Alcaftadine
编号 T2533
别名:
R89674,
Lastacaft
CAS 147084-10-4
分子式
C19H21N3O
分子量
307.39
靶点:
H1 receptor;
H2 receptor;
H4 receptor;
Alcaftadine is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.


生物活性
产品描述 |
Alcaftadine is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis. |
靶点活性 |
H1 receptor,8.5(pKi) H2 receptor,7.2(pKi) H4 receptor,5.8(pKi) |
体外活性 |
|
体内活性 |
化学信息
分子量 |
307.39 |
分子式 |
C19H21N3O |
CAS |
147084-10-4 |
溶解度 |
DMSO: 28 mg/mL (91.09 mM) Water: <1 mg/mL Ethanol: 61 mg/mL (198.44 mM) ( < 1 mg/ml refers to the product slightly soluble or insoluble ) |
储存条件 |
store at -80°C |
备注 |
For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months. |
配制溶液
1 mg | 5 mg | 10 mg | |
1 mM | 3.253 ml | 16.266 ml | 32.532 ml |
5 mM | 0.651 ml | 3.253 ml | 6.506 ml |
10 mM | 0.325 ml | 1.627 ml | 3.253 ml |
50 mM | 0.065 ml | 0.325 ml | 0.651 ml |