AMPAR antagonist/activator kit 包含AMPA 受体拮抗剂/激活剂,AMPA 受体介导中枢神经系统快速兴奋性突触传递,诱发和维持长时程的增强和抑制,参与调节学习、记忆活动,参与谷氨酸介导的兴奋性损伤、tau 蛋白的异常磷酸化及神经原纤维缠结的形成等。AMPA 受体数目和功能异常可能导致阿尔兹海默病的发生。TargetMol 为您提供32种精选AMPA 受体拮抗剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0051 | Urethane | 51-79-6 | 89.09 | 10mM | AChR; Antibacterial; Chloride channel; GABA Receptor; GluR; NMDAR; Parasite |
T0333 | Aniracetam | 72432-10-1 | 219.24 | 10mM | 5-HT Receptor; AChR; Dopamine Receptor; GluR; iGluR |
T0426 | Piracetam | 7491-74-9 | 142.16 | 10mM | GluR; iGluR |
T1884 | CX516 | 154235-83-3 | 241.29 | 10mM | GluR; iGluR |
T3379 | Decanoic Acid | 334-48-5 | 172.26 | 10mM | GluR; iGluR |
T3473 | (S)-ATPO | 252930-37-3 | 322.25 | 10mM | GluR |
T3957 | Farampator | 211735-76-1 | 231.26 | 10mM | GluR; iGluR |
T4113 | NBQX | 118876-58-7 | 336.28 | 10mM | GluR; iGluR |
T7304 | DNQX | 2379-57-9 | 252.14 | 10mM | GluR; iGluR |
T7178 | CNQX | 115066-14-3 | 232.15 | 10mM | GluR; iGluR |
T7579 | 1-BCP | 34023-62-6 | 233.26 | 10mM | GluR; iGluR |
T7580 | CX546 | 215923-54-9 | 247.29 | 10mM | Autophagy; iGluR |
T7706 | LY-404187 | 211311-95-4 | 342.46 | 10mM | GluR; iGluR |
T7823 | IDRA-21 | 22503-72-6 | 232.68 | 10mM | GluR |
T8435 | YM90K | 154164-30-4 | 309.66 | 10mM | GluR; iGluR |
T8458 | CNQX disodium | 479347-85-8 | 276.12 | 10mM | iGluR |
T8779 | HBT1 | 489408-02-8 | 386.39 | 10mM | GluR |
T16402 | Org-26576 | 1026791-61-6 | 204.23 | 10mM | GluR; iGluR |
TP2111L | TAT-GluA2 3Y acetate(1404188-93-7 free base) | TP2111L | 2634.02 | 10mM | GluR |
T15369L | gamma-DGG acetate(6729-55-1 free base) | T15369L | 264.23 | 10mM | GluR |
TP1944L1 | pep2-SVKI acetate | TP1944L1 | 1344.51 | 10mM | GluR |
T50094 | DL-Willardiine | 19772-76-0 | 199.16 | 10mM | Others |
T16977 | Talampanel | 161832-65-1 | 337.37 | 10mM | Apoptosis; GluR |
T12406 | PEPA | 141286-78-4 | 402.44 | 10mM | iGluR |
T19698 | CX614 | 191744-13-5 | 247.25 | 10mM | GluR |
T17179 | Tulrampator | 1038984-31-4 | 380.37 | 10mM | iGluR |
T15623 | JNJ-61432059 | 2035814-50-5 | 443.47 | 10mM | iGluR |
T13480 | (S)-(-)-5-Fluorowillardiine | 140187-23-1 | 217.15 | 10mM | iGluR |
T20571 | cis-PDA | 46026-75-9 | 173.17 | 10mM | GluR; iGluR; NMDAR |
T37734 | AMPA receptor modulator-2 | 2034181-36-5 | 404.29 | 10mM | GluR |
T15820 | Mibampator | 375345-95-2 | 438.6 | 10mM | iGluR |
T27951 | LY392098 | 211311-39-6 | 335.44 | 10mM | iGluR;GluR |