首页 Metabolism NADPH Acetohexamide
Acetohexamide
编号 T0816     别名: Dymelor, Acetohexamid, Gamadiabet
CAS 968-81-0     分子式 C15H20N2O4S     分子量 324.4
靶点: NADPH; Potassium Channel;
Acetohexamide is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity. It inhibits sulfonylurea receptor 1 (SUR1) linked to the inwardly rectifying potassium channel (KIR6.2) with Ki values of 22.9 and 14.2 µM in HEK293 cells transfected with the human receptor and in rat brain, respectively. Acetohexamide is metabolized in the liver to its active metabolite hydroxyhexamide.
选择批次  
规格 库存 单价 数量
50 mg 上海现货 236.00
100 mg 上海现货 425.00
200 mg 上海现货 512.00
1 mL * 10 mM (in DMSO) 上海现货 462.00
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生物活性

产品描述

Acetohexamide is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity. It inhibits sulfonylurea receptor 1 (SUR1) linked to the inwardly rectifying potassium channel (KIR6.2) with Ki values of 22.9 and 14.2 µM in HEK293 cells transfected with the human receptor and in rat brain, respectively. Acetohexamide is metabolized in the liver to its active metabolite hydroxyhexamide.

靶点活性

NADPH,

Potassium Channel,

体外活性

体内活性

化学信息

分子量

324.4

分子式

C15H20N2O4S

CAS

968-81-0

溶解度

DMSO: >10 mM

( < 1 mg/ml refers to the product slightly soluble or insoluble )

储存条件

0-4℃ for short term (days to weeks), or -20℃ for long term (months).

备注

For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

配制溶液

1 mg 5 mg 10 mg
1 mM 3.083 ml 15.413 ml 30.826 ml
5 mM 0.617 ml 3.083 ml 6.165 ml
10 mM 0.308 ml 1.541 ml 3.083 ml
50 mM 0.062 ml 0.308 ml 0.617 ml
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