agents. It is a long-acting, non-sedative antihistaminic used in the treatment of seasonal allergic rhinitis, asthma, allergic conjunctivitis, and chronic idiopathic urticaria.
选择批次  
规格 库存 单价 数量
5 mg 上海现货 575.00
10 mg 上海现货 920.00
50 mg 上海现货 2690.00
1 mL * 10 mM (in DMSO) 上海现货 630.00
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生物活性

产品描述

Astemizole is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to related agents. It is a long-acting, non-sedative antihistaminic used in the treatment of seasonal allergic rhinitis, asthma, allergic conjunctivitis, and chronic idiopathic urticaria.

靶点活性

H1 receptor,

Potassium Channel,

体外活性

体内活性

化学信息

分子量

458.58

分子式

C28H31FN4O

CAS

68844-77-9

溶解度

DMSO: 10 mM

( < 1 mg/ml refers to the product slightly soluble or insoluble )

储存条件

store at -80°C

备注

For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

配制溶液

1 mg 5 mg 10 mg
1 mM 2.181 ml 10.903 ml 21.806 ml
5 mM 0.436 ml 2.181 ml 4.361 ml
10 mM 0.218 ml 1.09 ml 2.181 ml
50 mM 0.044 ml 0.218 ml 0.436 ml
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